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(4R)-4-[(1S,2S,5R,7R,10R,11S,14R,15R,16S)-5,16-dihydroxy-2,15-dimethyltetracyclo[8.7.0.02,7.011,15]heptadecan-14-yl]-1-[4-(pyridin-2-yl)piperazin-1-yl]pentan-1-one
2-[(4-methyl-2-oxo-2H-chromen-7-yl)oxy]-N-(3-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}propyl)acetamide
2-[(7S)-2,8-dioxo-3,9-diazatricyclo[8.4.0.03,7]tetradeca-1(10),11,13-trien-9-yl]-N-(5-methyl-1,3-thiazol-2-yl)acetamide
2-(6,7-dimethoxy-2-methyl-4-oxo-3,4-dihydroquinazolin-3-yl)-N-(oxan-4-ylmethyl)acetamide
N-(2,2-dimethyloxan-4-yl)-2-[2-(4-methoxyphenyl)ethyl]-1-oxo-1,2-dihydroisoquinoline-4-carboxamide
(4R)-N-benzyl-4-[(1S,2S,5R,7R,10R,11S,14R,15R,16S)-5,16-dihydroxy-2,15-dimethyltetracyclo[8.7.0.02,7.011,15]heptadecan-14-yl]-N-methylpentanamide
(4R)-N-[3-(methylsulfanyl)phenyl]-4-[(1S,2S,5R,7S,9R,10R,11S,14R,15R,16S)-5,9,16-trihydroxy-2,15-dimethyltetracyclo[8.7.0.02,7.011,15]heptadecan-14-yl]pentanamide
methyl 2-{2-[(7S)-2,8-dioxo-3,9-diazatricyclo[8.4.0.03,7]tetradeca-1(10),11,13-trien-9-yl]acetamido}-5-methyl-1,3-thiazole-4-carboxylate
N-[2-(5-methoxy-1H-indol-1-yl)ethyl]-4-phenyloxane-4-carboxamide
N-[1-(2-methoxyethyl)-1H-indol-4-yl]-3-(2-methoxyphenyl)propanamide
(4R)-N-(4-phenylbutan-2-yl)-4-[(1S,2S,5R,7S,9R,10R,11S,14R,15R,16S)-5,9,16-trihydroxy-2,15-dimethyltetracyclo[8.7.0.02,7.011,15]heptadecan-14-yl]pentanamide
2-[1-(propan-2-yl)-1H-indol-3-yl]-N-(3,4,5-trimethoxyphenyl)acetamide
3-[(2H-1,3-benzodioxol-5-yl)carbamoyl]-2-[(4-methyl-1,4-diazepan-1-yl)methyl]propanoic acid
(4R)-4-[(1S,2S,5R,7R,10R,11S,14R,15R,16S)-5,16-dihydroxy-2,15-dimethyltetracyclo[8.7.0.02,7.011,15]heptadecan-14-yl]-N-[1-(2-methoxyethyl)-1H-indol-4-yl]pentanamide
ethyl 3-(2,3-dimethoxyphenyl)-3-(4-hydroxy-6-methyl-2-oxo-1,2-dihydropyridin-3-yl)propanoate
2-[(7S)-2,8-dioxo-3,9-diazatricyclo[8.4.0.03,7]tetradeca-1(10),11,13-trien-9-yl]-N-[2-(4-fluorobenzenesulfonyl)ethyl]acetamide
2-[(7S)-2,8-dioxo-3,9-diazatricyclo[8.4.0.03,7]tetradeca-1(10),11,13-trien-9-yl]-N-[2-(4-methoxyphenyl)ethyl]acetamide
N-[(3,4-dimethoxyphenyl)methyl]-2-[(7S)-2,8-dioxo-3,9-diazatricyclo[8.4.0.03,7]tetradeca-1(10),11,13-trien-9-yl]acetamide
2-[(7S)-2,8-dioxo-3,9-diazatricyclo[8.4.0.03,7]tetradeca-1(10),11,13-trien-9-yl]-N-(oxolan-2-ylmethyl)acetamide
1,6,7-trimethyl-8-(propan-2-yl)-1H,2H,3H,4H,8H-imidazo[1,2-g]purine-2,4-dione
2-[(7S)-2,8-dioxo-3,9-diazatricyclo[8.4.0.03,7]tetradeca-1(10),11,13-trien-9-yl]-N-[5-(propan-2-yl)-1,3,4-thiadiazol-2-yl]acetamide
(4R)-4-[(1S,2S,5R,7R,10R,11S,14R,15R,16S)-5,16-dihydroxy-2,15-dimethyltetracyclo[8.7.0.02,7.011,15]heptadecan-14-yl]-N-[5-(methoxymethyl)-1,3,4-thiadiazol-2-yl]pentanamide
3-methyl-N-{2-[(4-methyl-2-oxo-2H-chromen-7-yl)oxy]pyridin-3-yl}butanamide
2-[(4,8-dimethylquinazolin-2-yl)amino]-6-(propan-2-yl)-3,4-dihydropyrimidin-4-one
(4R)-N-(2-phenylethyl)-4-[(1S,2S,5R,7S,9R,10R,11S,14R,15R,16S)-5,9,16-trihydroxy-2,15-dimethyltetracyclo[8.7.0.02,7.011,15]heptadecan-14-yl]pentanamide
N-{[4-(4-methoxyphenyl)oxan-4-yl]methyl}-2-methyl-5-(propan-2-yl)-1,3-thiazole-4-carboxamide
2-[(7S)-2,8-dioxo-3,9-diazatricyclo[8.4.0.03,7]tetradeca-1(10),11,13-trien-9-yl]-N-(6-methylpyridin-2-yl)acetamide
4-[3-(1H-indol-1-yl)propanamido]benzamide
N-[1-(2-methoxyethyl)-1H-indol-4-yl]-1-methyl-2-oxo-1,2-dihydroquinoline-4-carboxamide
methyl 4-(4-phenyloxane-4-amido)benzoate
2-(2,2-dimethyl-3-oxopiperazin-1-yl)-N-[2-(5-methoxy-1H-indol-1-yl)ethyl]acetamide
N-(1,3-benzothiazol-2-yl)-2-[(3S)-2,5-dioxo-3-(propan-2-yl)-2,3,4,5-tetrahydro-1H-1,4-benzodiazepin-1-yl]acetamide
N-(1H-indol-6-yl)-2-(5-methyl-1H-indol-1-yl)acetamide
N-(6-methoxypyridin-3-yl)-2-[1-(propan-2-yl)-1H-indol-3-yl]acetamide
(3S)-3-(propan-2-yl)-2,3,4,5-tetrahydro-1H-1,4-benzodiazepine-2,5-dione
2-[(7S)-2,8-dioxo-3,9-diazatricyclo[8.4.0.03,7]tetradeca-1(10),11,13-trien-9-yl]-N-(2-hydroxyphenyl)acetamide
2-[(2S)-1-[(4aS,8aS)-4a-hydroxy-decahydroisoquinolin-2-yl]-3-methyl-1-oxobutan-2-yl]-2,3-dihydro-1H-isoindol-1-one
3-{8-methoxy-1H,2H,3H,4H,5H-pyrido[4,3-b]indole-2-carbonyl}-1-methyl-1H-indole
ethyl 2-{2-[(7S)-2,8-dioxo-3,9-diazatricyclo[8.4.0.03,7]tetradeca-1(10),11,13-trien-9-yl]acetamido}-4-methyl-1,3-thiazole-5-carboxylate
(4R)-4-[(1S,2S,5R,7R,10R,11S,14R,15R,16S)-5,16-dihydroxy-2,15-dimethyltetracyclo[8.7.0.02,7.011,15]heptadecan-14-yl]-1-(6,7-dimethoxy-1,2,3,4-tetrahydroisoquinolin-2-yl)pentan-1-one
2-[(3R)-2,5-dioxo-2,3,4,5-tetrahydro-1H-1,4-benzodiazepin-3-yl]-N-[2-(4-hydroxyphenyl)ethyl]acetamide
(2R)-3-phenyl-N-(pyridin-3-ylmethyl)-2-{[(1r,4r)-4-(propan-2-yl)cyclohexyl]formamido}propanamide
N-[2-(1H-indol-3-yl)ethyl]-3-(4-methyl-3-oxo-3,4-dihydroquinoxalin-2-yl)propanamide
N-(oxan-4-ylmethyl)-2-({12-oxo-6H,7H,8H,9H,10H,12H-azepino[2,1-b]quinazolin-2-yl}oxy)acetamide
ethyl 3-(4-hydroxy-2-oxo-1,2-dihydroquinolin-3-yl)-3-(7-methoxy-2-oxo-1,2-dihydroquinolin-3-yl)propanoate
5-methoxy-N-[1-(2-methoxyethyl)-1H-indol-4-yl]-1-methyl-4-oxo-1,4-dihydropyridine-2-carboxamide
N-{2-[(4-methyl-2-oxo-2H-chromen-7-yl)oxy]pyridin-3-yl}acetamide
methyl 5-(propan-2-yl)-2-[(4R)-4-[(1S,2S,5R,7S,9R,10R,11S,14R,15R,16S)-5,9,16-trihydroxy-2,15-dimethyltetracyclo[8.7.0.02,7.011,15]heptadecan-14-yl]pentanamido]-1,3-thiazole-4-carboxylate
N-cyclooctyl-2-[(7S)-2,8-dioxo-3,9-diazatricyclo[8.4.0.03,7]tetradeca-1(10),11,13-trien-9-yl]acetamide
N-[2-(5-chloro-1H-indol-3-yl)ethyl]-1-methyl-2-oxo-1,2-dihydroquinoline-4-carboxamide