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4-[(4aS,8aS)-4a-hydroxy-decahydroisoquinoline-2-carbonyl]-2-(propan-2-yl)-1,2-dihydroisoquinolin-1-one
2-(6,7-dimethoxy-2-methyl-4-oxo-3,4-dihydroquinazolin-3-yl)-N-(2,2-dimethyloxan-4-yl)acetamide
N-[2-(4-methoxyphenyl)ethyl]-2-[(3S)-3-methyl-2,5-dioxo-2,3,4,5-tetrahydro-1H-1,4-benzodiazepin-1-yl]acetamide
N-(1H-indol-4-yl)-2-(4-methoxyphenyl)acetamide
(4R)-4-[(1S,2S,5R,7R,10R,11S,14R,15R,16S)-5,16-dihydroxy-2,15-dimethyltetracyclo[8.7.0.02,7.011,15]heptadecan-14-yl]-N-(1-methyl-1H-indol-4-yl)pentanamide
2-[({[(2-methylpropyl)carbamoyl]methyl}carbamoyl)methyl]benzoic acid
3-(4-chloro-1H-indol-1-yl)-N-(1H-indol-4-yl)propanamide
ethyl 3-(4-hydroxy-2-oxo-1,2-dihydroquinolin-3-yl)-5-methylhexanoate
(4R)-4-[(1S,2S,5R,7R,10R,11S,14R,15R,16S)-5,16-dihydroxy-2,15-dimethyltetracyclo[8.7.0.02,7.011,15]heptadecan-14-yl]-N-(pyridin-4-ylmethyl)pentanamide
N-[2-(1H-indol-3-yl)ethyl]-2-(3-methyl-2-oxo-1,2-dihydroquinoxalin-1-yl)acetamide
(2R)-N-(oxan-4-ylmethyl)-3-phenyl-2-{[(1r,4r)-4-(propan-2-yl)cyclohexyl]formamido}propanamide
N-[(4-methoxyphenyl)methyl]-3-(3-oxo-3,4-dihydroquinoxalin-2-yl)propanamide
(4R)-N-[2-(2-methoxyphenyl)ethyl]-4-[(1S,2S,5R,7S,9R,10R,11S,14R,15R,16S)-5,9,16-trihydroxy-2,15-dimethyltetracyclo[8.7.0.02,7.011,15]heptadecan-14-yl]pentanamide
2-(azepan-1-ylmethyl)-5-hydroxy-4H-pyran-4-one
2-{[(4-carbamoylphenyl)carbamoyl]methyl}benzoic acid
N-[2-(1H-imidazol-4-yl)ethyl]-1-oxo-1,2-dihydroisoquinoline-4-carboxamide
methyl (2S)-2-[(3-methyl-4-oxo-2-phenyl-4H-chromen-8-yl)formamido]propanoate
2-[3-(1H-1,3-benzodiazol-2-yl)propanamido]-4,5-dimethoxybenzoic acid
(4R)-1-[4-(2-methoxyphenyl)piperazin-1-yl]-4-[(1S,2S,5R,7S,9R,10R,11S,14R,15R,16S)-5,9,16-trihydroxy-2,15-dimethyltetracyclo[8.7.0.02,7.011,15]heptadecan-14-yl]pentan-1-one
ethyl 4-[(4R)-4-[(1S,2S,5R,7S,9R,10R,11S,14R,15R,16S)-5,9,16-trihydroxy-2,15-dimethyltetracyclo[8.7.0.02,7.011,15]heptadecan-14-yl]pentanoyl]piperazine-1-carboxylate
2-[(1,6-dimethyl-4-oxo-1,4-dihydropyridin-3-yl)oxy]-N-(1H-indol-4-yl)acetamide
2-[(7S)-2,8-dioxo-3,9-diazatricyclo[8.4.0.03,7]tetradeca-1(10),11,13-trien-9-yl]-N-(3,4,5-trifluorophenyl)acetamide
N-(4-tert-butyl-1,3-thiazol-2-yl)-2-[(7S)-2,8-dioxo-3,9-diazatricyclo[8.4.0.03,7]tetradeca-1(10),11,13-trien-9-yl]acetamide
2-[(4-methyl-2-oxo-2H-chromen-7-yl)oxy]-N-{[1,2,4]triazolo[4,3-a]pyridin-3-ylmethyl}acetamide
3-[3-(6,7-dimethoxy-1,2,3,4-tetrahydroisoquinolin-2-yl)-3-oxopropyl]-1,2-dihydroquinoxalin-2-one
3-[(2-carbamoylphenyl)carbamoyl]-2-(pyrrolidin-1-ylmethyl)propanoic acid
2-[(7S)-2,8-dioxo-3,9-diazatricyclo[8.4.0.03,7]tetradeca-1(10),11,13-trien-9-yl]-N-(furan-2-ylmethyl)acetamide
3-methyl-N-{6-[(4-methyl-2-oxo-2H-chromen-7-yl)oxy]pyridin-3-yl}butanamide
N-(1H-indol-6-yl)-2-[(3S)-3-methyl-2,5-dioxo-2,3,4,5-tetrahydro-1H-1,4-benzodiazepin-1-yl]acetamide
ethyl 2-(2-{2-[(7S)-2,8-dioxo-3,9-diazatricyclo[8.4.0.03,7]tetradeca-1(10),11,13-trien-9-yl]acetamido}-1,3-thiazol-4-yl)acetate
N-(2,4-dimethoxyphenyl)-5-(1,2-dithiolan-3-yl)pentanamide
2-(7-methoxy-4-methyl-2-oxo-2H-chromen-3-yl)-N-[2-(4-methyl-1H-indol-1-yl)ethyl]acetamide
N-[2-(1H-indol-3-yl)ethyl]-2-(5-methyl-1H-indol-1-yl)acetamide
(4R)-N-(1,3-benzothiazol-2-yl)-4-[(1S,2S,5R,7S,9R,10R,11S,14R,15R,16S)-5,9,16-trihydroxy-2,15-dimethyltetracyclo[8.7.0.02,7.011,15]heptadecan-14-yl]pentanamide
2-[(3,4-dimethyl-2-oxo-2H-chromen-7-yl)oxy]-N-(3-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}propyl)acetamide
2-(5-{7,7-dimethyl-2,5-dioxo-1H,2H,3H,4H,5H,7H-furo[3,4-b]pyridin-4-yl}-2-methoxyphenoxy)acetamide
2-[(3R)-2,5-dioxo-2,3,4,5-tetrahydro-1H-1,4-benzodiazepin-3-yl]-N-[5-(2-methylpropyl)-1H-1,2,4-triazol-3-yl]acetamide
(4R)-4-[(1S,2S,5R,7R,10R,11S,14R,15R,16S)-5,16-dihydroxy-2,15-dimethyltetracyclo[8.7.0.02,7.011,15]heptadecan-14-yl]-N-(6-methoxy-1,3-benzothiazol-2-yl)pentanamide
(4R)-N-(2-methoxyphenyl)-4-[(1S,2S,5R,7S,9R,10R,11S,14R,15R,16S)-5,9,16-trihydroxy-2,15-dimethyltetracyclo[8.7.0.02,7.011,15]heptadecan-14-yl]pentanamide
(4R)-4-[(1S,2S,5R,7R,10R,11S,14R,15R,16S)-5,16-dihydroxy-2,15-dimethyltetracyclo[8.7.0.02,7.011,15]heptadecan-14-yl]-N-[(2-methoxyphenyl)methyl]pentanamide
6-hydroxy-2-[4-(methylsulfanyl)phenyl]-4H-chromen-4-one
2-hydroxy-5-(3-{3H-imidazo[4,5-b]pyridin-2-yl}propanamido)benzoic acid
methyl 2-(2-{7,7-dimethyl-2,5-dioxo-1H,2H,3H,4H,5H,7H-furo[3,4-b]pyridin-4-yl}-6-methoxyphenoxy)acetate
methyl 2-[(4R)-4-[(1S,2S,5R,7R,10R,11S,14R,15R,16S)-5,16-dihydroxy-2,15-dimethyltetracyclo[8.7.0.02,7.011,15]heptadecan-14-yl]pentanamido]-5-(propan-2-yl)-1,3-thiazole-4-carboxylate
(4R)-4-[(1S,2S,5R,7R,10R,11S,14R,15R,16S)-5,16-dihydroxy-2,15-dimethyltetracyclo[8.7.0.02,7.011,15]heptadecan-14-yl]-N-[4-(pyridin-3-yl)-1,3-thiazol-2-yl]pentanamide
(4R)-N-benzyl-4-[(1S,2S,5R,7R,10R,11S,14R,15R,16S)-5,16-dihydroxy-2,15-dimethyltetracyclo[8.7.0.02,7.011,15]heptadecan-14-yl]pentanamide
N-(dimethyl-1,3-thiazol-2-yl)-2-[(7S)-2,8-dioxo-3,9-diazatricyclo[8.4.0.03,7]tetradeca-1(10),11,13-trien-9-yl]acetamide
4-{3-[1-(propan-2-yl)-1H-indol-3-yl]propanamido}benzamide
ethyl 3-(4-hydroxy-2-oxo-1,2-dihydroquinolin-3-yl)-3-(3-hydroxy-4-methoxyphenyl)propanoate
5-(1,2-dithiolan-3-yl)-N-(5-methyl-1,3-thiazol-2-yl)pentanamide