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(1-{[methyl({[2-(propan-2-yl)-1,3-oxazol-4-yl]methyl})amino]methyl}cyclopentyl)methanol
3-[(4-methyl-6-{[1-(pyrazin-2-yl)propan-2-yl]amino}pyrimidin-2-yl)amino]phenol
2-{2-[(3-methoxyphenyl)methyl]morpholin-4-yl}-N-(thiophen-2-ylmethyl)acetamide
N-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-(pyrrolidine-1-sulfonyl)benzamide
1-{5H,6H-benzo[h]quinazolin-2-yl}-N-(1-hydroxy-2-methylpropan-2-yl)-5-methyl-1H-pyrazole-4-carboxamide
2-{4-[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl]-1-(2-methylpropyl)piperazin-2-yl}ethan-1-ol
3-[(2-methoxyethyl)sulfamoyl]-5-{1H-pyrazolo[3,4-b]pyridin-1-yl}benzoic acid
7-(2-cyclohexylethyl)-2-[(6-methylpyridin-2-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one
(2S)-2-amino-N-[1-(4-fluorophenyl)-4-(pyridin-3-yloxy)-1H-indazol-3-yl]butanamide
(3aS,6aR)-5-(2-amino-6-methylpyrimidin-4-yl)-3-[3-(morpholin-4-yl)propyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
3-[1-(2H-1,3-benzodioxol-4-ylmethyl)piperidin-3-yl]-N-[(5-methylfuran-2-yl)methyl]propanamide
1-[(2-{[2-(2,2-dimethyloxan-4-yl)-1H-imidazol-1-yl]methyl}phenyl)methyl]pyrrolidin-2-one
3-{2-[bis(propan-2-yl)carbamoyl]phenyl}-4-methoxy-N-methylbenzamide
1-(2-cyclopropyl-4-methylpyrimidine-5-carbonyl)-4-(1H-imidazol-1-yl)piperidine-4-carboxylic acid
3-{1-[3-(2-hydroxyphenyl)propanoyl]piperidin-4-yl}-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
(4S,4aS,8aR)-1-(3-methyl-1-propyl-1H-pyrazole-4-carbonyl)-4-phenyl-decahydroquinolin-4-ol
4-[(dimethylamino)methyl]-1-{[2-(propylsulfanyl)pyrimidin-5-yl]methyl}azepan-4-ol
{[3-(3,4-dimethylphenyl)-1H-pyrazol-4-yl]methyl}(ethyl)(pyridin-4-ylmethyl)amine
1-(1-acetylpiperidin-4-yl)-N-(pyridin-3-ylmethyl)piperidine-3-carboxamide
dimethyl[1-(1-{[2-(methylsulfanyl)phenyl]methyl}piperidin-4-yl)ethyl]amine
5-[(dimethyl-1H-1,2,4-triazol-1-yl)methyl]-3-[1-(4-methylphenyl)cyclopentyl]-1,2,4-oxadiazole
3-{8-[3-(5-methyl-1H-pyrazol-1-yl)propanoyl]-2-oxo-1-oxa-3,8-diazaspiro[4.5]decan-3-yl}propanoic acid
2-methyl-6-[1-(2-methyl-1,3-benzothiazol-6-yl)-1H-1,2,4-triazol-5-yl]-2H,3H,5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridin-3-one
1-[4-hydroxy-4-(hydroxymethyl)piperidin-1-yl]-2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)ethan-1-one
1-(propan-2-yl)-N-[2-(1H-1,2,4-triazol-5-ylsulfanyl)ethyl]piperidine-4-carboxamide
(3R,4R)-1-(4-aminopyrimidin-2-yl)-4-(4-methylpiperazin-1-yl)piperidin-3-ol
N-({5-[(4-cyanophenyl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)cyclobutanecarboxamide
3-{[4-(5-oxo-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-3-yl)piperidin-1-yl]methyl}benzonitrile
(3aS,6aR)-5-(2-aminoacetyl)-3-[2-(3-chlorophenyl)ethyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
1-[(2-butyl-1H-imidazol-4-yl)methyl]-3-(3-chlorobenzoyl)piperidine
1-methyl-2-(morpholin-4-yl)-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-1H-1,3-benzodiazole-5-carboxamide
4-methyl-N,N-bis(1,3-oxazol-4-ylmethyl)-3-phenyl-1H-pyrazole-5-carboxamide
N4-[1-(3,4-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-N1,N1-dimethylpiperidine-1,4-dicarboxamide
N-{[1-(cyclohex-1-ene-1-carbonyl)piperidin-3-yl]methyl}-4-methoxybenzene-1-sulfonamide
[(3R,4S)-4-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-1-[(4-methyl-1H-imidazol-5-yl)methyl]pyrrolidin-3-yl]methanol
N-[(3R,4S)-1-acetyl-4-cyclopropylpyrrolidin-3-yl]-7-fluoro-2-oxo-1,2-dihydroquinoline-4-carboxamide
2-(2-methoxyphenyl)-5-{[3-(pyrimidin-4-yl)piperidin-1-yl]methyl}pyrimidine
1-(6-fluoro-4-methylquinazolin-2-yl)-N-[2-(3-fluorophenyl)ethyl]azepan-4-amine
(2R)-2-[3-(4-chlorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl]pyrrolidine
2-(adamantan-1-yl)-4-hydroxy-N-methyl-N-(oxan-2-ylmethyl)pyrimidine-5-carboxamide
7-cyclopentyl-2-(3-propyl-1H-pyrazole-4-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
3-[3-(hydroxymethyl)-3-(3-methylbut-2-en-1-yl)piperidine-1-carbonyl]-1H,2H,5H,6H,7H-cyclopenta[b]pyridin-2-one
methyl 3-[({5-[(cyclohexylmethyl)sulfanyl]-4-(4-fluorophenyl)-4H-1,2,4-triazol-3-yl}methyl)sulfamoyl]thiophene-2-carboxylate
N-cyclopropyl-N-{[2-(3,4-dimethoxyphenyl)-7-methylquinolin-3-yl]methyl}propanamide
(4aS,8aR)-6-[3-(6-oxo-1,4,5,6-tetrahydropyridazin-3-yl)propanoyl]-1-propyl-decahydro-1,6-naphthyridin-2-one
1-methyl-4-({5-[2-(1H-pyrrol-1-yl)ethyl]-1,2,4-oxadiazol-3-yl}methyl)piperazine
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-4-oxo-4H-chromene-2-carboxamide
2-(4-{1-[3-(5-methylfuran-2-yl)butyl]piperidin-4-yl}piperazin-1-yl)ethan-1-ol
3-(oxolan-3-yl)-5-(4-phenylbutyl)-1,2,4-oxadiazole
8-{[(3S,4R)-3,4-dihydroxy-4-methylpiperidin-1-yl]methyl}-3-oxatricyclo[7.3.1.05,13]trideca-1(12),5(13),6,8,10-pentaen-2-one