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(4-{[methyl(4-methylpyrimidin-2-yl)amino]methyl}oxan-4-yl)methanol
N2-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl]-5-fluoro-N4,N4-dimethylpyrimidine-2,4-diamine
2-benzyl-N-methyl-N-{[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]methyl}-1,3-thiazole-4-carboxamide
1-{2-oxo-2-[(2R,3R,6R)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]ethyl}piperidin-2-one
2-{1-[(4-ethoxyphenyl)methyl]-4-(1H-pyrazol-3-ylmethyl)piperazin-2-yl}ethan-1-ol
N-[(dimethyl-1,2-oxazol-4-yl)methyl]-1-(thiophene-2-carbonyl)piperidin-4-amine
2-(1-ethyl-1H-pyrazole-4-carbonyl)-7-[(3-methoxyphenyl)methyl]-2,7-diazaspiro[4.5]decane
4-{[3-(methanesulfonylmethyl)piperidin-1-yl]methyl}benzonitrile
(1S,5R)-3-[3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
6-[4-(3-phenylpropyl)-1,4-diazepan-1-yl]pyrimidin-4-amine
1-(2H-1,3-benzodioxol-5-ylmethyl)-4-{[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}piperazine
2-benzyl-9-[(4-methyl-1H-imidazol-2-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
2-(adamantan-1-yl)-N-[3-hydroxy-2-(thiophen-2-ylmethyl)propyl]acetamide
1-methyl-4-[(1S,5R)-6-(3-methylbut-2-en-1-yl)-7-oxo-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]-1,2-dihydroquinolin-2-one
1-(3,4-dihydro-2H-1-benzopyran-3-carbonyl)-4-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidine
N-(2,1,3-benzothiadiazol-5-ylmethyl)-N-methyl-5-(1H-pyrazol-1-ylmethyl)furan-2-carboxamide
2-amino-4-(1H-indol-5-yl)-5-methyl-6-(1-methyl-1H-pyrazol-4-yl)pyridine-3-carbonitrile
[(2S,6S)-4-(3,5-dimethyl-1-benzofuran-2-carbonyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(9),10,12-trien-6-yl]methanol
(2S,4S)-4-amino-N-methyl-1-{[5-(pyridin-2-yl)thiophen-2-yl]sulfonyl}pyrrolidine-2-carboxamide
2-{3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidin-1-yl}-3-(pyrrolidin-1-yl)pyrazine
4-[2-(1-methyl-1H-imidazol-2-yl)benzoyl]morpholine
N-(2,4-difluorophenyl)-3-{[(furan-3-ylmethyl)(methyl)amino]methyl}benzamide
3-({[4-(benzyloxy)phenyl]methyl}amino)-1-methylpyrrolidin-2-one
{[5-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}[(6-methoxypyridin-3-yl)methyl]methylamine
N-methyl-3-(4-methyl-1,3-thiazol-5-yl)-N-[(4-methyl-1H-imidazol-2-yl)methyl]propanamide
(2,2-dimethyl-3-{2-[1-(piperidin-4-yl)-1H-1,2,3-triazol-4-yl]-1H-imidazol-1-yl}propyl)dimethylamine
N-[1-(3,4-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-3-(propan-2-yl)-1,2-oxazole-5-carboxamide
1-{[(3R,4R)-4-(hydroxymethyl)-1-(5-phenyl-1,3,4-thiadiazol-2-yl)pyrrolidin-3-yl]methyl}piperidin-4-ol
2-{4-[(4-hydroxy-3-methylphenyl)methyl]piperazin-1-yl}quinoline-4-carboxylic acid
2-cyclohexyl-1-{4-[2-(oxolan-2-yl)-3H-imidazo[4,5-b]pyridin-3-yl]piperidin-1-yl}ethan-1-one
3-{1-[(5-acetylthiophen-3-yl)methyl]piperidin-3-yl}-N-(5-chloro-2-methoxyphenyl)propanamide
3-[(7-{[4-(benzyloxy)piperidin-1-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)methyl]phenol
1-(5-{3-[2-(methylsulfanyl)benzoyl]piperidine-1-carbonyl}thiophen-2-yl)ethan-1-one
5-{[(3-methoxyphenyl)methyl]amino}-N,N-dimethyl-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
5-fluoro-N-(3-hydroxypropyl)-2-methoxy-N-[(5-methylthiophen-2-yl)methyl]benzamide
2-benzyl-8-(pyridin-4-ylmethyl)-2,8-diazaspiro[4.5]decan-3-one
5-{1-[2-(2-chlorophenyl)ethyl]-1H-imidazol-2-yl}-N,N-dimethylpyrimidin-2-amine
9-[(1-ethyl-1H-pyrazol-3-yl)methyl]-2-[(5-methylpyrazin-2-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
N-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-5-oxo-1-[4-(propan-2-yl)phenyl]pyrrolidine-3-carboxamide
(3R,5S)-5-[(2,3-dihydro-1H-inden-5-yloxy)methyl]-N-[2-(morpholin-4-yl)ethyl]-1-(naphthalen-2-ylmethyl)piperidine-3-carboxamide
1-{[2-(2-ethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-2-(3-methoxyphenyl)piperidine
{2-[3-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)phenoxy]ethyl}(methyl)amine
4-(methoxymethyl)-6-{4-[4-(2-methylphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}pyrimidine
5-(4-chloro-2-methoxyphenoxymethyl)-N-[(2S)-oxolan-2-ylmethyl]-1,2-oxazole-3-carboxamide
(2-{4-[4-(3-methylphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}-2-oxoethyl)urea
9-(6-cyclopropylpyrimidin-4-yl)-2-(2-hydroxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
1-[5-(3-fluorophenyl)-4-(4-methylphenyl)pyrimidin-2-yl]-1,4-diazepan-5-one
3-cyclopentyl-1-{3-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}propan-1-one
2-({cyclopropyl[(1-methyl-1H-pyrazol-4-yl)methyl]amino}methyl)-6-methylquinolin-4-ol
2-(dimethylamino)-7-(3-methyl-1H-pyrazole-5-carbonyl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one