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ethyl 3-benzyl-1-(oxan-4-yl)piperidine-3-carboxylate
N-[(1-methylpyrrolidin-3-yl)methyl]-4H,5H,6H,7H,8H-cyclohepta[b]thiophene-2-carboxamide
(3E)-N-(1-hydroxybutan-2-yl)-N-(thiophen-3-ylmethyl)pent-3-enamide
1-(carbamoylmethyl)-N-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)piperidine-4-carboxamide
N-(1-{1-[4-(4-chlorophenyl)butanoyl]piperidin-4-yl}-1H-pyrazol-5-yl)cyclopropanecarboxamide
1'-({4-[(dimethylamino)methyl]thiophen-2-yl}methyl)-1-methyl-1,2-dihydrospiro[indole-3,3'-piperidine]-2-one
1-methyl-1'-{2-methylimidazo[1,2-a]pyridine-6-carbonyl}-1,2-dihydrospiro[indole-3,3'-piperidine]-2-one
(1S,5R)-3-[2-(2-ethyl-1H-imidazol-1-yl)acetyl]-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-[(5-ethyl-1,3,4-thiadiazol-2-yl)methyl]-1-(2-methyl-6-propylpyrimidin-4-yl)piperidin-4-amine
methyl 3-{1-[(3-methyl-1,2,4-thiadiazol-5-yl)carbamoyl]piperidin-4-yl}propanoate
3-(morpholine-4-sulfonyl)-5-(1H-pyrazol-1-yl)benzoic acid
(2R,3R,6R)-3-(2,3-difluorophenyl)-N,N-dimethyl-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carboxamide
N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl}-N-(oxolan-2-ylmethyl)pyridine-4-carboxamide
N,1-diethyl-3-(2-methylpropyl)-N-[2-(morpholin-4-yl)ethyl]-1H-pyrazole-5-carboxamide
1-[1-methyl-3-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-2-{[1,2,4]triazolo[1,5-a]pyrimidin-6-yl}ethan-1-one
N-[2-(2-chlorophenyl)ethyl]-4-{[(1,1-dioxo-1λ6-thiolan-3-yl)methyl]amino}-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
3-[(1-butanoylpyrrolidin-3-yl)methyl]benzoic acid
2-hydroxy-4-methyl-N-{[2-(4-methyl-1,4-diazepan-1-yl)pyridin-3-yl]methyl}benzamide
2-(4-{[(1S,5R)-3-(2,3-dihydro-1H-inden-2-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}-3-methyl-1H-pyrazol-1-yl)ethan-1-ol
3-[3-(4-methoxyphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-1H-indazole
(2S)-2-amino-N-({2-[4-(pyridin-2-yl)piperazin-1-yl]pyridin-3-yl}methyl)propanamide
1-[(1-{[4-(furan-2-yl)phenyl]methyl}piperidin-4-yl)methyl]-4-methylpiperazine
1-(4-{[(2,1,3-benzoxadiazol-5-ylmethyl)amino]methyl}-2-methoxyphenoxy)-3-(diethylamino)propan-2-ol
N-[(2-fluorophenyl)methyl]-N-(2-hydroxyethyl)-4,5,6-trimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
2-(4-acetylphenoxy)-1-{3-[(3,4-dimethylphenyl)amino]piperidin-1-yl}ethan-1-one
N-{[7-(3-cyclohexylpropanoyl)-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-3-ethyl-1-methyl-1H-pyrazole-5-carboxamide
1-[(3R,4R)-3-hydroxy-4-(hydroxymethyl)piperidin-1-yl]-5-phenylpentane-1,5-dione
3-(3,4-dimethoxyphenyl)-5-[(2-methoxyethyl)sulfamoyl]benzoic acid
(2S,4S)-N-methyl-1-(naphthalen-1-ylmethyl)-4-({[2-(trifluoromethyl)phenyl]methyl}amino)pyrrolidine-2-carboxamide
1-[4-(methoxymethyl)-5-methyl-1,2-oxazole-3-carbonyl]-N-(pyridin-3-ylmethyl)piperazine-2-carboxamide
4-[4-(oxolane-2-carbonyl)piperazin-1-yl]-6-(pyrrolidin-1-yl)pyrimidin-2-amine
[(3R,4R)-4-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-1-(5-propyl-1,3,4-thiadiazol-2-yl)pyrrolidin-3-yl]methanol
5-chloro-N-[(1,3-dimethyl-1H-pyrazol-5-yl)methyl]-4,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
3-[2-(5-amino-1,3,4-thiadiazol-2-yl)propan-2-yl]-1-[3-(5-ethyl-4H-1,2,4-triazol-3-yl)phenyl]urea
1-[4-(4-{[2-(4-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazin-1-yl)phenyl]ethan-1-one
2-(2,1,3-benzoxadiazol-5-ylmethyl)-7-[(2-fluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
(2S,4S)-4-(2,5-dimethylfuran-3-amido)-N-ethyl-1-(1H-imidazol-4-ylmethyl)pyrrolidine-2-carboxamide
N-[2-({3-[3-(propan-2-yloxy)benzoyl]piperidin-1-yl}methyl)quinolin-5-yl]acetamide
1-[5-(2-methoxyacetyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl]-3-(2-methyl-1H-imidazol-1-yl)propan-1-one
N-(2-{1-[(4-ethylphenyl)methyl]-1H-1,2,4-triazol-5-yl}ethyl)acetamide
2-[(2-chloro-4-fluorophenyl)methyl]-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
6-[(3R,4R)-3-{[(2-hydroxyethyl)(methyl)amino]methyl}-4-(hydroxymethyl)pyrrolidin-1-yl]pyridine-2-carbonitrile
{[2-cyclopropylmethanesulfonyl-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}(methyl)[(3-methyl-1,2-oxazol-5-yl)methyl]amine
6-{4-[1-(dimethylamino)ethyl]phenyl}-N,N-dimethylpyrazin-2-amine
N-ethyl-5-({3-[2-(2-methylphenyl)pyridin-4-yl]pyrrolidin-1-yl}methyl)pyrimidin-2-amine
4-(6-cyclopropylpyrimidin-4-yl)-1-phenylpiperazin-2-one
N-(2-hydroxyethyl)-N-[(1-methyl-1H-imidazol-2-yl)methyl]-2-[1-(propan-2-yl)piperidin-4-yl]acetamide
1-(1H-1,2,3-benzotriazol-4-yl)-3-{2-[(trifluoromethyl)sulfanyl]ethyl}urea
2-(2-chloro-4-fluorophenoxymethyl)-N-[1-(1-methyl-1H-pyrazol-4-yl)ethyl]-1,3-oxazole-4-carboxamide
[1-(3-fluoropyridin-2-yl)-4-(2-phenylethyl)piperidin-4-yl]methanol