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(3aS,6aS)-2-cyclobutanecarbonyl-5-{[4-(methylcarbamoyl)phenyl]methyl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-methyl-1-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-1,2-dihydroquinoxalin-2-one
2-(5-{3-[2-(4-fluorophenyl)ethyl]piperidine-1-carbonyl}-1H-1,3-benzodiazol-1-yl)ethan-1-ol
3-{2-[(1S,5R)-3-[(dimethyl-1,2-oxazol-4-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-oxoethyl}-1,3-oxazolidin-2-one
N-methyl-3-{4-[1-(piperidin-1-yl)ethyl]phenyl}pyrazin-2-amine
4-[5-(3-fluoro-5-methylphenyl)-4-phenyl-1H-imidazol-1-yl]-N,N-dimethylbutanamide
1-{5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-4-(5-methylpyridin-2-yl)piperidin-4-ol
3-{[4-(2-hydroxyethyl)piperazin-1-yl]sulfonyl}-N-(oxolan-3-yl)benzamide
2-{5-[(2-oxo-1,3-oxazolidin-3-yl)methyl]-3-(pyridin-4-yl)-1H-1,2,4-triazol-1-yl}benzoic acid
2-[3-({methyl[(5-methylfuran-2-yl)methyl]amino}methyl)phenyl]-6-(pyridin-4-yl)-3,4-dihydropyrimidin-4-one
N-[(4-methoxypyridin-2-yl)methyl]-4-sulfamoylbenzamide
N-{[1-(1H-pyrazol-3-ylmethyl)piperidin-3-yl]methyl}quinoline-8-sulfonamide
3-(2-{3-[2-(2,6-difluorophenyl)ethyl]piperidin-1-yl}-2-oxoethyl)-1,3-oxazolidin-2-one
3-{1-[7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carbonyl]pyrrolidin-2-yl}pyridine
N-ethyl-N-[2-(3-methoxyphenoxy)ethyl]-2-(methylamino)pyridine-3-carboxamide
3-ethoxy-1-{3-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}propan-1-one
4-[2-(dimethyl-1,2-oxazol-4-yl)pyrrolidine-1-carbonyl]-7-fluoro-2-methylquinoline
1-methyl-N-[(4-methylphenyl)(pyridin-4-yl)methyl]-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
N-[(3S,4R)-1-[1-ethyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]-4-(propan-2-yl)pyrrolidin-3-yl]acetamide
1-cyclopentyl-3-methyl-5-(thiophen-2-yl)-1H,4H-pyrazolo[3,4-d]imidazole
5-(azepane-1-carbonyl)-1-(2-methylpropyl)-4-oxo-N-(thiophen-2-ylmethyl)-1,4-dihydropyridine-3-carboxamide
(5S)-5-({[(4-methoxy-2,3,6-trimethylphenyl)methyl](pyridin-4-ylmethyl)amino}methyl)pyrrolidin-2-one
4-cyclobutyl-6-methyl-N-[2-(1-methylpyrrolidin-2-yl)ethyl]pyrimidin-2-amine
N-[(3S,4R)-1-(5-chloro-3-fluoropyridin-2-yl)-4-(4-methoxyphenyl)pyrrolidin-3-yl]acetamide
N-[(2S)-1-methoxy-3-phenylpropan-2-yl]-2-oxo-6-(propan-2-yl)-1,2-dihydropyridine-3-carboxamide
(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)({[8-methyl-2-(piperidine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl})amine
N-benzyl-3-{1-[(4-methoxyphenyl)methyl]piperidin-4-yl}-N-methylpropanamide
2-(2-amino-4,6-dimethylpyrimidin-5-yl)-1-[4-(pyridin-3-ylmethyl)-1,4-diazepan-1-yl]ethan-1-one
N-[2-(ethanesulfonyl)ethyl]-7-methylpyrazolo[1,5-a]pyrimidine-6-carboxamide
2-[4-(4-cyclopentyl-1H-1,2,3-triazol-1-yl)piperidin-1-yl]-6-methylpyridine-3-carboxamide
N-(2-ethoxyphenyl)-3-[(2S)-4-methyl-2-(propan-2-yl)piperazin-1-yl]propanamide
1-(2-methoxyphenyl)-4-{1-[1-(propan-2-yl)piperidin-4-yl]piperidin-3-yl}piperazine
6-[(5-cyclopentyl-1,2,4-oxadiazol-3-yl)methyl]-5,6-dihydro-1,6-naphthyridin-5-one
methyl 8-[2-(1H-imidazol-4-yl)ethyl]-9-oxo-2,8-diazaspiro[5.5]undecane-2-carboxylate
7-(3-chlorophenyl)-9-methoxy-4-[(2-methoxyphenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-(1,4-dioxan-2-ylmethyl)-N-methyl-1-[4-(2-methyl-1,3-thiazol-4-yl)phenyl]piperidin-4-amine
5-cyclopropanecarbonyl-3-(4-phenylphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
N,N,5-trimethyl-2-{[1-(thiomorpholin-4-yl)hex-5-en-2-yl]oxy}pyrimidin-4-amine
1-methyl-4-[7-(oxolane-3-carbonyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]-1,4-diazepane
3-{[(4-fluorophenyl)methyl]sulfanyl}-1-[4-(3-methylpyridin-2-yl)piperazin-1-yl]propan-1-one
2-{1-[(4-methoxy-3-methylphenyl)methyl]-3-oxopiperazin-2-yl}-N-methylacetamide
5-(azepane-1-carbonyl)-N-[2-(1H-indol-3-yl)ethyl]-1-(2-methylpropyl)-4-oxo-1,4-dihydropyridine-3-carboxamide
1-[2-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)pyrimidin-4-yl]piperidin-4-ol
3-[5-(3-methyl-2-phenylbutanoyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]propanoic acid
N-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-N-methyl-1-(2-methylphenyl)piperidin-4-amine
3-{[(6-fluoro-4-hydroxyquinolin-2-yl)methyl](2-hydroxyethyl)amino}-1λ6-thiolane-1,1-dione
1-[2-(2,6-dimethoxyphenoxy)ethyl]-3-methoxy-1,2-dihydropyridin-2-one
{[2-(methoxymethyl)pyrimidin-5-yl]methyl}(methyl)(quinolin-5-ylmethyl)amine
6-[1-(3-methylpiperidine-3-carbonyl)piperidin-4-yl]pyrimidin-4-ol
1-(3-{[(4-fluorophenyl)methyl]amino}phenyl)pyrrolidin-2-one