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{[5-(2,3-dihydro-1-benzothiophene-2-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}(ethyl)methylamine
1-[(2-butyl-1H-imidazol-4-yl)methyl]-4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazine
4-{3-[3-(4-fluorophenyl)oxolan-3-yl]-1,2,4-oxadiazol-5-yl}-1-(propan-2-yl)piperidine
N-[2-(6-oxo-3-phenyl-1,6-dihydropyridazin-1-yl)ethyl]-5-(propan-2-yl)-1,2-oxazole-3-carboxamide
N-[3-(4-methoxyphenyl)propyl]-6-{[(1r,4r)-4-hydroxycyclohexyl]amino}pyridine-3-carboxamide
4-(1-cyclopropyl-6-oxopiperidine-3-carbonyl)-1-[(3,5-dimethylphenyl)methyl]piperazin-2-one
N-[(2-aminopyrimidin-5-yl)methyl]-N-methyl-3-(3-phenyl-1,2,4-oxadiazol-5-yl)propanamide
(3S,4R)-4-(2H-1,3-benzodioxol-5-yl)-1-(1-methyl-1H-pyrrole-2-carbonyl)pyrrolidine-3-carboxylic acid
N-(2-hydroxy-3-methoxypropyl)-N-methyl-2-[(propan-2-yl)amino]pyrimidine-5-carboxamide
3-[({[2-(2-methylphenoxy)pyridin-3-yl]methyl}amino)methyl]phenol
N-(3,5-dichlorophenyl)-3-(methanesulfonylmethyl)piperidine-1-carboxamide
6-[(diethylamino)methyl]-N-(isoquinolin-5-yl)pyrazolo[1,5-a]pyrimidine-3-carboxamide
(3S,4R)-4-(2,3-dimethoxyphenyl)-1-[2-(2-oxopyrrolidin-1-yl)acetyl]pyrrolidine-3-carboxylic acid
1-[1-(5-chlorothiophene-2-carbonyl)piperidin-4-yl]-N-cyclopropylpiperidine-3-carboxamide
2-(3,5-dimethyl-1H-pyrazol-4-yl)-2-[(2,7,8-trimethylquinolin-4-yl)formamido]acetic acid
N-cyclohexyl-4-{[1-(1H-imidazol-1-yl)propan-2-yl]amino}piperidine-1-carboxamide
(4aR,7aS)-1-[2-(dimethylamino)acetyl]-4-(2-propoxyacetyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-(4-{4-[(4aS,8aR)-decahydroisoquinoline-2-carbonyl]-2-methoxyphenoxy}piperidin-1-yl)ethan-1-one
N-(1-butyl-1H-1,2,3,4-tetrazol-5-yl)-3-(2-methylphenyl)piperidine-1-carboxamide
N-[(8-methoxyquinolin-5-yl)methyl]-N,2-dimethyl-2,8-diazaspiro[4.5]decane-3-carboxamide
N7-[1-(cyclopropylmethyl)-1H-pyrazol-5-yl]-2,N3,N3-trimethyl-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-3,7-dicarboxamide
N-(4-{1-[(2-methoxyphenyl)methyl]-1H-imidazol-2-yl}phenyl)acetamide
1-[(3R,4S)-3-amino-4-propylpyrrolidin-1-yl]-3-(4-methyl-1,3-thiazol-5-yl)propan-1-one
N,2,5-trimethyl-N-[(5-methyl-1H-1,3-benzodiazol-2-yl)methyl]pyrazolo[1,5-a]pyrimidin-7-amine
2-(2,6-dioxo-1,3-diazinan-1-yl)-N-methyl-N-{[3-(trifluoromethyl)phenyl]methyl}acetamide
4-{4-[(methylsulfanyl)methyl]piperidin-1-yl}-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaene
2-(2-amino-4,6-dimethylpyrimidin-5-yl)-1-(6-hydroxy-1,4-oxazepan-4-yl)ethan-1-one
ethyl 4-[4-(4-amino-5-cyanopyrimidin-2-yl)piperazin-1-yl]piperidine-1-carboxylate
5-butyl-1-(4-chlorophenyl)-4-(2-hydroxyacetyl)piperazin-2-one
9-[2-(3-fluorophenyl)acetyl]-2-(2-methoxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-(5-carbamoyl-2-methylphenyl)-4-[(3S,4R)-4-hydroxyoxolan-3-yl]-1,4-diazepane-1-carboxamide
1-{2-[4-amino-6-(benzylamino)-1,3,5-triazin-2-yl]phenyl}ethan-1-one
[(3R,4R)-4-(azepan-1-ylmethyl)-1-[4-(trifluoromethyl)pyrimidin-2-yl]pyrrolidin-3-yl]methanol
5-(2-butyl-2,5-dihydro-1H-pyrrole-1-carbonyl)-3-(2-methylpropyl)-1,2-oxazole
1-[3-(5-methylfuran-2-yl)butyl]-4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazine
2-{4-[4-ethyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}pyrazine
3-[2-(6-methoxynaphthalen-2-yl)morpholine-4-carbonyl]-2-methylphenol
8-{[4-methoxy-3-(methoxymethyl)phenyl]methyl}-1-oxa-8-azaspiro[4.6]undecane
N,8-dimethyl-3-{[methyl(prop-2-en-1-yl)amino]methyl}-N-(2-phenylethyl)imidazo[1,2-a]pyridine-2-carboxamide
2-(4-methyl-1-oxo-1,2-dihydrophthalazin-2-yl)-N-[1-(3-methylpyridin-2-yl)propyl]acetamide
methyl (2S)-2-phenyl-2-({1-[4-(pyrazine-2-amido)phenyl]piperidin-4-yl}amino)acetate
N-{2-ethyl-4-[2-(pyridin-3-yl)-1H-imidazol-1-yl]phenyl}acetamide
11-[(2-methoxyethyl)amino]-4-[(4-methylphenyl)methyl]-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
2-[(3,5-difluorophenyl)methyl]-8-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-2,8-diazaspiro[4.5]decan-3-one
5-(morpholin-4-yl)-2-[3-oxo-3-(pyrrolidin-1-yl)propyl]-2,3-dihydropyridazin-3-one
1-[4-(4-fluorophenyl)-4-hydroxypiperidin-1-yl]-2-[2-(propan-2-yl)-1H-imidazol-1-yl]propan-1-one
methyl({4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}){[3-(1H-1,2,3,4-tetrazol-5-yl)phenyl]methyl}amine
1-benzyl-8-[(5-ethylfuran-2-yl)methyl]-3-(2-methoxyethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-(3,5-dimethyl-1-benzofuran-2-carbonyl)-2-(2-methoxyphenyl)pyrrolidine
N4-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-2,4-diamine