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N-[(2-ethyl-3,5-dimethyl-1H-indol-7-yl)methyl]-2-(pyrrolidin-1-yl)acetamide
2-(2-aminoethyl)-N-[2-(pyridin-3-yloxy)phenyl]morpholine-4-carboxamide
3-(6-fluoropyridin-3-yl)-1-methyl-1-[1-(4-methylpyridin-2-yl)propan-2-yl]urea
1-[2-(cyclohexylmethyl)morpholin-4-yl]-4-(1H-pyrazol-4-yl)butan-1-one
ethyl 3-[(3-chlorophenyl)methyl]-1-[3-(4-methyl-1,3-thiazol-5-yl)propanoyl]piperidine-3-carboxylate
N-[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)ethyl]-3-(4,5,6,7-tetrahydro-2H-indazol-3-yl)propanamide
3-[(3R,7S,8aS)-3-(hydroxymethyl)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(3,4-dimethylphenyl)urea
(2S,4R)-4-(dimethylamino)-1-(9H-fluorene-9-carbonyl)pyrrolidine-2-carboxylic acid
methyl (2S)-1-{5-[3-(2-fluorophenyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}pyrrolidine-2-carboxylate
N-[2-(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)ethyl]-1-(propan-2-yl)-1H-pyrazole-4-carboxamide
propyl 2-methyl-3-oxo-4-phenyl-2,9-diazaspiro[5.5]undecane-9-carboxylate
2-(1,4-dimethylpiperazin-2-yl)-N-{[2-(2-fluorophenyl)-3-methyl-1H-indol-5-yl]methyl}acetamide
1-(2-aminoethyl)-N-(2-methoxyethyl)-N-(naphthalen-1-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
[(3R,4R)-1-cyclobutanecarbonyl-4-{[(2-methoxyethyl)(methyl)amino]methyl}pyrrolidin-3-yl]methanol
N-(1-{2-[cyclohexyl(methyl)amino]-4-methylpyrimidin-5-yl}ethyl)pent-4-enamide
2-(2,5-dihydro-1H-pyrrole-1-carbonyl)-3,4,7-trimethyl-1H-indole
methyl 2-(tert-butylsulfamoyl)-6-{[4-(methylsulfanyl)phenyl]methyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
8-(4,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carbonyl)-3-methyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-[(3S,4R)-4-propyl-1-{[6-(trifluoromethyl)pyridin-3-yl]methyl}pyrrolidin-3-yl]methanesulfonamide
N,4-dimethyl-2-(propan-2-yl)-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}pyrimidine-5-carboxamide
4-{3-[(3R,4R)-4-ethyl-3,4-dihydroxypiperidin-1-yl]propoxy}benzamide
2-[methyl(piperidin-4-yl)amino]-1-[3-(2-methylphenoxymethyl)piperidin-1-yl]ethan-1-one
3-[3-(1H-1,3-benzodiazol-5-yl)-1,2,4-oxadiazol-5-yl]-N,N-dimethylpiperidine-1-carboxamide
(3aS,6aS)-2-(ethanesulfonyl)-5-[(2-ethylpyrimidin-4-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
[1-({1-[(trimethylpyrazin-2-yl)methyl]piperidin-3-yl}methyl)-1H-1,2,3-triazol-4-yl]methanamine
3-(azetidine-1-sulfonyl)-N-{[1-(ethoxymethyl)cyclopropyl]methyl}benzamide
2-[4-(2-methoxyphenoxy)piperidin-1-yl]-1,3-thiazole-4-carboxamide
(3S,4R)-1-{[3-(morpholin-4-yl)phenyl]methyl}-4-(pyridin-3-yl)pyrrolidine-3-carboxylic acid
8-(2,3-dihydro-1H-inden-2-yl)-1-ethyl-3-[(3-methoxyphenyl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
(2S)-3-methyl-2-({3-[(2-methylprop-2-en-1-yl)oxy]phenyl}formamido)butanamide
4-(1H-imidazol-2-yl)-1-[2-(methylsulfanyl)benzoyl]piperidine
N-(3-chloro-4-fluorophenyl)-3-{1-[(3-methyl-1H-1,2,4-triazol-5-yl)methyl]piperidin-4-yl}propanamide
5-({[1-(5-amino-1,3,4-thiadiazol-2-yl)ethyl]carbamoyl}amino)-2-chloro-N-(propan-2-yl)benzamide
2-({[2-methyl-6-(piperidin-4-yl)pyrimidin-4-yl]amino}methyl)adamantan-2-ol
N-[(5-methylpyrazin-2-yl)methyl]-2-(1H-pyrazol-1-yl)butanamide
1-[(3aR,5R,6S,7aS)-5,6-dihydroxy-octahydro-1H-isoindol-2-yl]-2-[(1-ethyl-1H-indol-3-yl)sulfanyl]ethan-1-one
4-methyl-2-{2-[3-(4-methyl-4H-1,2,4-triazol-3-yl)piperidin-1-yl]-2-oxoethyl}-1,2-dihydrophthalazin-1-one
2-[3-(4-benzyl-1H-pyrazol-5-yl)piperidin-1-yl]pyridine-3-carboxamide
({4-ethyl-5-[1-(1H-imidazol-4-ylmethyl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)dimethylamine
4-[4-(3-hydroxypyrrolidin-1-yl)pyrimidin-2-yl]-1-(3-methoxyphenyl)piperazin-2-one
[1-({[1-(pyridin-2-ylmethyl)piperidin-4-yl]amino}methyl)cyclopentyl]methanol
N-[(5-ethyl-1,3,4-thiadiazol-2-yl)methyl]-2,6-dimethylimidazo[1,2-a]pyridine-3-carboxamide
1-(3-chloropyridin-2-yl)-4-(5-methylpyridin-2-yl)piperidin-4-ol
1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-4-(pyridin-3-ylmethyl)-1,4-diazepane
[4-({1-[1-(pyrazine-2-carbonyl)piperidin-4-yl]pyrrolidin-3-yl}methyl)phenyl]methanol
N-{[7-methoxy-2-(pyrrolidin-1-yl)quinolin-3-yl]methyl}-N-(oxolan-2-ylmethyl)furan-3-carboxamide
4-(5-methylpyridin-2-yl)-1-[(3-phenoxyphenyl)methyl]piperidin-4-ol
N-ethyl-2-methyl-N-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}-5-sulfamoylbenzamide
2-(1-{[2-(furan-2-yl)pyrimidin-5-yl]methyl}pyrrolidin-2-yl)-1,3-benzothiazole
1-{4-[(4aR,8aS)-1-[1-(4-chlorophenyl)cyclobutanecarbonyl]-decahydro-1,6-naphthyridine-6-carbonyl]thiophen-2-yl}ethan-1-one