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4-{4-[1-(adamantan-1-yl)-1H-imidazol-2-yl]-1H-1,2,3-triazol-1-yl}piperidine
N,N-diethyl-2-{3-[3-(1-methyl-1H-imidazol-2-yl)phenyl]-1H-pyrazol-1-yl}acetamide
(1R,3s,6r,8S)-4-[(3R,4R)-4-(2-ethyl-4-methyl-1H-imidazol-5-yl)-1-methylpyrrolidine-3-carbonyl]-4-azatricyclo[4.3.1.13,8]undecane
3-chloro-5-({3-[3-(piperidin-1-yl)azetidine-1-carbonyl]-1,2-oxazol-5-yl}methoxy)pyridine
4-{[2-(furan-2-yl)-1H-imidazol-1-yl](4-methylphenyl)methyl}pyridine
2-cyclopropyl-9-[2-(dimethylamino)propanoyl]-2,9-diazaspiro[5.5]undecan-3-one
2-methoxy-N-[5-oxo-1-(3-phenylpropyl)pyrrolidin-3-yl]acetamide
2-({[(5-ethylpyridin-2-yl)methyl](methyl)amino}methyl)-4-hydroxyquinoline-6-carboxamide
N-(2,5-dimethoxyphenyl)-3-[(2R,6R)-6-methyl-2-(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridin-1-yl]-3-oxopropanamide
5-fluoro-N2,N4,N4-trimethyl-N2-(1,2-oxazol-3-ylmethyl)pyrimidine-2,4-diamine
1-(2,3-dihydro-1H-inden-5-yl)-2-(4-methyl-1H-imidazol-5-yl)-1H-imidazole
1-[9-(2,3-dihydro-1H-inden-2-yl)-3,9-diazaspiro[5.5]undecan-3-yl]-3,3-dimethylbutan-1-one
2-(2,5-dioxoimidazolidin-1-yl)-N-[6-(propan-2-yloxy)-1-(2,2,2-trifluoroethyl)-1H-indazol-3-yl]acetamide
6-ethyl-3-[1-(pyridin-3-yl)propan-2-yl]-3,4-dihydroquinazolin-4-one
({4-[1-(1H-indole-2-carbonyl)piperidin-2-yl]phenyl}methyl)dimethylamine
N-[2-(3-ethyl-1,2,4-oxadiazol-5-yl)ethyl]-4-(1-phenyl-1H-pyrazol-4-yl)pyrimidin-2-amine
(3S,4R)-4-(2-methoxyphenyl)-1-[2-(2-oxo-1,2-dihydropyridin-1-yl)acetyl]pyrrolidine-3-carboxylic acid
(3R)-1-{5-[(4-benzylpiperidin-1-yl)methyl]-1,2-oxazole-3-carbonyl}pyrrolidin-3-ol
N-[cyclopropyl(pyridin-2-yl)methyl]-3-(1H-imidazol-2-yl)-N-methylbenzamide
N-{[4-(3-methoxyphenyl)-5-({[3-(trifluoromethyl)phenyl]methyl}sulfanyl)-4H-1,2,4-triazol-3-yl]methyl}cyclopropanecarboxamide
2-ethoxy-1-{4-[4-methyl-5-(morpholin-4-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}ethan-1-one
4-methyl-N-[2-(2-phenoxyethoxy)phenyl]pyridine-3-carboxamide
4-(2,4-difluorophenyl)-3-[3-(morpholin-4-yl)propyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
3-methyl-7-[(3-methylthiophen-2-yl)methyl]-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
9-(4-chloro-1-methyl-1H-pyrrole-2-carbonyl)-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
1-[4-(2-phenoxyacetyl)piperazin-1-yl]-2-(1H-pyrazol-1-yl)butan-1-one
3-{[(6-fluoro-4-hydroxyquinolin-2-yl)methyl](2-phenylethyl)amino}propanamide
1-{1-[(4-hydroxyphenyl)methyl]piperidin-3-yl}-3-phenylpropan-1-one
6-(3,4-dimethylpiperazin-1-yl)-N-{3-[2-(propan-2-yl)-1H-imidazol-1-yl]propyl}pyridine-3-carboxamide
3-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-3-methyl-1-[4-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)phenyl]urea
2-(2-{1-[1-(4-methoxyphenyl)cyclopropanecarbonyl]piperidin-4-yl}-1H-imidazol-1-yl)acetamide
2-[2-(propan-2-yl)-1H-imidazol-1-yl]-1-[4-(thiophene-2-carbonyl)piperazin-1-yl]propan-1-one
2-(2,5-dihydro-1H-pyrrole-1-carbonyl)-N-methyl-N-(2-phenylethyl)-2,3-dihydro-1H-inden-2-amine
3-[methyl({[3-(3-methylphenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl})amino]propane-1,2-diol
N-{3-[3-(2-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-3-oxopropyl}methanesulfonamide
({2-[2-(1H-imidazol-1-yl)ethoxy]-3-methoxyphenyl}methyl)[1-(3-methylpyridin-2-yl)ethyl]amine
2-amino-4-(1,2-dimethyl-1H-imidazol-5-yl)-6-[1-(4-fluorophenyl)-1H-pyrazol-4-yl]pyridine-3-carbonitrile
6-[(3S,5R)-3-(hydroxymethyl)-5-{[(2-methoxyethyl)(methyl)amino]methyl}piperidine-1-carbonyl]-1,3-dimethyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-{4-[1-(cyclohex-1-en-1-ylmethyl)-1H-1,2,3-triazol-4-yl]phenyl}acetamide
4-{1-[4-(pyrrolidin-1-ylmethyl)benzoyl]piperidin-4-yl}thiomorpholine
3-(3-chlorophenyl)-3-(3-hydroxyphenyl)-N-methyl-N-(1-methylpiperidin-4-yl)propanamide
3-(3-methoxyphenyl)-5-(thian-4-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
1'-(4-cyclopentylpyrimidin-2-yl)-5-methyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N-[(3S,4R)-1-(5-chloropyridine-3-carbonyl)-4-(4-methoxyphenyl)pyrrolidin-3-yl]acetamide
N-(2-methyl-1-benzofuran-7-yl)-9-oxa-2-azaspiro[5.5]undecane-2-carboxamide
9-methoxy-7-(2-methylphenyl)-4-(thiophen-2-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
6-[3-(4-phenylpiperazin-1-yl)piperidine-1-carbonyl]pyridin-3-ol
N-(2-methoxyethyl)-1-[1-(3-methylbenzoyl)piperidin-4-yl]piperidine-3-carboxamide
3-({5-[3-(2-fluorophenyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}(methyl)amino)propane-1,2-diol
1-{1'-[2-(propan-2-ylsulfanyl)acetyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}propan-1-one