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3-(7-methoxy-2,3,4,5-tetrahydro-1H-3-benzazepine-3-carbonyl)-2-methyl-4,5,6,7-tetrahydro-1H-indol-4-one
N-({1-[(3-fluoro-2,4-dimethylphenyl)methyl]pyrrolidin-3-yl}methyl)furan-2-carboxamide
1-[5-(methoxymethyl)furan-2-carbonyl]-4-phenylpiperidine-4-carbonitrile
1-[(3R,4R)-3-(hydroxymethyl)-4-[(4-methylpiperazin-1-yl)methyl]pyrrolidin-1-yl]-3-(pyridin-2-yl)propan-1-one
2-(2-ethyl-4-methyl-6-oxo-1,6-dihydropyrimidin-5-yl)-N-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)acetamide
(3R,4R)-4-(4-hydroxypiperidin-1-yl)-1-{[4-(2-methylpropyl)phenyl]methyl}piperidin-3-ol
3-[({[2-(pyrimidin-2-yl)-1,3-thiazol-4-yl]methyl}amino)methyl]piperidin-3-ol
1-cyclobutanecarbonyl-N-[3-(1H-1,2,3-triazol-1-yl)propyl]piperidine-4-carboxamide
(1R,5R)-6-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]-3-(pyridine-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
2-{[3-(2-methylphenoxy)azetidin-1-yl]methyl}-1-propyl-1H-imidazole
8-[(4-{octahydropyrrolo[1,2-a]piperazine-2-carbonyl}-1,3-oxazol-2-yl)methoxy]quinoline
N-methyl-5-{[2-(methylsulfanyl)ethyl]amino}-1-(2-phenylethyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
3-{3-[2-(4-fluorophenyl)ethyl]piperidine-1-carbonyl}pyridazine
2-{5-[4-(1H-pyrazol-3-yl)phenyl]-3-(1H-1,2,4-triazol-1-ylmethyl)-1H-1,2,4-triazol-1-yl}ethan-1-ol
4-(5-methylpyridin-2-yl)-1-(1,3-thiazol-2-yl)piperidin-4-ol
2-cyclopropyl-N-[(4-fluorophenyl)methyl]-3-oxo-2,9-diazaspiro[5.5]undecane-9-carboxamide
{1-[4-(methoxymethyl)-5-methyl-1,2-oxazole-3-carbonyl]-3-(prop-2-en-1-yl)piperidin-3-yl}methanol
N-methyl-N-[1-(2-phenylethyl)piperidin-3-yl]-3-(pyridin-3-yl)propanamide
5-chloro-2-methyl-3-{2-[2-(1-methyl-1H-imidazol-2-yl)-1H-imidazol-1-yl]ethyl}-1H-indole
2-(4-chloro-1H-pyrazol-1-yl)-N-(3-hydroxy-3-methylbutyl)-N-methylpropanamide
1-ethyl-N-{1-[1-(4-methoxyphenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}-1H-pyrazole-3-carboxamide
1-[(1R,5R)-3-methanesulfonyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-(pyridin-2-ylsulfanyl)ethan-1-one
4-{2-[(3,4-dimethoxyphenyl)methyl]-1,3-benzoxazole-6-carbonyl}piperazin-2-one
3-(2-amino-1,3-thiazol-4-yl)-N-(2,3,4,9-tetrahydro-1H-carbazol-6-ylmethyl)propanamide
N-[2-(diethylamino)ethyl]-N-ethyl-5-(furan-2-yl)-1-[4-(2-methoxyphenyl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide
N-{2-[2-(hydroxymethyl)piperidin-1-yl]ethyl}-4,5,6-trimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
(1-{[2-(4-chlorophenyl)pyrimidin-5-yl]methyl}-3-ethylpiperidin-3-yl)methanol
8-cyclopentyl-2-[(3-methoxyphenyl)methyl]-2,8-diazaspiro[4.5]decan-3-one
4-methyl-6-[3-(propan-2-yloxy)phenyl]pyrimidin-2-amine
1-(adamantan-2-yl)-4-({3-[(2-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)piperazine
1-[2-(dimethylamino)ethyl]-N-methyl-6-oxo-N-(quinolin-5-ylmethyl)piperidine-3-carboxamide
8-[1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-1-oxa-8-azaspiro[4.6]undecane
4-chloro-N-[(3S,5S,9R)-2,8-dioxo-1,7-diazatricyclo[7.3.0.03,7]dodecan-5-yl]benzamide
(1R,5R)-6-(2-ethylbenzoyl)-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
4-(morpholin-4-yl)-N,N-bis(propan-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carboxamide
6-[(2R,3R,6R)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]pyridin-3-ol
4-[4-(2H-1,3-benzodioxol-5-ylmethyl)piperazin-1-yl]-2-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-2,3-dihydro-1H-isoindole-1,3-dione
6-methoxy-2-[4-(piperidin-3-yl)benzoyl]-1,2,3,4-tetrahydroisoquinoline
N-(2-hydroxyethyl)-4-methoxy-N-[(2E)-3-phenylprop-2-en-1-yl]cyclohexane-1-carboxamide
1-(2-ethyl-1H-1,3-benzodiazol-6-yl)-3-[(1-ethyl-1H-imidazol-2-yl)methyl]-3-methylurea
7-chloro-3-({ethyl[(1-methyl-1H-imidazol-2-yl)methyl]amino}methyl)-1,2-dihydroquinolin-2-one
N-(1H-imidazol-2-ylmethyl)-N-methyl-6-oxo-1-[2-(pyridin-2-yl)ethyl]piperidine-3-carboxamide
N-cyclopropyl-1-[(3-methoxyphenyl)methyl]-5-(pyridine-2-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
4-(azepane-1-carbonyl)-2-(2-ethylpyrimidin-5-yl)-6-methylquinoline
4-({spiro[azepane-4,2'-chromene]-1-yl}carbonyl)-1λ6-thiane-1,1-dione
8-[4-(4-hydroxypiperidin-1-yl)pyrimidin-2-yl]-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
1-(pyridin-3-ylmethyl)-4-[3-(4H-1,2,4-triazol-4-yl)benzoyl]-1,4-diazepane
2-(dimethyl-1,3-thiazol-5-yl)-1-{4-[hydroxy(thiophen-2-yl)methyl]piperidin-1-yl}ethan-1-one
1-{3-[3-(3-methylthiophen-2-yl)phenyl]-1H-pyrazol-1-yl}propan-2-ol
2-{5-cyclopropyl-4-[4-(propan-2-yl)piperazine-1-carbonyl]-1H-pyrazol-1-yl}-4-(5-methylfuran-2-yl)pyrimidine