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1-methyl-8-[(3-methylphenyl)methanesulfonyl]-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
1-[5,6-dimethyl-2-(trifluoromethyl)pyrimidin-4-yl]-4-(oxan-2-ylmethyl)piperidine-4-carboxylic acid
methyl 2-methyl-2-(2-{1-[(2-methylphenyl)methyl]-3-oxopiperazin-2-yl}acetamido)propanoate
N-cyclopropyl-2-(dimethyl-1,2-oxazol-4-yl)-N-({4-[(3-methyloxetan-3-yl)methoxy]phenyl}methyl)acetamide
1-[2-(4-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}piperidin-1-yl)-2-oxoethyl]imidazolidine-2,4-dione
1-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-3-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidine
5-[3-(2-phenylethyl)-1,2,4-oxadiazol-5-yl]-N-(pyrrolidin-3-yl)pyridin-2-amine
methyl 1-(2-methoxyethyl)-2-oxo-3-{[5-(propan-2-yl)-1,3,4-oxadiazol-2-yl]methyl}-2,3-dihydro-1H-1,3-benzodiazole-5-carboxylate
1-[4-(furan-2-yl)pyrimidin-2-yl]-N-(1-methoxybutan-2-yl)-5-methyl-1H-pyrazole-4-carboxamide
2-(1H-pyrazol-1-yl)-N-{[2-(pyrimidin-2-yl)-1,3-thiazol-4-yl]methyl}butanamide
4-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-1,2-dihydropyridin-2-one
1'-(2-methoxypyrimidine-5-carbonyl)-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
4-(4-{1-[(2R)-3,4-dihydro-2H-1-benzopyran-2-ylmethyl]-1H-imidazol-2-yl}-1H-1,2,3-triazol-1-yl)piperidine
N-[(5-chloro-1H-1,3-benzodiazol-2-yl)methyl]-1-(propan-2-yl)piperidin-4-amine
benzyl 3-(4-hydroxy-2-methylpyrimidine-5-amido)pyrrolidine-1-carboxylate
N-[2-(4-methoxyphenyl)ethyl]-5-methyl-N-[(1-methylpiperidin-4-yl)methyl]pyrazine-2-carboxamide
2-[9-hydroxy-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-1,3-thiazole-4-carboxamide
1-[1-(2-methylquinoline-4-carbonyl)piperidin-3-yl]-2-phenylethan-1-one
N-methyl-2-(4-methyl-1-oxo-1,2-dihydrophthalazin-2-yl)-N-{[2-(methylamino)pyrimidin-5-yl]methyl}acetamide
4-[2-(4-{[2-(propan-2-yl)pyrimidin-4-yl]methyl}piperazin-1-yl)ethyl]morpholine
3-methyl-7-[(5-propylfuran-2-yl)methyl]-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
N-{1-[1-(1-benzofuran-2-carbonyl)piperidin-4-yl]-2-(2-fluorophenyl)ethyl}-N,2-dimethylfuran-3-carboxamide
1-(cyclopropylmethyl)-N-ethyl-5-(pyridin-3-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-[(2S,4R)-4-[(4-methoxyphenyl)sulfanyl]-1-{[3-(trifluoromethyl)phenyl]methyl}pyrrolidine-2-carbonyl]-4-methyl-1,4-diazepane
2-[(3R,4S)-3-[(dimethylsulfamoyl)amino]-4-(propan-2-yl)pyrrolidin-1-yl]-6-methylpyridine-3-carbonitrile
(3S,4S)-4-(4-fluorophenyl)-1-(quinoxaline-5-carbonyl)piperidin-3-ol
4-hydroxy-N-methyl-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-2-[(phenylsulfanyl)methyl]pyrimidine-5-carboxamide
5-{[(5-chloropyridin-3-yl)oxy]methyl}-N-methyl-N-[(3-methyl-1,2-oxazol-5-yl)methyl]-1,2-oxazole-3-carboxamide
N-ethyl-6-(4-fluorophenyl)-7-(3-methylbut-2-en-1-yl)-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
5-{4-[(2R,6S)-2,6-dimethylmorpholin-4-yl]piperidin-1-yl}-1-ethyl-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazole
(3R,4S)-4-cyclopropyl-1-[4-methyl-2-(propan-2-yl)-1,3-thiazole-5-carbonyl]pyrrolidin-3-amine
2-({2-[2-(1H-imidazol-1-yl)ethyl]piperidin-1-yl}methyl)pyridine
2-(4-{[4-methoxy-3-(methoxymethyl)phenyl]methyl}-1-(2-phenylethyl)piperazin-2-yl)ethan-1-ol
9-[3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)propyl]-2-(propan-2-yl)-2,9-diazaspiro[5.5]undecan-3-one
N-(cyclopent-3-en-1-yl)-5-(pyrrolidin-2-yl)thiophene-2-carboxamide
1-{2-[3-(1,3-benzoxazol-2-yl)piperidin-1-yl]-2-oxoethyl}-5-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
6-[4-methoxy-3-(pyrrolidin-1-ylmethyl)phenoxy]pyridine-2-carbonitrile
(4-{5-[4-(2-phenylethyl)piperidine-1-carbonyl]pyridin-2-yl}phenyl)methanol
N-(2,1,3-benzothiadiazol-5-ylmethyl)-N-methyl-3-(piperidin-3-yl)benzamide
N-[3-(dimethylamino)propyl]-1-(4-ethylbenzenesulfonyl)-N-methylpiperidin-3-amine
(3S,4S)-4-[(dimethylamino)methyl]-1-[1-methyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]piperidin-3-ol
(2,1,3-benzoxadiazol-4-ylmethyl)(methyl)[(1-phenyl-1H-pyrazol-4-yl)methyl]amine
N-{2-[(4-chlorophenyl)methoxy]ethyl}-2-cyclopropyl-4-methylpyrimidine-5-carboxamide
3-[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]propanamide
1-({3-[(4-fluoro-3-methylphenyl)carbamoyl]phenyl}methyl)piperidine-4-carboxamide
2-(dimethylamino)-4-methyl-N-{[(2S)-5-oxopyrrolidin-2-yl]methyl}-N-(pyridin-3-ylmethyl)pyrimidine-5-carboxamide
N-methyl-1-(3-methyl-1H-indole-2-carbonyl)-N-[2-(pyridin-2-yl)ethyl]piperidin-3-amine
8-(4,6-dimethylpyrimidin-2-yl)-3-{2-[(2-methoxyethyl)(methyl)amino]ethyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
5-methyl-N-[2-(1-phenyl-1H-pyrazol-4-yl)ethyl]-1,3,4-oxadiazol-2-amine
1-(2,3-dihydro-1H-inden-2-yl)-4-{[3-(3-methoxyphenyl)-1,2-oxazol-5-yl]methyl}piperidin-4-ol