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(2R)-2-[(4-cyclopentylpyrimidin-2-yl)amino]propanamide
6-{[(2R,3R)-3-amino-2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl]carbonyl}-2-methyl-2,3-dihydropyridazin-3-one
N-{[2-(4-acetylpiperazin-1-yl)-5,8-dimethoxyquinolin-3-yl]methyl}-2-methyl-N-(oxolan-2-ylmethyl)-1,3-thiazole-4-carboxamide
({1-[2-(4-chlorophenyl)ethyl]piperidin-3-yl}methyl)(methyl){[1,2,4]triazolo[1,5-a]pyrimidin-2-ylmethyl}amine
2-{1-[(2,3-difluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]acetamide
2-{4-cyclohexyl-1-[(2-fluoro-4-methoxyphenyl)methyl]piperazin-2-yl}ethan-1-ol
methyl 3-benzamido-5-({[3-(propan-2-yl)-1H-pyrazol-5-yl]formamido}methyl)benzoate
N-(furan-2-ylmethyl)-2-[6-oxo-4-(pyrrolidin-1-yl)-1,6-dihydropyridazin-1-yl]-N-(prop-2-en-1-yl)acetamide
4-methyl-1-[3-(1H-1,2,3,4-tetrazol-1-yl)-5-(2,3,4-trimethoxyphenyl)benzoyl]piperidine
2-(3-chloro-2-fluorophenyl)pyridine-3-carboxamide
2-methoxy-1-{3-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}ethan-1-one
3-(1H-1,3-benzodiazol-2-ylmethyl)-6-methoxy-3,4-dihydroquinazolin-4-one
N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-3-(1-methyl-1H-pyrazol-4-yl)propanamide
(3aR,6aS)-5-({4-[(dimethylamino)methyl]thiophen-2-yl}methyl)-1-oxo-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-[(2-aminopyridin-3-yl)methyl]-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
7-[(3R,4S)-4-hydroxy-3,4-dimethylpiperidine-1-carbonyl]-1,2,3,4-tetrahydroquinoxalin-2-one
N-[(4-methoxyphenyl)methyl]-N-[(3-methylphenyl)methyl]oxane-4-carboxamide
(4aR,8aS)-N,N-dimethyl-1-(2-phenylpropanoyl)-decahydro-1,6-naphthyridine-6-sulfonamide
4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-N-[2-(6-hydroxy-2-methylpyrimidin-4-yl)ethyl]benzamide
1-(cyclohexyloxy)-3-[2-(1H-imidazol-2-yl)-1H-imidazol-1-yl]propan-2-ol
1-{4-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl}-2-[methyl(propan-2-yl)amino]ethan-1-one
2-{[5-chloro-2-(propan-2-yloxy)phenyl]methyl}-2,9-diazaspiro[5.5]undecan-3-one
2-(3,6-dioxo-1,2,3,6-tetrahydropyridazin-1-yl)-N-[(4-ethylphenyl)methyl]-N-(2-methoxyethyl)acetamide
3-(2,4-dimethoxyphenyl)-5-[(methylsulfanyl)methyl]-1,2,4-oxadiazole
N-(1,2-oxazol-3-ylmethyl)-3-(1H-pyrazol-4-yl)benzamide
N-{[4-(hydroxymethyl)oxan-4-yl]methyl}-N,6-dimethylpyridine-2-carboxamide
N-[4-methyl-1-(pentan-3-yl)-1H-pyrazol-5-yl]-2-[(propan-2-yl)amino]pyrimidine-5-carboxamide
4-methyl-2-({3-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl}methyl)phenol
5-{[methyl({1-[2-(2-methylphenyl)ethyl]piperidin-3-yl}methyl)amino]methyl}pyrimidin-2-amine
3-[(3S,4R)-1-[(2,3-dimethoxyphenyl)methyl]-4-[4-(2-fluorophenyl)piperazin-1-yl]piperidin-3-yl]-N-[(2-fluorophenyl)methyl]propanamide
5-{[(3-fluorophenyl)methyl]amino}-1-methyl-N-[2-(morpholin-4-yl)ethyl]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
3-[4-chloro-2-(trifluoromethyl)phenyl]-1-(2-oxopiperidin-3-yl)urea
2-hydroxy-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]naphthalene-1-carboxamide
N-{1-[3-(oxan-4-yl)-1H-1,2,4-triazol-5-yl]propyl}acetamide
3-[(3R,7S,8aS)-3-[(1S)-1-hydroxyethyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(4-chlorophenyl)urea
2-[5-(oxolan-2-yl)-3-(propan-2-yl)-1H-1,2,4-triazol-1-yl]pyridine
3-[2-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-1-(3-methylcinnolin-5-yl)urea
5-{1-[3-(1H-1,3-benzodiazol-2-yl)propanoyl]pyrrolidin-2-yl}-N-methylthiophene-2-carboxamide
(1S,5R)-6-(cyclobutylmethyl)-3-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}-3,6-diazabicyclo[3.2.2]nonan-7-one
2-[4-({methyl[(2-methyl-1H-imidazol-4-yl)methyl]amino}methyl)piperidin-1-yl]ethan-1-ol
5-ethyl-N4-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}-6-methylpyrimidine-2,4-diamine
(3aR,6aS)-5-{[4-ethoxy-3-(hydroxymethyl)phenyl]methyl}-1-oxo-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-(5-fluoropentyl)-3-methyl-1,2-dihydroquinoxalin-2-one
N-[1-(5-methyl-1-benzofuran-2-carbonyl)piperidin-4-yl]pyrimidin-2-amine
3-({2-[1-(5-methylthiophene-2-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}methyl)pyridine
2-[2-(quinolin-8-yl)-1H-1,3-benzodiazol-1-yl]ethan-1-ol
(1S,5R)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-(1,3-thiazole-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-(4-methoxy-2-methylphenyl)-3-[1-(oxan-4-yl)piperidin-3-yl]propanamide
N-[2-methoxy-1-(pyridin-2-yl)ethyl]-N-methyl-2-(1H-pyrazol-1-yl)benzamide
1-[4-methyl-2-({2-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}amino)pyrimidin-5-yl]ethan-1-one