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2-{5-[2-(1H-1,2,4-triazol-5-yl)benzoyl]-3H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}pyridine
6-amino-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]pyridine-3-carboxamide
2-ethyl-5-{2-[2-(thiophen-2-yl)ethyl]piperidine-1-carbonyl}pyrimidine
1-(4-chlorophenyl)-N-{[1-(cyclohex-1-ene-1-carbonyl)piperidin-3-yl]methyl}cyclopropane-1-carboxamide
1-[(1R,2R,6S,7S)-4-azatricyclo[5.2.1.02,6]decan-4-yl]-2-(4-methanesulfonylphenyl)ethan-1-one
N-{1-benzyl-2-methyl-7-[2-(pyridin-3-yl)piperidine-1-carbonyl]-1H-1,3-benzodiazol-5-yl}-2-methylpropanamide
(3aR,6aR)-2-cyclopropanecarbonyl-5-[(1-ethyl-1H-imidazol-2-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-amino-6-cyclopentyl-4-(2,4,5-trimethoxyphenyl)pyridine-3-carbonitrile
9-{[3-ethoxy-4-methoxy-5-(prop-2-en-1-yl)phenyl]methyl}-1,4,9-triazaspiro[5.5]undecan-5-one
ethyl 2-{9-[(2-fluorophenyl)methyl]-1-(hydroxymethyl)-3,9-diazaspiro[5.5]undecan-3-yl}acetate
1,9-dimethyl-4-[2-oxo-2-(piperidin-1-yl)ethyl]-1,4,9-triazaspiro[5.6]dodecan-10-one
6-[(diethylamino)methyl]-N-[(3-methylphenyl)methyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide
N-{2-[(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)amino]ethyl}-4-(piperidin-3-yl)benzamide
7-cyclohexyl-2-[2-(morpholin-4-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one
1-benzyl-5-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-3-(1H-1,2,4-triazol-1-ylmethyl)-1H-1,2,4-triazole
7-[(3,4-difluorophenyl)methyl]-2-(3-methyl-5,6-dihydro-1,4-dioxine-2-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
4-{[5-(4-aminopyrimidin-2-yl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}-1λ6-thiomorpholine-1,1-dione
1-ethyl-N-[(4-methoxyphenyl)methyl]-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-{3-[(1-cyclohexyl-1H-1,2,4-triazol-5-yl)methoxy]phenyl}-1H-1,2,3,4-tetrazole
1-ethyl-6-methyl-3-(3-phenylpiperazine-1-carbonyl)-1,2-dihydropyridin-2-one
4-[3-(2,5-dimethoxyphenyl)pyrrolidine-1-carbonyl]-1λ6-thiane-1,1-dione
1-{2-[1-(2-methoxy-5-methylbenzoyl)piperidin-4-yl]ethyl}pyrrolidin-2-one
2-[2-(3-methoxyphenyl)ethyl]-4-{4-[2-(4-oxo-3,4-dihydrophthalazin-1-yl)propanoyl]piperazin-1-yl}-2,3-dihydro-1H-isoindole-1,3-dione
5-acetyl-N,6-dimethyl-N-{[3-(3-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl}-2-oxo-1,2-dihydropyridine-3-carboxamide
3-benzoyl-1-[1-(3-phenylpropyl)-1H-1,2,3-triazole-4-carbonyl]piperidine
1-[2-({imidazo[2,1-b][1,3]thiazol-6-ylmethyl}amino)pyrimidin-4-yl]piperidin-3-ol
2-[(3R,4S)-3-(2-methyl-1H-pyrrole-3-amido)-4-(propan-2-yl)pyrrolidin-1-yl]acetic acid
1,3-dimethyl-5-{2-[6-(methylsulfanyl)-1,2,3,4-tetrahydroisoquinolin-2-yl]-2-oxoethyl}imidazolidine-2,4-dione
4-({3-[2-(2,6-difluorophenyl)ethyl]piperidin-1-yl}methyl)-2-methoxyphenol
N-cyclopropyl-5-methyl-4-{[(4-phenyloxan-4-yl)methyl]amino}thieno[2,3-d]pyrimidine-6-carboxamide
4-benzyl-1-[(dimethyl-1,2-oxazol-4-yl)methyl]piperidine
(2S,4R)-4-[2-(2,3-dihydro-1H-inden-5-yloxy)-2-methylpropanamido]-N-ethyl-1-methylpyrrolidine-2-carboxamide
N4-(1H-1,3-benzodiazol-2-ylmethyl)-N4-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine
5-[(4-fluorophenyl)methyl]-3-[(2-methyl-1,3-oxazol-4-yl)methyl]-5-(piperidin-4-yl)imidazolidine-2,4-dione
4-ethyl-3-(1-{2H,3H-thieno[3,4-b][1,4]dioxine-5-carbonyl}piperidin-4-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
1-{4-[(3R,4S)-3-(dimethylamino)-4-propylpyrrolidine-1-carbonyl]phenyl}pyrrolidin-2-one
N-[2-(cyclohexylsulfanyl)ethyl]-1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
N-(carbamoylmethyl)-2-[1-(2,2-diphenylethyl)-3-oxopiperazin-2-yl]acetamide
6-{2-[(4-methoxyphenyl)methyl]-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}pyridin-3-ol
2-(2H-1,3-benzodioxol-5-yl)-N-({2-methylimidazo[2,1-b][1,3]thiazol-6-yl}methyl)acetamide
4-{[4-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-2-(pyridin-3-yl)morpholine
4-[2-(aminomethyl)-7-chloro-2,3-dihydro-1-benzofuran-5-yl]-3-fluorobenzene-1-sulfonamide
methyl (2S)-1-({4-[(5-acetamidothiophen-2-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}methyl)pyrrolidine-2-carboxylate
methyl 2-(ethylsulfamoyl)-6-(3-phenylpropanoyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
N-{2-[1-(4-chloro-2-methylphenyl)-3-(ethoxymethyl)-1H-1,2,4-triazol-5-yl]ethyl}acetamide
4-(6-ethyl-2-methylquinoline-4-carbonyl)-1λ6-thiomorpholine-1,1-dione
N-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)-2-[4-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]acetamide
methyl 6-{4-[(4-fluorophenyl)methyl]-1,4-diazepan-1-yl}pyrimidine-4-carboxylate
(3aR,7aS)-2-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}-2,3,3a,4,7,7a-hexahydro-1H-isoindole
6-chloro-2-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}quinoline