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(3aR,6aR)-2-[2-(1H-indol-3-yl)ethyl]-5-methanesulfonyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-(4-{2-methyl-4-oxo-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl}phenyl)imidazolidine-2,4-dione
4-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
3-(1-butyl-1H-imidazol-2-yl)-1-(3,5-dimethyl-1-benzofuran-2-carbonyl)piperidine
{[2-(4-methoxy-2,3-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)(pyrazin-2-ylmethyl)amine
1-(2-methyl-1H-pyrrole-3-carbonyl)-3-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
1-{2-[(3aR,7aS)-5-methyl-2,3,3a,4,7,7a-hexahydro-1H-isoindol-2-yl]-2-oxoethyl}-3-butyl-4-ethyl-4,5-dihydro-1H-1,2,4-triazol-5-one
4-(2-chloro-4-fluorophenyl)-5-(cyclopropylmethyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
6-(2-{imidazo[1,2-a]pyridin-2-yl}ethyl)-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
6-cyclobutyl-2-{3-[(3-ethylmorpholin-4-yl)methyl]phenyl}-3,4-dihydropyrimidin-4-one
dimethyl(3-{2-[1-(2-methyl-1H-pyrrole-3-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}propyl)amine
4-(3-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)pyridine
1-(2-methylbenzenesulfonyl)-4-(1H-pyrazol-1-yl)piperidine-4-carboxylic acid
N-[(1S,3aS,6aS)-octahydropentalen-1-yl]-2,6-difluoro-3-methoxybenzamide
N-butyl-3-{[4-(2-methoxyethyl)piperazin-1-yl]methyl}-N-methylimidazo[1,2-a]pyridine-2-carboxamide
5-(2H-1,3-benzodioxol-5-ylmethyl)-1-(3-methoxypropyl)-5-methylpiperidin-2-one
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]acetamide
N-[2-(1H-imidazol-2-yl)ethyl]-1,3-dimethyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
5-amino-N-{2-[4-(cyclopentylmethyl)morpholin-2-yl]ethyl}-1H-pyrazole-3-carboxamide
N-[(2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)methyl]-5-[1-(piperidin-1-yl)ethyl]furan-2-carboxamide
1-{2-[4-(3-phenylbutyl)piperazin-1-yl]ethyl}-N-(propan-2-yl)-1H-1,2,3-triazole-4-carboxamide
[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl](methyl)[(2R)-2-phenylbutyl]amine
1-{2-[(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)amino]ethyl}-4-oxo-5-phenoxy-1,4-dihydropyridine-3-carboxylic acid
N-ethyl-N-(4-hydroxybutyl)-1,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
2-amino-6-methyl-N-(2-{[2-(morpholin-4-yl)ethyl]carbamoyl}phenyl)pyrimidine-4-carboxamide
1-[4-({4-[(2-methyl-1,3-thiazol-4-yl)methyl]piperazin-1-yl}methyl)thiophen-2-yl]ethan-1-one
N-[(3-hydroxypyrrolidin-3-yl)methyl]-5-phenyl-1,3-oxazole-4-carboxamide
4-chloro-N-{[1-methyl-2-(methylsulfanyl)-1H-imidazol-5-yl]methyl}-1H-pyrrolo[2,3-b]pyridin-6-amine
N-{[2-(2,4-difluorophenoxy)pyridin-3-yl]methyl}-2-methylpentanamide
N-[(3R,5S)-5-(hydroxymethyl)-1-methylpyrrolidin-3-yl]-2,6-dimethylpyrimidine-4-carboxamide
6-cyclopropyl-N-[2-(4-fluorobenzenesulfonyl)ethyl]pyrimidin-4-amine
2-methoxy-N-{4-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]phenyl}acetamide
1-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-4-(1H-pyrazol-3-yl)piperidine
2-oxo-N-(3-phenylprop-2-yn-1-yl)-N-propyl-2H-chromene-3-carboxamide
5-{1-[3-(hydroxymethyl)-4-methoxyphenyl]-1H-imidazol-2-yl}thiophene-2-carboxylic acid
[(2,3-dimethyl-1H-indol-7-yl)methyl](methyl)[1-(1,2-oxazol-3-yl)ethyl]amine
2-methyl-6-[3-(phenylamino)piperidine-1-carbonyl]-4H,7H-pyrazolo[1,5-a]pyrimidin-7-one
2-(4-{5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl}-1,4-diazepan-1-yl)-1,3-benzothiazole
N-[2-({5-[(4-benzylpiperidin-1-yl)methyl]-1,2-oxazol-3-yl}formamido)ethyl]acetamide
2-amino-6-cyclopropyl-4-[3-(3,4-dimethoxyphenyl)-1H-pyrazol-4-yl]pyridine-3-carbonitrile
1-{8-chloro-1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-yl}-3-[methyl(1-methylpyrrolidin-3-yl)amino]propan-1-one
2-methyl-5-[3-(4-propylphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]pyrimidine
2-(3,4-dichlorophenyl)-1-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]ethan-1-one
N-methyl-3-phenyl-N-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-1H-pyrazole-5-carboxamide
5-ethyl-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-1,3-oxazole-4-carboxamide
3-[(3R,4S)-1-(5-ethylthiophene-2-carbonyl)-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propan-1-ol
3-[5-(4-chlorophenyl)-1H-pyrrol-2-yl]-1-[4-(dimethylamino)azepan-1-yl]propan-1-one
2-(1H-1,3-benzodiazol-2-yl)-N-butyl-N-[(2-fluorophenyl)methyl]acetamide
N-ethyl-5-(3-fluorophenoxymethyl)-N-(pyridin-2-ylmethyl)-1H-pyrazole-3-carboxamide
5-tert-butyl-4-{[(3R,4R)-4-hydroxy-4-(2-methoxyethyl)-3-methylpiperidin-1-yl]methyl}furan-2-carboxamide