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1-{[4-(1H-imidazol-1-yl)phenyl]methyl}-4-[(2-methylphenyl)methyl]piperazine
2-(3-chlorophenyl)-N-{1-[(4-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}acetamide
2-[3-(1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-N-(2-acetamidophenyl)acetamide
[1-({methyl[1-methyl-6-(pyridin-3-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]amino}methyl)cyclopentyl]methanol
N-[(3R,4S)-4-cyclopropyl-1-[(3-ethyl-1,2-oxazol-5-yl)methyl]pyrrolidin-3-yl]oxane-4-carboxamide
2-{5-[4-(2-amino-6-methylpyrimidin-4-yl)piperazine-1-carbonyl]-1H-pyrazol-3-yl}phenol
4-benzyl-1-({6-methylimidazo[1,2-a]pyridin-2-yl}methyl)-3-(piperidin-4-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
N-[(3R,4R)-4-(piperidin-1-yl)oxolan-3-yl]-1H-pyrrolo[2,3-b]pyridin-6-amine
[1-({5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl}methyl)-3-(3-methylbut-2-en-1-yl)piperidin-3-yl]methanol
8-[2-(3-fluoro-4-methylphenyl)acetyl]-2-(2-hydroxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
N'-(2-ethoxyphenyl)-N-(1H-imidazol-2-ylmethyl)propanediamide
N-[(2S,4R,6S)-2-(2-methylpropyl)-6-[4-(pyrimidin-2-yloxy)phenyl]oxan-4-yl]acetamide
7-fluoro-N-[(3S,4S)-4-methoxy-1-(propan-2-yl)pyrrolidin-3-yl]quinazolin-4-amine
7-[2-(2H-1,3-benzodioxol-5-yloxy)propanoyl]-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-3-carboxamide
3-{1-[(2-hydroxyphenyl)methyl]piperidin-3-yl}-N-[4-(trifluoromethyl)phenyl]propanamide
(1R,7S)-3-[(3,4-dimethylphenyl)methyl]-N-methyl-4-oxo-N-(1,3-thiazol-2-ylmethyl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
6-[3-(dimethylamino)phenyl]-N,N-dimethylpyridine-2-carboxamide
(1-{[1-(2,4,6-trimethylbenzenesulfonyl)piperidin-3-yl]methyl}-1H-1,2,3-triazol-4-yl)methanol
(1R,5R)-6-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propanoyl]-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
6-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]pyridin-2-amine
[1-(adamantan-2-yl)-3-[(2-methylphenyl)methyl]piperidin-3-yl]methanol
1,5,6-trimethyl-3-{3-phenyl-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl}-1,2-dihydropyridin-2-one
methyl 4-({[1-(7-methanesulfonyl-4-methylquinazolin-2-yl)piperidin-3-yl]formamido}methyl)benzoate
N-[(2R,3R)-2-methoxy-1'-(3-phenylprop-2-yn-1-yl)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]thiophene-2-carboxamide
5-(1,7-dimethyl-1H-indole-2-carbonyl)-10-methoxy-3,4,5,6-tetrahydro-2H-1,5-benzoxazocine
N-[(3R,4S)-4-cyclopropyl-1-(3-methylpyrazin-2-yl)pyrrolidin-3-yl]-2-[(2-methoxyethyl)(methyl)amino]acetamide
3-{[4-(2,5-dimethylpyrimidin-4-yl)piperazin-1-yl]methyl}quinoline
3-methyl-N-{[6-(morpholin-4-yl)pyrimidin-4-yl]methyl}-3H-[1,2,3]triazolo[4,5-b]pyridine-6-carboxamide
N-[2-(4-amino-6-hydroxypyrimidin-2-yl)ethyl]-3-(1-methylpiperidin-3-yl)propanamide
1-{5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepin-8-yl}-2-(3-methylpiperidin-1-yl)propan-1-one
4-(2,6-dimethoxyphenyl)-N-methylbenzamide
methyl 3-{[(1R,2R,4R)-bicyclo[2.2.1]hept-5-en-2-ylformamido]methyl}-5-(2-chlorobenzenesulfonamido)benzoate
4-[4-(pyridin-3-ylmethoxy)piperidine-1-carbonyl]-1,2,3,4-tetrahydroquinolin-2-one
(4aS,7aR)-4-[2-(dimethylamino)acetyl]-6,6-dioxo-N-(propan-2-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
1-[5-(methoxymethyl)furan-2-carbonyl]-2-(thiophen-2-yl)azetidine
2-(pyridin-4-ylmethyl)-8-(1H-pyrrole-3-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
1-methyl-N-[1-(3-methyl-1,2,4-oxadiazol-5-yl)propyl]-3-propyl-1H-pyrazole-5-carboxamide
N-methyl-N-[(2E)-3-phenylprop-2-en-1-yl]-6-(piperidin-4-yl)pyrimidin-4-amine
1,7-dimethyl-N-[1-(1-methyl-1H-pyrazol-5-yl)propyl]-1H-indole-2-carboxamide
4-[3-(4-methyl-1,3-thiazol-5-yl)propanamido]-N-phenylpiperidine-1-carboxamide
8-[2-(oxolan-3-yl)ethyl]-3-(2-phenoxyethyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-(1-cycloheptylpiperidin-3-yl)-1-methyl-4-phenylpiperidine-4-carboxamide
methyl({2-[4-methyl-2-(1H-pyrazol-4-yl)phenoxy]ethyl})amine
5-cyclopropanecarbonyl-1'-[(1-methyl-1H-indol-2-yl)methyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
4-{[7-methyl-2-(3-methylphenyl)quinolin-3-yl]methyl}piperazine-1-carboxamide
{3-methyl-1-[4-(propan-2-yl)phenyl]-1H-1,2,4-triazol-5-yl}methanol
[3-(3-methoxypropyl)-1-(1,3-thiazol-2-ylmethyl)piperidin-3-yl]methanol
4-(pyridin-3-yl)-N-[3-(1H-1,2,4-triazol-1-yl)propyl]pyrimidin-2-amine
1-(2-butanamidoethyl)-N-[1-(thiophen-2-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
3-[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]-N-(4,5,6,7-tetrahydro-1-benzothiophen-3-ylmethyl)propanamide