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N-[(3S,4R)-1-{[5-(1,2-oxazol-3-yl)thiophen-2-yl]sulfonyl}-4-propylpyrrolidin-3-yl]acetamide
1-(4-acetyl-4-phenylpiperidin-1-yl)-2-(morpholin-2-yl)ethan-1-one
1-[4-(2-amino-1,3-benzothiazole-5-carbonyl)piperazin-1-yl]-2-phenoxyethan-1-one
N-[2-(4,6-dimethylpyrimidin-2-yl)ethyl]-3-hydroxy-1,2-oxazole-5-carboxamide
butyl 2-[2-(1H-imidazol-4-yl)ethyl]-3-oxo-2,9-diazaspiro[5.5]undecane-9-carboxylate
3-{[(furan-3-ylmethyl)(methyl)amino]methyl}-N-(trimethyl-1H-pyrazol-4-yl)benzamide
3-(morpholine-4-sulfonyl)-N-(pyrimidin-4-ylmethyl)benzamide
6-methyl-N-[(1-methyl-2-oxo-1,2,3,4-tetrahydroquinolin-4-yl)methyl]-4-oxo-4H-pyran-2-carboxamide
(3aS,6aR)-3-[2-(4-methoxyphenyl)ethyl]-5-(oxan-4-yl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
2-[4-(4-acetyl-3,5-dimethyl-1H-pyrazol-1-yl)phenoxy]propanamide
1-{2-methyl-2,7-diazaspiro[4.5]decan-7-yl}-2-(prop-2-en-1-ylsulfanyl)ethan-1-one
3-[(3S,4R)-1-[(2-chlorophenyl)methyl]-4-(morpholin-4-yl)piperidin-3-yl]-N-(3-methylphenyl)propanamide
5-(4-methyl-2-oxo-1,2-dihydroquinolin-3-yl)thiophene-2-carboxylic acid
ethyl 5-(oxolane-3-carbonyl)-1-(2-phenylethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
(furan-2-ylmethyl)(methyl)[(5-{[(2-methylphenyl)methyl]sulfanyl}-4-(oxolan-2-ylmethyl)-4H-1,2,4-triazol-3-yl)methyl]amine
4-{3-[3-(2-methoxyphenoxy)azetidin-1-yl]-2,2-dimethylpropyl}morpholine
2-{[4-(3-methoxyphenyl)-2-methyl-3-oxopiperazin-1-yl]methyl}benzoic acid
1,3-dimethyl-N-[1-(1,3-thiazol-2-yl)propyl]-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
1-{4-[(3-fluoro-4-methoxyphenyl)methyl]-1-methyl-1,4,9-triazaspiro[5.5]undecan-9-yl}-2-methoxyethan-1-one
N-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)-8-fluoroquinoline-2-carboxamide
N-(2-aminoethyl)-4-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzamide
[(2-methoxyphenyl)methyl](prop-2-en-1-yl)(1,3-thiazol-2-ylmethyl)amine
(3S,4R)-1-(carbamoylmethyl)-4-(3-methoxyphenyl)pyrrolidine-3-carboxylic acid
2-[1-methyl-5-(3,4,5-trifluorophenyl)-1H,4H-pyrazolo[3,4-d]imidazol-3-yl]pyridine
3-(4-methylphenoxymethyl)-1-(1,3-thiazol-4-ylmethyl)piperidine
2-(2-{1-[2-(difluoromethoxy)benzoyl]piperidin-4-yl}-1H-imidazol-1-yl)acetamide
1-cyclopentyl-3-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}urea
N-[2-(dimethylamino)-1-phenylethyl]-3-ethyl-N-methyl-1H-pyrazole-5-carboxamide
N3-benzyl-N5-(1-benzylpyrrolidin-3-yl)-4-oxo-1-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide
2-({[3-(methylsulfanyl)phenyl]methyl}carbamoyl)acetic acid
2-[3-(3-benzyl-1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)propanamido]-2-methylpropanoic acid
2-[(4aS,8aR)-1-(4-hydroxybutyl)-2-oxo-decahydro-1,6-naphthyridin-6-yl]-6-(propan-2-yl)pyridine-3-carbonitrile
[(2S,6S)-4-[5-(propan-2-yl)-1,3,4-thiadiazol-2-yl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(9),10,12-trien-6-yl]methanol
2-cyclopentyl-9-(2-fluorobenzenesulfonyl)-2,9-diazaspiro[5.5]undecan-3-one
1-[9-hydroxy-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-3-(1,2-oxazolidin-2-yl)propan-1-one
N-[2-(morpholin-4-yl)ethyl]-3-[(thiophen-2-ylmethyl)amino]benzamide
1-cyclopentyl-4-[4-(2-methylphenyl)-1,4-diazepane-1-carbonyl]pyrrolidin-2-one
7-(cyclobutylmethyl)-2-[2-(pyridin-4-ylsulfanyl)acetyl]-2,7-diazaspiro[4.5]decan-6-one
2-{[(2-methyl-1,3-benzothiazol-5-yl)oxy]methyl}-N-[1-(5-methyl-1H-1,2,4-triazol-3-yl)ethyl]-1,3-oxazole-4-carboxamide
N-{3-[4-amino-6-(benzylamino)-1,3,5-triazin-2-yl]phenyl}acetamide
N-benzyl-2-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidine-1-sulfonamide
N-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-5-ethyl-2-methylpyrimidin-4-amine
5-methyl-1-{2-[2-(4-methylpentyl)morpholin-4-yl]-2-oxoethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-{4-[3-(dimethylamino)pyrrolidine-1-carbonyl]-2-methylphenyl}furan-2-carboxamide
(3R,4R)-1-[4-(ethylamino)pyrimidin-2-yl]-4-[4-(pyridin-2-yl)piperazin-1-yl]piperidin-3-ol
4-(5,6-dimethylpyrimidin-4-yl)-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
1-[1-(2-phenylethyl)-5-(quinoxalin-5-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl]piperidin-4-ol
8-{[2-(5-methylfuran-2-yl)phenyl]methyl}-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
4-{1-[4-(2-oxopiperidin-1-yl)butanoyl]piperidin-3-yl}benzoic acid
1-cyclopentanecarbonyl-4-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]piperidine