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2-{3-[2-(3-methoxyphenyl)ethyl]piperidine-1-carbonyl}-5-methylpyrazine
N-methyl-N-[(5-methyl-1H-pyrazol-3-yl)methyl]-2-[(quinolin-8-yloxy)methyl]-1,3-oxazole-4-carboxamide
N-methyl-N-{[2-(2-methylpropoxy)phenyl]methyl}-2-(pyrrolidin-1-yl)acetamide
2-(5-acetylthiophen-3-yl)-1-[3-(2-methylphenyl)piperidin-1-yl]ethan-1-one
6-[3-(1-phenylcyclopropyl)-1-propyl-1H-1,2,4-triazol-5-yl]-5H-[1,3]thiazolo[3,2-a]pyrimidin-5-one
(5S,9aS,9bS)-5-[2-(4-methoxyphenyl)pyrimidin-5-yl]-2-phenyl-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
1-{[3-(1-phenylcyclopropyl)-1,2,4-oxadiazol-5-yl]methyl}pyrrolidin-2-one
methyl 4-{[1-benzyl-2,4-dioxo-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decan-8-yl]methyl}benzoate
1-[3-(hydroxymethyl)-3-(3-methylbut-2-en-1-yl)piperidin-1-yl]-2-(3-methyl-1,2-oxazol-5-yl)ethan-1-one
N-methyl-5-oxo-N-[2-(phenylsulfanyl)ethyl]-1-(pyridin-3-ylmethyl)pyrrolidine-3-carboxamide
[3-(1H-imidazol-1-yl)propyl](pyridin-2-ylmethyl)(pyridin-3-ylmethyl)amine
{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}(methyl){4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}amine
(2S)-2-acetamido-N-[(1-methyl-1H-imidazol-2-yl)methyl]-4-(methylsulfanyl)butanamide
2-[3-(1H-imidazol-1-yl)propyl]-6-methyl-4-(trifluoromethyl)pyridine
1-{4-[(2-methylphenyl)sulfanyl]piperidin-1-yl}-3-(1H-1,2,4-triazol-1-yl)propan-1-one
1-(2-methoxyethyl)-4-[1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]piperazine
6-tert-butyl-N,1-dimethyl-N-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
1-(2-methylphenyl)-4-{[2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]methyl}-1,4-diazepane
2-{1-[(4-chloro-3-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-N-(propan-2-yl)acetamide
(1R,4S)-1,7,7-trimethyl-3-oxo-N-[3-(pyridin-3-yloxy)propyl]-2-oxabicyclo[2.2.1]heptane-4-carboxamide
(4aS,7aR)-1-[(4-hydroxyphenyl)methyl]-4-(pyridin-3-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[2-(1-methylpyrrolidin-2-yl)ethyl]-3-{[1-(2-phenylethyl)piperidin-4-yl]oxy}benzamide
2-(5-cyano-6-methyl-1,2,3,4-tetrahydro-2,7-naphthyridin-2-yl)-N-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)acetamide
N,N-bis(propan-2-yl)-2-[5-(pyrrolidin-1-ylmethyl)pyridin-2-yl]benzamide
N-[(1-ethyl-1H-imidazol-2-yl)methyl]-N-methyl-2-(1-oxo-1,2-dihydroisoquinolin-2-yl)acetamide
4-methyl-N-[2-methyl-3-(pyrrolidine-1-carbonyl)phenyl]-1,2,3,6-tetrahydropyridine-1-carboxamide
(4aS,7aR)-1-{6-methylimidazo[2,1-b][1,3]thiazole-5-carbonyl}-4-propyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-[5-(3-fluorophenyl)-1,2,4-triazin-3-yl]azocane
2-(2,2-diphenylethyl)-4-(4-methylpyrimidine-5-carbonyl)morpholine
5-(3,4-dimethylphenoxymethyl)-3-[3-(methoxymethyl)pyrrolidine-1-carbonyl]-1,2-oxazole
5-({1,9-dimethyl-1,4,9-triazaspiro[5.5]undecan-4-yl}methyl)-N-propylpyrimidin-2-amine
[(3R,4S)-1-[(5-methylnaphthalen-1-yl)methyl]-4-(morpholin-4-ylmethyl)pyrrolidin-3-yl]methanol
N'-cyclopentyl-N-[(5-phenyl-1H-pyrazol-3-yl)methyl]butanediamide
N-[(2R,3R)-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-3-phenoxypropanamide
1-[1-(3-methoxybenzoyl)piperidin-4-yl]-3-(pyrrolidine-1-carbonyl)piperidine
1-[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)ethyl]-3-[5-(2-methylphenyl)-1,3,4-thiadiazol-2-yl]urea
(2R)-N-[1-benzyl-4-(morpholin-4-yl)-1H-indazol-3-yl]oxolane-2-carboxamide
1-(3-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}piperidin-1-yl)-2-(phenylsulfanyl)ethan-1-one
N-(3-methoxypropyl)-6-[4-(pyrrolidin-1-yl)piperidin-1-yl]-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
3-[2-(3,4-difluorophenyl)ethyl]-1-(1H-pyrazole-4-carbonyl)piperidine
N-[(5-chloro-3-methyl-2-phenyl-1H-indol-7-yl)methyl]-2,5-dimethyl-1,3-oxazole-4-carboxamide
2-{2-[(2R,3R,6R)-3-(3-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]ethoxy}ethan-1-ol
(3E)-2-{[2-(1H-imidazol-1-yl)ethyl](methyl)amino}-5,5-dimethylhex-3-enoic acid
3-(1-{[3-(4-chlorophenyl)-1H-pyrazol-4-yl]methyl}piperidin-4-yl)-N-(2-methoxyethyl)propanamide
3-butyl-4-(5-methoxy-1H-indazole-3-carbonyl)-1-methylpiperazin-2-one
5-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-3-(3-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
5-phenyl-N-[2-(3-phenylpyrrolidin-1-yl)ethyl]-1,2-oxazole-3-carboxamide
6-chloro-N,N-dimethyl-3-({methyl[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)ethyl]amino}methyl)imidazo[1,2-a]pyridine-2-carboxamide
5,8-dimethyl-2-({[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]amino}methyl)quinolin-4-ol
N-[1-(cyclohexylmethyl)piperidin-3-yl]-4-(1H-1,2,4-triazol-1-yl)butanamide