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N-[2-(dimethylsulfamoyl)ethyl]-1-methyl-2-oxo-1,2-dihydroquinoline-3-carboxamide
2-(7-chloro-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-2-[4-(hydroxymethyl)phenyl]acetic acid
N-benzyl-4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperazine-1-sulfonamide
1-(benzyloxy)-8-(thian-4-yl)-1,8-diazaspiro[4.5]decan-2-one
4-[1-(8-chloroquinolin-2-yl)pyrrolidin-3-yl]benzoic acid
2-(2-{[(6-hydroxy-2-methylpyrimidin-4-yl)methyl]amino}pyrimidin-4-yl)pyridine-4-carboxylic acid
1-(2-{[4-(3-hydroxy-3-methylbutyl)phenyl]formamido}ethyl)piperidine-3-carboxamide
6-(aminomethyl)-2-[(4-methoxyphenyl)methyl]-3,4-dihydropyrimidin-4-one
N-[1-(3-ethyl-1,2,4-oxadiazol-5-yl)ethyl]-3,6-dimethyl-2-(1H-pyrazol-4-yl)quinoline-4-carboxamide
6-[3-(1H-pyrazol-1-yl)propyl]-5,6-dihydro-1,6-naphthyridin-5-one
4-{1-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]piperidin-4-yl}pyrimidin-2-amine
(2-{[(6-methoxy-2H-1,3-benzodioxol-5-yl)methyl][(2-methylphenyl)methyl]amino}ethyl)dimethylamine
{[2-methanesulfonyl-1-(oxolan-2-ylmethyl)-1H-imidazol-5-yl]methyl}[(1-methyl-1H-imidazol-2-yl)methyl](propan-2-yl)amine
6-{3-[1-(2-ethoxyethyl)-1H-pyrazol-3-yl]phenyl}-N,N-dimethylpyrimidin-4-amine
3-{2-[(2-methoxyethyl)(methyl)amino]ethyl}-8-(oxan-4-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
4-(3-benzyl-1H-1,2,4-triazol-5-yl)-N-(3-chlorophenyl)butanamide
N-ethyl-N-[(5-propyl-1,2,4-oxadiazol-3-yl)methyl]-2-(pyridin-3-yl)acetamide
N-ethyl-N-(2-hydroxyethyl)-6-(4-methoxyphenyl)-7-methyl-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
2-(diethylamino)-1-(4-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)ethan-1-one
2-(2,3-dihydro-1H-inden-1-yl)-N-{[5-(2-methylpropyl)-1,2-oxazol-3-yl]methyl}acetamide
2-[1-(4-methyl-1H-imidazole-5-carbonyl)azetidin-3-yl]pyridine
8-{[1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}-8-azaspiro[4.5]decane-7,9-dione
N-[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]-2-(thiophen-2-yl)-1,3-thiazole-4-carboxamide
N-methyl-5-[4-(1H-pyrazol-1-ylmethyl)piperidine-1-carbonyl]pyridin-2-amine
N-[(1-ethyl-5-oxopyrrolidin-3-yl)methyl]-5-(2-methoxyacetamido)-1-(2-phenylethyl)-1H-1,3-benzodiazole-7-carboxamide
6-methyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-2-(1-methyl-1H-pyrazol-4-yl)-N-(propan-2-yl)quinoline-4-carboxamide
2-(1-benzothiophen-5-yl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
6-ethyl-N4,5-dimethyl-N4-[(5-methyl-1,2-oxazol-3-yl)methyl]pyrimidine-2,4-diamine
1-(2,3-dihydro-1H-inden-2-yl)-4-[(4-fluoro-3-methoxyphenyl)methyl]piperazine
3-(2-{3-ethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}-2-oxoethyl)-4-(3-methylbutyl)piperazin-2-one
1-[(2-fluorophenyl)methyl]-3-hydroxy-3-({methyl[2-(1H-pyrazol-4-yl)ethyl]amino}methyl)piperidin-2-one
[(3R,4R)-4-[(4-ethylpiperazin-1-yl)methyl]-1-{6-methylthieno[2,3-d]pyrimidin-4-yl}pyrrolidin-3-yl]methanol
1-{5,7-dimethylpyrido[2,3-d]pyrimidin-4-yl}-3-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]piperidine
ethyl 2-{4-[(2-methylphenyl)sulfanyl]piperidin-1-yl}-1,3-oxazole-4-carboxylate
1-cyclopropanecarbonyl-N-[4-(3-fluorophenyl)phenyl]pyrrolidine-2-carboxamide
6-methyl-5-{5-[3-(1H-1,2,4-triazol-5-yl)phenyl]-1,2,4-oxadiazol-3-yl}-1,2,3,4-tetrahydro-2,7-naphthyridine
5-{3-[2-(3,4-difluorophenyl)ethyl]piperidine-1-carbonyl}-2-(propan-2-yl)-3,4-dihydropyrimidin-4-one
(3R,5S)-N-(4-fluorophenyl)-1-(naphthalen-2-ylmethyl)-5-(piperidine-1-carbonyl)piperidine-3-carboxamide
methyl 4-({4-[4-(piperidine-1-carbonyl)phenoxy]piperidin-1-yl}methyl)benzoate
2-(5-amino-1,3,4-thiadiazol-2-yl)-N-(1,2,3,4-tetrahydronaphthalen-2-yl)acetamide
(3S,4R)-1-(2-ethoxybenzoyl)-4-(2-methylphenyl)pyrrolidine-3-carboxylic acid
2-{4-[(3-hydroxyazetidin-1-yl)methyl]phenyl}-6-[2-(1H-pyrazol-1-yl)ethyl]-3,4-dihydropyrimidin-4-one
6-(3-chlorophenyl)-N-(cyclopropylmethyl)-7-(3-methylbut-2-en-1-yl)-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
4-(4-chlorophenyl)-N-[2-(N-methylmethanesulfonamido)ethyl]butanamide
2-amino-4-(2-chloro-5-methoxy-4-propoxyphenyl)-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
7-chloro-N-methyl-N-[(3-methylpyridin-2-yl)methyl]-2-(1H-pyrazol-4-yl)quinoline-4-carboxamide
2-chloro-4-[3-(3-chlorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]pyridine
ethyl 4-{[(1R,2S)-2-{imidazo[1,2-b]pyridazine-3-amido}cyclobutyl]amino}piperidine-1-carboxylate
N-[(4-ethyl-1,3-thiazol-2-yl)methyl]-6-[methyl(pyridin-3-ylmethyl)amino]pyridine-3-carboxamide
1-(5-{[2-(dimethyl-1,2-oxazol-4-yl)pyrrolidin-1-yl]methyl}-1-methyl-1H-pyrrol-3-yl)ethan-1-one