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1-[(4aS,8aS)-4a-hydroxy-decahydro-2,7-naphthyridin-2-yl]-3-phenylpropan-1-one
2-[3-(1-ethyl-1H-imidazol-2-yl)piperidin-1-yl]-1,3-benzoxazole
2-(2-ethyl-1H-imidazol-1-yl)-1-[5-(2-methylpropyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl]ethan-1-one
4-{2-[3-hydroxy-3-(hydroxymethyl)piperidine-1-carbonyl]phenyl}-1λ6-thiomorpholine-1,1-dione
N-[(5-benzyl-1,2,4-oxadiazol-3-yl)methyl]-1H-pyrrolo[2,3-b]pyridin-6-amine
{[2-(piperidin-1-yl)-2,3-dihydro-1H-inden-2-yl]methyl}(pyridin-4-ylmethyl)amine
N-(1-hydroxybutan-2-yl)-2-(2-oxoazepan-1-yl)-N-(thiophen-3-ylmethyl)acetamide
2-methoxy-N-[(3-methyloxetan-3-yl)methyl]-2-phenylacetamide
7-methyl-2-(1H-pyrazol-4-yl)-N-[1-(pyridin-4-yl)propyl]quinoline-4-carboxamide
{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl}[(4-methyl-1H-imidazol-5-yl)methyl](oxolan-2-ylmethyl)amine
4-chloro-N,N-diethyl-3-({[2-(5-methylfuran-2-yl)ethyl]carbamoyl}amino)benzamide
N-{[5-(furan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-4-(1H-imidazol-1-yl)benzamide
[(2S)-1-[2-(4-ethylpiperazin-1-yl)-2,3-dihydro-1H-indene-2-carbonyl]pyrrolidin-2-yl]methanol
4-(oxolan-3-yl)-4H,5H,6H,7H-[1,3]thiazolo[5,4-c]pyridin-2-amine
5-({[(8-methoxyquinolin-5-yl)methyl](methyl)amino}methyl)pyrimidin-2-amine
2-(4-chloro-1H-pyrazol-1-yl)-1-[(3R,5R)-3-(hydroxymethyl)-5-(morpholin-4-ylmethyl)piperidin-1-yl]ethan-1-one
{1-[(5-cyclopropyl-1-methyl-1H-pyrazol-4-yl)methyl]-3-(cyclopropylmethyl)piperidin-3-yl}methanol
[(3R,4R)-1-(5-propylthiophene-3-carbonyl)-4-(pyrrolidin-1-ylmethyl)pyrrolidin-3-yl]methanol
5-{[2-(2,3-dihydro-1,4-benzodioxin-6-yl)-1H-imidazol-1-yl]methyl}-3-(propan-2-yl)-1,2-oxazole
N-(1H-1,3-benzodiazol-2-yl)-2-[(2,1,3-benzoxadiazol-5-ylmethyl)(methyl)amino]acetamide
2-[1-(2,4-difluorophenyl)-5-{[methyl(pyridin-3-ylmethyl)amino]methyl}-1H-1,2,4-triazol-3-yl]acetamide
2-ethyl-9-[(2-methyl-1,3-thiazol-4-yl)methyl]-4-phenyl-2,9-diazaspiro[5.5]undecan-3-one
1-{5-[(2,3-difluorophenyl)methyl]-1-[(3-methoxyphenyl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl}piperidin-3-ol
5-methyl-1-propyl-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}-1H-pyrazole-4-carboxamide
(2R,6R)-4-cyclobutanecarbonyl-11-methoxy-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
2-{3-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyrimidin-4-amine
5-({methyl[(3-{2-[4-(2,3,4-trimethoxybenzoyl)piperazin-1-yl]ethoxy}phenyl)methyl]amino}methyl)pyrrolidin-2-one
benzyl[(4-methyl-1,3-thiazol-5-yl)methyl]{[5-methyl-2-(5-methylthiophen-2-yl)-1,3-oxazol-4-yl]methyl}amine
1-[4-(2-methoxyphenyl)pyrimidin-2-yl]-5-methyl-N-[(6-methylpyridin-2-yl)methyl]-1H-pyrazole-4-carboxamide
4-({3-[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl}methyl)-1H-pyrazole-3-carboxylic acid
2-[2-(dimethylamino)ethyl]-9-(2-ethylpyridine-4-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
5-[1-(3-fluorobenzoyl)piperidin-4-yl]-5-(pyridin-3-yl)-3-[2-(thiophen-2-yl)ethyl]imidazolidine-2,4-dione
(2S,4S)-N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-4-{[(2-chlorophenyl)methyl]amino}-1-(propan-2-yl)pyrrolidine-2-carboxamide
5-{1-[3-(naphthalen-1-yl)prop-2-ynoyl]pyrrolidin-2-yl}thiophene-2-carboxamide
4-[1-(2-methylphenyl)-1H-pyrazol-4-yl]-N-(thiophen-3-ylmethyl)pyrimidin-2-amine
1-[(2-chloro-6-fluorophenyl)methyl]-5-(methoxymethyl)-3-(2-methyl-1,3-thiazol-4-yl)-1H-1,2,4-triazole
2-[4-(1,4-dithiepan-6-yl)-1-[(6-methylpyridin-2-yl)methyl]piperazin-2-yl]ethan-1-ol
1-(3,6-dimethyl-1-benzofuran-2-carbonyl)-2-[2-(1H-pyrazol-1-yl)ethyl]piperidine
N-[(3S,4R)-4-(4-methoxyphenyl)-1-{[1,2,3,4]tetrazolo[1,5-a]pyridine-7-carbonyl}pyrrolidin-3-yl]acetamide
3-(3-ethylphenoxy)-N-(3-methyl-1,2,4-thiadiazol-5-yl)azetidine-1-carboxamide
N-ethyl-5-{[3-(3-phenyl-1,2,4-oxadiazol-5-yl)piperidin-1-yl]methyl}pyrimidin-2-amine
(furan-2-ylmethyl)(3-methylbutan-2-yl)(pyridin-2-ylmethyl)amine
(1R,5R)-6-(1H-1,2,3-benzotriazole-5-carbonyl)-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
N-(4-{[4-(oxan-4-yl)piperazin-1-yl]methyl}phenyl)acetamide
2-(2-methylphenyl)-1-[7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carbonyl]pyrrolidine
3-methyl-2-[(3-propyl-1H-pyrazol-5-yl)formamido]butanoic acid
N-{4-[(benzyloxy)methyl]-2-oxo-1,2,3,4-tetrahydroquinolin-7-yl}pyridine-3-carboxamide
(3aR,6aR)-2-cyclohexyl-5-(4-methylpyrimidine-5-carbonyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
(4aS,8aR)-1-[2-(methylamino)ethyl]-6-{pyrazolo[1,5-a]pyrimidine-3-carbonyl}-decahydro-1,6-naphthyridin-2-one
2-(2-amino-4,6-dimethylpyrimidin-5-yl)-N-butyl-N-[(2-fluorophenyl)methyl]acetamide