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4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-N-methyl-N-[1-(pyridin-2-yl)ethyl]benzamide
1-[9-hydroxy-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-methylbutan-1-one
5-cyclopropyl-N-[2-(1-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-1,3,4-oxadiazol-2-amine
(2S)-3-(1H-indol-3-yl)-2-(2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazol-1-yl)propan-1-ol
3,4-diethoxy-N-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}benzamide
1-(4-fluoro-2-{6-[(pyridin-2-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}phenyl)ethan-1-one
1-{3-[(dimethylsulfamoyl)amino]phenyl}-3-[2-(ethanesulfonyl)ethyl]urea
N-[(1R,2S)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]-2-[4-(pyrimidin-2-yl)piperazin-1-yl]acetamide
4-(7-chloro-3,5-dimethyl-1-benzofuran-2-carbonyl)morpholine
8-(2-aminopyrimidin-4-yl)-3-{2-[3-(dimethylamino)pyrrolidin-1-yl]ethyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-(4-chloro-2-ethylphenyl)-4-[2-(methylsulfanyl)ethyl]piperazine-1-carboxamide
N-(2,3-dihydro-1,4-benzodioxin-6-yl)-3-[1-(3-methylthiophene-2-carbonyl)piperidin-4-yl]propanamide
1-(1-benzothiophene-5-carbonyl)-3-(2-methylphenyl)pyrrolidin-3-ol
(3R,9aR)-3-(propan-2-yl)-8-(thiophene-2-carbonyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
(4aS,8aR)-6-(quinolin-2-yl)-decahydro-1,6-naphthyridine-4a-carboxylic acid
N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-2,3-dihydro-1,4-benzodioxine-2-carboxamide
N-{[(2S,4S)-4-fluoro-1-(5-methyl-1-propyl-1H-pyrazole-4-carbonyl)pyrrolidin-2-yl]methyl}-2,5-dimethylfuran-3-carboxamide
4-[3-(2-chlorophenyl)-1H-pyrazol-5-yl]-1-[(2R)-oxolane-2-carbonyl]piperidine
(3R,4R)-1-(5,6-dimethylpyrazin-2-yl)-4-methyl-3-(propan-2-yl)pyrrolidin-3-ol
2-[5-(5-cyclobutyl-1,2,4-oxadiazol-3-yl)-6-methyl-1,2,3,4-tetrahydro-2,7-naphthyridin-2-yl]-5-fluoropyrimidin-4-amine
4-{1-[(dimethyl-1H-1,2,4-triazol-5-yl)methyl]piperidin-3-yl}benzoic acid
3-[(4-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperazin-1-yl)methyl]-1H-indole
3-methyl-1-{2-phenylimidazo[1,2-a]pyridine-6-carbonyl}piperidine
1-{4-[4-cyclopropyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-ethoxyethan-1-one
(2S)-2-amino-1-(4-{4-[(4-phenyl-1,2,3,6-tetrahydropyridin-1-yl)methyl]-1H-1,2,3-triazol-1-yl}piperidin-1-yl)propan-1-one
{[1-(2-methoxyethyl)-1H-imidazol-2-yl]methyl}(methyl)(oxan-4-ylmethyl)amine
2-ethyl-4-[(3-fluoro-2-methylphenyl)methyl]-1-(propan-2-yl)piperazine
9-(4-aminopyridine-2-carbonyl)-2-benzyl-2,9-diazaspiro[5.5]undecan-3-one
2-ethyl-N-{[(2R,3R,5S)-2-(2-fluorophenyl)-5-(hydroxymethyl)-1-methylpyrrolidin-3-yl]methyl}pyrimidine-5-carboxamide
1-[(2-fluorophenyl)methyl]-2-methyl-3-[2-oxo-2-(piperazin-1-yl)ethyl]-4,5,6,7-tetrahydro-1H-indol-4-one
3-(1,3-benzothiazol-2-yl)-1-[3-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]propan-1-one
2-methyl-2-(thiophen-2-ylformamido)-N-[1-(1H-1,2,4-triazol-5-yl)ethyl]propanamide
N-[2-(2,4-difluorophenyl)-1-[1-(3-oxo-2,3-dihydro-1H-indene-1-carbonyl)piperidin-4-yl]ethyl]-N-methylcyclopropanecarboxamide
5-(2,6-difluorophenoxymethyl)-N-(oxan-2-ylmethyl)-1,2-oxazole-3-carboxamide
1-[(3-fluorophenyl)methyl]-4-(4-methyl-1,3-thiazol-2-yl)piperazine
N3-ethyl-N5-(3-methylbutyl)-1-(2-methylpropyl)-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
(3S,4R)-3-(dimethylamino)-4-(propan-2-yl)-N-[2-(propan-2-yl)phenyl]pyrrolidine-1-carboxamide
4-[(1-cyclopentylpiperidin-4-yl)oxy]-3-methoxy-N-[3-(methylsulfanyl)propyl]benzamide
4-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]-1-methyl-2-phenylpiperazine
2-cyclopentyl-2-phenyl-N-[(1s,4s)-4-[4-(pyrrolidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]cyclohexyl]acetamide
N-[2-(dimethylamino)ethyl]-5-[2-(morpholin-2-yl)acetyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
2-{1-[(3-chloro-5-fluoro-4-methoxyphenyl)methyl]piperidin-4-yl}-N-methylacetamide
6-(2-chlorophenyl)-7-methyl-8-oxo-N-pentyl-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
N-(1,3-dimethyl-1H-pyrazol-4-yl)-2-[(1-methylpiperidin-4-yl)(pyridin-4-ylmethyl)amino]acetamide
N-[(2,2-dimethyl-1-phenylcyclopropyl)methyl]-1-methanesulfonyl-N-methylpiperidin-4-amine
methyl N-(2-{4-[(2-methylphenyl)methyl]piperazin-1-yl}-2-oxoethyl)carbamate
3-(4,5-dimethyl-1H-pyrazol-3-yl)-1-[3-(pyridin-3-yl)azetidin-1-yl]propan-1-one
N-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}-N-methyl-2-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}acetamide
1-{3-[2-(2-fluorophenyl)ethyl]piperidin-1-yl}ethan-1-one
2-{3-[(dimethylamino)methyl]-3-hydroxypyrrolidine-1-carbonyl}-5,7-dimethylquinolin-8-ol