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8-[5-(2-ethoxyethyl)-3-(2-methylpropyl)-1H-1,2,4-triazol-1-yl]quinoline
3-[4-(2-methoxyphenyl)piperazin-1-yl]-N,N-dimethylpiperidine-1-sulfonamide
4-ethyl-3-(1-{2-methoxy-5H,6H,7H-cyclopenta[b]pyridine-3-carbonyl}piperidin-4-yl)-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
1-(2,3-dimethylphenyl)-4-{[4-(3-methylphenyl)-4H-1,2,4-triazol-3-yl]methyl}piperazine
N-{1,9-dioxaspiro[5.5]undecan-4-yl}-1,2,3,4-tetrahydroquinoline-6-carboxamide
(3S,4S)-1-{[7-methyl-2-(thiophen-2-yl)quinolin-3-yl]methyl}piperidine-3,4-diol
(1S,4S)-2-{[5-(pyrimidin-2-ylsulfanyl)furan-2-yl]methyl}-2-azabicyclo[2.2.1]heptane
3-(3-chloro-2-ethoxyphenyl)-1-cyclopropyl-1-[(3-hydroxyphenyl)methyl]urea
4-(1,3-dimethyl-1H-pyrazol-4-yl)-N-[(4-methoxyphenyl)methyl]-N-methylpyrimidin-2-amine
3-{4-[2-methyl-6-(morpholin-4-yl)pyrimidin-4-yl]piperidin-1-yl}propan-1-ol
methyl (2R,4S)-4-hydroxy-1-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]piperidine-2-carboxylate
4-{5-[(cyclohexylmethyl)sulfanyl]-4-(oxolan-2-ylmethyl)-4H-1,2,4-triazol-3-yl}-1-[(4-methoxyphenyl)methyl]piperidine
3-(5-ethyl-1-methyl-1H-1,2,4-triazol-3-yl)-1-methyl-1-{[1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}urea
N-[2-(4-fluorophenyl)ethyl]-2-[4-methyl-3-oxo-2-(propan-2-yl)piperazin-1-yl]acetamide
(1S,9R)-11-(3-propyl-1H-pyrazole-5-carbonyl)-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-6-one
4-(2-methoxyethyl)-N-[3-(2-methyl-1,3-thiazol-4-yl)phenyl]piperazine-1-carboxamide
2-(5-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-(2-{4-methyl-5H,6H,7H-cyclopenta[d]pyrimidin-2-yl}ethyl)acetamide
1-[(3R,4S)-3-amino-4-(4-methoxyphenyl)pyrrolidin-1-yl]-3-(1-methyl-1H-pyrazol-5-yl)propan-1-one
2-(5-{[3-(thiophene-2-carbonyl)piperidin-1-yl]methyl}-1,2,4-oxadiazol-3-yl)pyridine
8-methoxy-2-{[2-(1H-pyrazol-1-ylmethyl)-1,4-oxazepan-4-yl]methyl}quinoline
4-{[5-(3-methyl-1,2-oxazol-5-yl)furan-2-yl]sulfonyl}-2-(trifluoromethyl)morpholine
(2R,3S,6R)-3-(3,5-difluorophenyl)-5-(3,6-dimethylpyrazin-2-yl)-1,5-diazatricyclo[5.2.2.02,6]undecane
3-(5-{1-[(2-chlorophenyl)methyl]-1H-imidazol-2-yl}thiophen-3-yl)prop-2-yn-1-ol
N-(1-{1-[(2-hydroxy-4-methoxyphenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)benzamide
(3aS,6aS)-2-[5-fluoro-4-(methylamino)pyrimidin-2-yl]-5-methanesulfonyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-[(7-fluoro-2-oxo-1,2-dihydroquinolin-3-yl)methyl]-3-phenyl-1H-pyrazole-4-carboxamide
3-methyl-6-(5-{spiro[2.5]octan-1-yl}-1,2,4-oxadiazol-3-yl)pyridazine
2-{[4-(4-fluorophenyl)piperazin-1-yl]methyl}-8-methoxyquinoline
N-[1-(4-chlorophenyl)-5-oxopyrrolidin-3-yl]-5-methyl-1-propyl-1H-pyrazole-4-carboxamide
{1-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]-4-{[2-(trifluoromethyl)phenyl]methyl}piperidin-4-yl}methanol
2-[4-(3-methylpyridin-4-yl)piperazin-1-yl]-4-(3,3,3-trifluoropropyl)pyrimidine
5-[5-(furan-2-ylmethyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl]-3-phenyl-1,2-oxazole
1-({2-[(2-chlorophenyl)methoxy]-6-methylquinolin-3-yl}methyl)piperidin-4-ol
2-methyl-3-{4-[4-(2-methylpropyl)-1H-1,2,3-triazol-1-yl]piperidine-1-carbonyl}-1,8-naphthyridine
8-(2-amino-2-methylpropyl)-3-(2-ethylbutyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-[bis(4-fluorophenyl)methyl]-4-(1H-imidazol-2-ylmethyl)piperazine
6-[({2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}amino)methyl]-1,4-oxazepan-6-ol
3,5,7-trimethyl-N-[1-(oxolan-2-ylmethyl)piperidin-4-yl]-1H-indole-2-carboxamide
9-[(2-aminopyridin-3-yl)methyl]-2-(2-phenylethyl)-2,9-diazaspiro[5.5]undecan-3-one
4,6-dimethyl-2-{3'-oxo-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-1-yl}pyridine-3-carbonitrile
[(3R,4R)-4-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-1-[(5-ethylfuran-2-yl)methyl]pyrrolidin-3-yl]methanol
8-methyl-1-(3-methylbutyl)-3-[3-(pyridin-4-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
8-[6-(propan-2-yl)-2-(trifluoromethyl)pyrimidin-4-yl]-1-oxa-8-azaspiro[4.5]decane
4-{[(1-butyl-3-methyl-1H-1,2,4-triazol-5-yl)methyl]sulfanyl}pyridine
N,N-dimethyl-2-{methyl[(4-methyl-1H-imidazol-5-yl)methyl]amino}propanamide
1-{5-cyclobutanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-2-(pyrrolidin-1-yl)ethan-1-one
1-benzyl-N,N-dimethyl-5-[(6-methyl-4-oxo-4H-chromen-3-yl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-[(3R,4R)-4-(4-methylpiperazin-1-yl)oxolan-3-yl]-2-propyl-1,3-thiazole-4-carboxamide
6-methyl-1-({7-methylimidazo[1,2-a]pyridin-2-yl}methyl)-4-(trifluoromethyl)-1,2-dihydropyridin-2-one
N-[2-(azepan-1-yl)ethyl]-N-ethyl-6-fluoro-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide