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2-{5-[(4,5-dimethylfuran-2-yl)methyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}-1-propyl-1H-imidazole
1-[1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-4-[2-(pyrrolidin-1-yl)ethyl]piperazine
5-(oxolan-2-yl)-N-{pyrazolo[1,5-a]pyrimidin-3-ylmethyl}thiophene-2-carboxamide
3-propyl-4-[1-(thiophene-2-carbonyl)piperidin-4-yl]morpholine
methyl({[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}){[2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]methyl}amine
8-(2-propoxyacetyl)-2-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
2-amino-4-[2-(benzyloxy)phenyl]-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
2-{3-[2-(2,6-difluorophenyl)ethyl]piperidine-1-carbonyl}-6-methylpyridine
(3S,4R)-1-(1,4-dithiepan-6-yl)-4-(pyridin-3-yl)pyrrolidine-3-carboxylic acid
1-(cyclopropylmethyl)-4-[4-ethyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
N-methyl-N-[2-(oxan-2-yl)ethyl]-2-(trifluoromethyl)benzamide
4-(3-chlorophenyl)-3-(1-methyl-5-oxopyrrolidin-3-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
N-[2-(2-methylpropanesulfonyl)ethyl]-3-(pyridin-2-yl)-1H-pyrazole-5-carboxamide
1-[(4-chlorophenyl)methyl]-N-[(1-ethylpyrrolidin-2-yl)methyl]-1H-1,2,3-triazole-4-carboxamide
N-{[(2S,4S)-4-fluoropyrrolidin-2-yl]methyl}-3-{[(3R)-3-methylpiperazin-1-yl]sulfonyl}benzamide
(1S,4S)-2-[2-(methylsulfanyl)phenyl]-5-{[3-(trifluoromethyl)phenyl]methyl}-2,5-diazabicyclo[2.2.1]heptan-3-one
2-{[methyl({1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}methyl)amino]methyl}phenol
N-(2-methoxyethyl)-2-methyl-N-(thiophen-3-ylmethyl)imidazo[1,2-a]pyridine-6-carboxamide
5-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl]isoquinoline
N-({1-[(2,3-dimethoxyphenyl)methyl]pyrrolidin-3-yl}methyl)-2,2-difluoroacetamide
6-[2-(piperidin-1-ylmethyl)phenoxy]pyridine-3-carbonitrile
5-[2-(propan-2-yl)-1,3-thiazole-4-carbonyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxylic acid
2-[1-(2,2-diphenylethyl)-3-oxopiperazin-2-yl]-N-(2-methoxyethyl)acetamide
1-[2-methyl-4-(1,2,3,6-tetrahydropyridin-1-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl]-2-(1H-pyrrol-1-yl)ethan-1-one
N-methyl-5-{[(6-methylpyridin-3-yl)oxy]methyl}-N-[2-(oxan-2-yl)ethyl]-1,2-oxazole-3-carboxamide
N-[(2S,4R,6R)-2-(1-ethyl-1H-pyrazol-4-yl)-6-(4-fluoro-3-methoxyphenyl)oxan-4-yl]acetamide
1-[2-(pyridin-4-yl)ethyl]-3-(1,3,4-thiadiazol-2-yl)urea
3-[(3-aminopyrrolidin-1-yl)sulfonyl]-N-methyl-N-[2-(1,2,4-oxadiazol-3-yl)ethyl]benzamide
4-[4-(4-fluorophenyl)-1H-1,2,3-triazol-1-yl]-N-(4-methoxyphenyl)piperidine-1-carboxamide
4-({1-[(4-methanesulfonylphenyl)methyl]piperidin-2-yl}methyl)morpholine
1-[(5-ethylpyridin-2-yl)methyl]-4-[2-(methylsulfanyl)ethyl]piperazine
N,N-diethyl-1-[2-(5-oxo-5,6-dihydro-1,6-naphthyridin-6-yl)acetyl]piperidine-3-carboxamide
N-benzyl[(2,4-dimethyl-6-oxo-1,6-dihydropyridin-3-yl)amino]sulfonamide
2-methyl-N-[1-(5-methyl-1H-1,2,4-triazol-3-yl)ethyl]-5-phenylpyrazolo[1,5-a]pyrimidin-7-amine
{1-[1-(cyclopent-1-ene-1-carbonyl)piperidin-4-yl]-2-phenylethyl}(methyl)(pyridin-4-ylmethyl)amine
1-{[1-({3-[(2-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)piperidin-4-yl]methyl}pyrrolidin-2-one
1-(diethylamino)-3-[2-methoxy-4-({[2-(4-methylpiperazin-1-yl)ethyl]amino}methyl)phenoxy]propan-2-ol
N-(1-cyanocyclopentyl)-5-(2-methylpropyl)-1,2-oxazole-3-carboxamide
2-methyl-N-[4-(trifluoromethyl)pyrimidin-2-yl]-4,5,6,7-tetrahydro-1,3-benzothiazol-4-amine
1-[1-(2,3-dihydro-1H-inden-5-yl)-3-(oxan-4-yl)-1H-1,2,4-triazol-5-yl]ethan-1-ol
N-[2-(2-ethylphenoxy)ethyl]-N-methyl-2-(pyrrolidin-1-yl)acetamide
1-(4-methoxyphenyl)-4-{9-oxo-octahydro-1H-pyrazino[1,2-a]piperazin-2-yl}butane-1,4-dione
N-[(4-ethyl-1,3-thiazol-2-yl)methyl]-6-[3-(methoxymethyl)pyrrolidin-1-yl]pyridine-3-carboxamide
N-{[1-(2-acetylbenzoyl)piperidin-3-yl]methyl}-2-(2-methoxyphenoxy)acetamide
1-{1-oxo-1-[4-(pyrimidin-2-yloxy)piperidin-1-yl]propan-2-yl}pyrrolidin-2-one
4-{[2-(3-hydroxypropyl)-3-oxo-2,9-diazaspiro[5.5]undecan-9-yl]methyl}benzonitrile
2-amino-4-(1-ethyl-3-methyl-1H-pyrazol-4-yl)-6-(4-hydroxy-3-methoxyphenyl)pyridine-3-carbonitrile
3,5-dimethyl-N-(1,4-oxazepan-6-ylmethyl)benzene-1-sulfonamide
(2S)-N-(4-methoxy-3-pentanamidophenyl)oxolane-2-carboxamide
3-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]-1-(4-methyl-1,2,3-thiadiazole-5-carbonyl)piperidine