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(3S,4R)-4-(2,3-dimethoxyphenyl)-1-(3,6-dimethylpyrazin-2-yl)pyrrolidine-3-carboxylic acid
[(5-ethylpyridin-2-yl)methyl](methyl){[5-(oxolan-3-ylmethyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}amine
3-{5-[4-methyl-2-(propan-2-yl)-1,3-thiazol-5-yl]-1,2,4-oxadiazol-3-yl}pyridazine
(2S,4S)-1-(2,3-dihydro-1H-inden-2-yl)-4-{[(4-methoxynaphthalen-1-yl)methyl]amino}-N-methylpyrrolidine-2-carboxamide
5-[(1R,5R)-3-azabicyclo[3.3.1]nonane-3-carbonyl]-2-methylphenol
2-[4-(cyclopropanesulfonyl)morpholin-3-yl]-N-[2-(5-ethyl-1,2,4-oxadiazol-3-yl)ethyl]acetamide
2-methyl-5-(4-{[2-(propan-2-yl)-1,3-oxazol-4-yl]methyl}piperazin-1-yl)-2,3-dihydropyridazin-3-one
5-(3-cyclohexyl-1H-pyrazol-4-yl)-1-(oxolan-3-yl)-4-phenyl-1H-imidazole
2-(2-ethyl-1H-imidazol-1-yl)-N-{pyrazolo[1,5-a]pyridin-3-ylmethyl}acetamide
2-[(2-chlorophenyl)methyl]-4-[2-(1H-pyrazol-1-yl)benzoyl]morpholine
(3R,4R)-1-{[4-(2-hydroxyethoxy)phenyl]methyl}-3-methyl-4-(oxan-4-yl)piperidin-4-ol
N-[2-(4-fluorophenyl)ethyl]-N-{[2-(3-hydroxypiperidin-1-yl)-5,8-dimethoxyquinolin-3-yl]methyl}furan-3-carboxamide
N-(1H-indol-4-ylmethyl)-6-oxo-1-[3-(2-oxopyrrolidin-1-yl)propyl]piperidine-3-carboxamide
1-[1-(5-ethylpyrimidin-2-yl)piperidin-4-yl]piperidin-4-ol
N-{2-[4-(hydroxymethyl)piperidin-1-yl]-5,6,7,8-tetrahydroquinazolin-5-yl}-2-(propan-2-yloxy)acetamide
2-[4-methyl-2-(1H-pyrazol-1-yl)phenyl]pyridine-3-carbonitrile
5-{2-[7-(cyclobutylmethyl)-6-oxo-2,7-diazaspiro[4.5]decan-2-yl]-2-oxoethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-[2-(2-oxo-1,3-oxazolidin-3-yl)ethyl]-2-(3-phenylpropyl)-1,3-benzoxazole-5-carboxamide
2,8-dimethyl-4-{1H,2H,3H,4H-pyrrolo[1,2-a]pyrazine-2-carbonyl}quinoline
2-{3-[4-(4-methylphenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}pyridin-4-amine
1-[(4-fluorophenyl)methyl]-4-(4-methyl-1,3-thiazol-2-yl)-1,4-diazepane
(1R,5R)-6-benzyl-3-(oxane-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
5-(3-ethyl-5-methyl-1,2-oxazole-4-carbonyl)-N-(2-hydroxyethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
N-[(3S,4R)-1-(1-benzofuran-3-carbonyl)-4-(4-methylphenyl)pyrrolidin-3-yl]acetamide
1-[4-(2-chlorophenoxy)piperidin-1-yl]-2-(morpholin-4-yl)ethan-1-one
4-{4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]benzoyl}-2-ethyl-1-(propan-2-yl)piperazine
2-(dimethyl-1H-1,2,4-triazol-1-yl)-1-[1-(2-fluorophenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]ethan-1-one
(4aR,7aS)-1-cyclobutanecarbonyl-4-[(dimethyl-1H-1,2,4-triazol-5-yl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-(1,3-benzothiazol-2-ylmethyl)-6-[(diethylamino)methyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide
2-methyl-N-({1-[(3-methyl-1H-indol-2-yl)methyl]piperidin-4-yl}methyl)propanamide
N-[2-(1H-imidazol-4-yl)ethyl]-5-(propan-2-yl)-1,3-oxazole-4-carboxamide
N-[5-(3-methyl-1H-pyrazol-1-yl)quinolin-8-yl]acetamide
3-(2-chlorophenyl)-N-[(2-methyl-1,3-thiazol-4-yl)methyl]-3-phenylpropanamide
2-(3,4-dichlorophenyl)-4-(1,3-thiazol-2-yl)morpholine
3,5-dimethyl-N-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]-4-oxo-3H,4H-thieno[2,3-d]pyrimidine-6-carboxamide
2-[(3S,4R)-4-amino-1-[4-(1H-pyrazol-1-yl)benzoyl]pyrrolidin-3-yl]ethan-1-ol
2-{[(1S,6R)-3-methyl-3,9-diazabicyclo[4.2.1]nonan-9-yl]methyl}quinolin-4-ol
N-[3-(2-ethoxyphenyl)propyl]-6-ethyl-1,5-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
N-(2-{1-[2-(dimethylamino)ethyl]-5-oxopyrrolidin-2-yl}ethyl)-2-(1H-imidazol-2-yl)benzamide
(3S,9aR)-8-(4-chlorobenzenesulfonyl)-3-[(4-chlorophenyl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
dimethyl[(5-{1-oxa-8-azaspiro[4.6]undecane-8-carbonyl}furan-2-yl)methyl]amine
1-{[2-(2-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-(3-methoxybenzoyl)piperazine
methyl 2-[2-(2-methylpropyl)-3-oxo-2,8-diazaspiro[4.5]decan-8-yl]-2-phenylacetate
[3-(2-phenoxyethyl)-1-(9H-purin-6-yl)piperidin-3-yl]methanol
1-{1-[(3,4-dimethoxyphenyl)methyl]piperidin-3-yl}-4-(2-methoxyphenyl)piperazine
2-(methoxymethyl)-1-{[3-(methylsulfanyl)phenyl]methyl}piperidine
2-(3-ethoxyphenyl)-2-{methyl[2-(morpholin-4-yl)ethyl]amino}acetic acid
4-{1-[3-(4-methoxyphenyl)-1H-pyrazole-5-carbonyl]piperidin-4-yl}morpholine
2-methoxy-6-[5-(methoxymethyl)-3-methyl-1H-pyrazol-4-yl]-N,N-bis(propan-2-yl)benzamide
N-[1-(5-{[(2-fluorophenyl)methyl]sulfanyl}-4-methyl-4H-1,2,4-triazol-3-yl)-2-phenylethyl]-2,3,4-trimethoxybenzamide