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2,2,6,6-tetramethyl-N-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]piperidin-4-amine
1-(2-amino-5-ethylpyrimidin-4-yl)-3-[(dimethylamino)methyl]pyrrolidin-3-ol
1-[4-(benzenesulfonyl)piperazin-1-yl]-2-{8-methylimidazo[1,2-a]pyridin-3-yl}ethan-1-one
2-cyclopropyl-9-(2-ethoxyacetyl)-4-phenyl-2,9-diazaspiro[5.5]undecan-3-one
3-(4-methylphenoxymethyl)-1-(1H-pyrrole-3-carbonyl)piperidine
2-[(5-methylfuran-2-yl)methyl]-7-[(3-methylphenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
4-chloro-1,5-dimethyl-N-{2-[(trifluoromethyl)sulfanyl]ethyl}-1H-pyrazole-3-carboxamide
1-[1-(2,4-dimethylbenzoyl)piperidin-4-yl]-N-(oxolan-2-ylmethyl)piperidine-4-carboxamide
3-[2-(2,6-difluorophenyl)ethyl]-1-[2-(1H-1,2,4-triazol-3-yl)benzoyl]piperidine
N-[(3-methylpyridin-2-yl)methyl]-2-[3-(trifluoromethyl)phenoxymethyl]-1,3-oxazole-4-carboxamide
4-methyl-2-({1-[3-(trifluoromethyl)phenyl]-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl}methyl)-1H-imidazole
N-(1-ethyl-1H-pyrazol-5-yl)-2-{4-[5-(3-methyl-1,2,4-oxadiazol-5-yl)pyridin-2-yl]-1H-pyrazol-1-yl}acetamide
methyl 5-{4-[(4-fluorophenyl)methyl]-5-oxo-3-(propan-2-yl)-1,4-diazepan-1-yl}-5-oxopentanoate
1-(furan-2-ylmethyl)-N-[(4-oxo-3,4-dihydroquinazolin-2-yl)methyl]piperidine-3-carboxamide
3-(1,3-dimethyl-1H-pyrazol-4-yl)-1-[(5-methylpyrazin-2-yl)methyl]urea
2-(4-{[6-(piperidine-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}piperazin-1-yl)pyrimidine
8-(2-methoxypyridine-3-carbonyl)-1-methyl-3-phenyl-1,8-diazaspiro[4.5]decane
5-[(1,3-benzothiazol-2-ylmethyl)amino]-N-methyl-1-(2-phenylethyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
(2S,4R)-1-benzyl-4-({[3-(benzyloxy)phenyl]methyl}amino)-N-methylpyrrolidine-2-carboxamide
1-(2-chloro-6-fluoro-3-methylbenzoyl)-3-(2-fluorophenyl)pyrrolidine
5-{2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}-10-methoxy-3,4,5,6-tetrahydro-2H-1,5-benzoxazocine
(2R,3R,6R)-5-[(1R,5S,6R)-3-azabicyclo[3.1.0]hexane-6-carbonyl]-3-(4-methylphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
1-[1-(1,3-benzoxazol-2-yl)piperidin-4-yl]-N-tert-butylpiperidine-3-carboxamide
N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
6-amino-N-({1-[(4-methyl-1H-imidazol-5-yl)methyl]piperidin-3-yl}methyl)pyridine-3-carboxamide
4-[2-(ethoxymethyl)-7-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]thiomorpholine
1-[(2R)-3,4-dihydro-2H-1-benzopyran-2-ylmethyl]-3-(dimethyl-1,2-oxazol-4-yl)urea
3-{1-[2-(2,3-dihydro-1H-isoindol-2-yl)acetyl]piperidin-3-yl}benzoic acid
5-(2,3-difluorophenyl)-1-[(1-methylpyrrolidin-3-yl)methyl]-4-phenyl-1H-imidazole
8-[(2S)-3-hydroxy-2-methylpropyl]-2-[(3-methoxyphenyl)methyl]-2,8-diazaspiro[4.5]decan-3-one
2-(2H-1,3-benzodioxol-5-yloxy)-1-{3-[(dimethylamino)methyl]-3-hydroxypyrrolidin-1-yl}ethan-1-one
(3S,4R)-3-acetamido-N-ethyl-4-(5-methylfuran-2-yl)pyrrolidine-1-carboxamide
N-[(4-chloro-3-methyl-1H-pyrazol-5-yl)methyl]-N-[(1-methyl-1H-imidazol-2-yl)methyl]cyclopropanamine
2-(3,4,5-trimethoxyphenyl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
3-{4-[(2,3,4-trimethoxyphenyl)methyl]piperazin-1-yl}propanamide
N-[(4-phenyloxan-4-yl)methyl]quinoline-5-carboxamide
5-[8-(cyclopropylmethyl)-9-oxo-2,8-diazaspiro[5.5]undecane-2-carbonyl]pyridine-2-carbonitrile
2-(3-fluoro-4-hydroxyphenyl)-1-[4-(pyridin-3-ylmethoxy)piperidin-1-yl]ethan-1-one
3-(1-ethyl-1H-imidazol-2-yl)-1-[(3-methoxyphenyl)methyl]piperidine
2-[4-(1,3-benzothiazol-2-ylmethyl)-1-[(2-ethoxyphenyl)methyl]piperazin-2-yl]ethan-1-ol
5-{3-[4-(2-methylphenyl)piperazin-1-yl]piperidine-1-carbonyl}-1H-1,2,3-benzotriazole
5-fluoro-2-(3-methoxyphenyl)-N-methylpyrimidin-4-amine
8-{[3-(benzyloxy)phenyl]methyl}-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
3-[(2-fluorophenyl)formamido]-N-[3-(1H-1,2,4-triazol-1-yl)propyl]propanamide
4-{2-[(1-benzylpyrrolidin-3-yl)carbamoyl]ethyl}-N,N-dimethylpiperidine-1-carboxamide
(2S,4R)-4-{[(3,5-dimethoxyphenyl)methyl]amino}-N-ethyl-1-(naphthalen-2-ylmethyl)pyrrolidine-2-carboxamide
1-cyclopentyl-N-[3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)propyl]piperidine-3-carboxamide
4-[1-(2,3-dihydro-1H-inden-2-yl)-3-methyl-1H-1,2,4-triazol-5-yl]benzene-1-sulfonamide
4-[4-(3-hydroxyprop-1-yn-1-yl)thiophen-2-yl]-3-methyl-1-(2-methylphenyl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
dimethyl(2-{[(3-methylthiophen-2-yl)methyl]({[3-(1H-pyrazol-1-yl)phenyl]methyl})amino}ethyl)amine