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1-(3,5-dimethylphenyl)-4-[4-(pyridin-3-yl)pyrimidin-2-yl]piperazin-2-one
6-(cyclopropylmethoxy)-1-[(3-methoxyphenyl)methyl]-4-(1,3-thiazole-4-carbonyl)-1,4-diazepan-2-one
N-[2-(6-fluoro-1H-1,3-benzodiazol-2-yl)ethyl]-1-(2-methoxyacetyl)piperidine-4-carboxamide
N-{[3-fluoro-5-(trifluoromethyl)phenyl]methyl}-3-methoxy-2,2-dimethylpropanamide
N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-1-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidine-5-carboxamide
ethyl 5-[ethyl(2,2,2-trifluoroethyl)carbamoyl]-1H-imidazole-4-carboxylate
N-({5-cyclobutanecarbonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-4-methylpyrimidine-5-carboxamide
1-(2,5-dihydro-1H-pyrrole-2-carbonyl)-N-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]piperidine-4-carboxamide
(2-{2-[1-(2-ethoxypyridine-3-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}ethyl)dimethylamine
N-{4-[4-(benzylamino)piperidin-1-yl]phenyl}-2-phenoxyacetamide
[(3R,4R)-1-[(2,5-difluorophenyl)methyl]-4-(pyrrolidin-1-ylmethyl)pyrrolidin-3-yl]methanol
N-{2-methyl-2H,4H,5H,6H-cyclopenta[c]pyrazol-3-yl}-2-{1H-pyrazolo[3,4-b]pyridin-1-yl}acetamide
ethyl 5-[3-(methylcarbamoyl)-6-oxo-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-4-yl]-2-oxo-2,3-dihydro-1H-imidazole-4-carboxylate
N-cyclohexyl-2-{1-[(2,4-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
ethyl 3-[(3-chlorophenyl)methyl]-1-[3-(6-oxo-1,4,5,6-tetrahydropyridazin-3-yl)propanoyl]piperidine-3-carboxylate
N-[2-(diethylamino)ethyl]-N-methyl-3-(morpholine-4-carbonyl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-[1-(morpholine-4-carbonyl)piperidin-4-yl]-1-(propan-2-yl)-1H-pyrazole-4-carboxamide
3-cyclobutyl-1-{[2-(2-fluoro-4-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1H-1,2,4-triazole
1-cyclohexyl-4-{2-[3-oxo-1-(propan-2-yl)piperazin-2-yl]acetyl}piperazin-2-one
1-(1-{[2-(trifluoromethyl)phenyl]methyl}-1H-1,2,3-triazole-4-carbonyl)piperidine-3-carboxamide
(3R)-3-cyclopropyl-4,4-dimethyl-1-(6-methylpyridine-3-carbonyl)pyrrolidin-3-ol
6-[(4-cyclohexyl-4H-1,2,4-triazol-3-yl)methyl]-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
2-(1-{[3-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-methyl-1H-pyrazol-4-yl]methyl}piperidin-4-yl)-1,3-benzoxazole
2-[(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)amino]-N-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)acetamide
5-(1H-1,3-benzodiazol-1-ylmethyl)-N-{pyrazolo[1,5-a]pyridin-3-ylmethyl}-1H-pyrazole-3-carboxamide
N-[3-(4-methyl-1,3-thiazol-2-yl)propyl]imidazo[2,1-b][1,3]thiazole-6-carboxamide
1-{2,6-dimethylimidazo[1,2-a]pyridine-3-carbonyl}-3-(2-methoxyphenoxy)azetidine
2-{imidazo[2,1-b][1,3]thiazol-6-yl}-N-methyl-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}acetamide
2-{2-[4-(2-methylphenyl)-4H-1,2,4-triazol-3-yl]ethyl}phenol
4-[7-(1-phenylcyclopropanecarbonyl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl]morpholine
3-[(3R,4S)-1-(2,6-difluoro-3-methoxybenzoyl)-4-(morpholin-4-yl)piperidin-3-yl]propan-1-ol
2-{3-cyclopropyl-5-[2-phenyl-1-(1H-1,2,3,4-tetrazol-1-yl)ethyl]-1H-1,2,4-triazol-1-yl}pyridine
1-[2-(3-fluorophenyl)ethyl]-6-oxo-N-[3-(propan-2-yloxy)propyl]piperidine-3-carboxamide
(1R,5R)-3-benzoyl-6-[(2-fluoro-4-methoxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane
7-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}-1,2,3,4-tetrahydroisoquinoline
(2S,4S)-1-benzyl-4-{[(2,6-difluorophenyl)methyl]amino}-N-ethylpyrrolidine-2-carboxamide
4-(2,4-dichlorophenyl)-6-methoxypyrimidin-2-amine
5-{4-[(4-fluorophenyl)methyl]piperazine-1-carbonyl}-2-(pyrrolidin-1-yl)pyrimidine
1-{1-[2-(dimethylamino)-4-methylpyrimidine-5-carbonyl]piperidin-4-yl}piperidin-4-ol
N-[2-(3-phenylpyrrolidin-1-yl)ethyl]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
2-{2-[(2S,4R)-4-(dimethylamino)-2-(hydroxymethyl)pyrrolidin-1-yl]-2-oxoethyl}-4-methyl-1,2-dihydrophthalazin-1-one
N,1-dimethyl-N-[(4-phenoxyphenyl)methyl]-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
5-(2-fluorophenoxymethyl)-N-(2-phenoxyethyl)-1H-pyrazole-3-carboxamide
2-(3-methoxypropyl)-8-(2-propyl-1,3-thiazole-4-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
(3aS,6aS)-N-(4-chloro-2-fluorophenyl)-octahydropyrrolo[2,3-c]pyrrole-1-carboxamide
2-{[(1R,3S)-1,3-dihydroxy-7-azaspiro[3.5]nonan-7-yl]methyl}-3,5-dimethyl-1,4-dihydropyridin-4-one
N-[(1-ethylpyrrolidin-2-yl)methyl]-6-(4H-1,2,4-triazol-4-yl)pyridine-3-carboxamide
4-[2-(1H-pyrazol-1-yl)ethyl]-1-(2,3,4,5-tetrahydro-1-benzoxepine-4-carbonyl)piperidine
ethyl 2-[(3aS,6aR)-2-oxo-3-(pyridin-2-ylmethyl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-5-yl]pyridine-3-carboxylate
N-ethyl-5-{[methyl(2,2,6,6-tetramethylpiperidin-4-yl)amino]methyl}pyrimidin-2-amine