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N-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]-4-(1H-1,2,3,4-tetrazol-1-yl)benzamide
3-{[4-(furan-2-carbonyl)-1,4-diazepan-1-yl]methyl}-8-methyl-1,2-dihydroquinolin-2-one
2-(4-{[3-(2-hydroxyethyl)-4-[(2-methylphenyl)methyl]piperazin-1-yl]methyl}phenoxy)ethan-1-ol
1-{[1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}-3-(3-methylthiophene-2-carbonyl)piperidine
4-(2-hydroxybenzoyl)-1-(2-phenylphenyl)piperazin-2-one
N-[(3S,4S)-4-hydroxy-1,1-dioxo-1λ6-thiolan-3-yl]-3-(3-hydroxy-3-methylbutyl)-N-(2-hydroxyethyl)benzamide
(2S)-2-amino-3-hydroxy-1-[4-(naphthalen-2-yl)piperazin-1-yl]propan-1-one
4-(3-tert-butyl-1H-1,2,4-triazol-5-yl)-N-(pyridin-4-ylmethyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
(1R,6S)-3-(5-methanesulfonyl-2-methylpyrimidin-4-yl)-9-methyl-3,9-diazabicyclo[4.2.1]nonane
8-[3-(dimethyl-1,2-oxazol-4-yl)propanoyl]-2-(2-methoxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
ethyl 5-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propanoyl]-1-[(4-methoxyphenyl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
N-[2-(dimethylamino)ethyl]-N-methyl-3-{[1-(3-phenylprop-2-ynoyl)piperidin-4-yl]oxy}benzamide
1-(3-{5-[(dimethylamino)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-2-(pyridin-2-ylsulfanyl)ethan-1-one
methyl({[3-(methylsulfanyl)phenyl]methyl}){4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}amine
3-(2-hydroxyethyl)-4-{pyrazolo[1,5-a]pyridine-7-carbonyl}piperazin-2-one
N-(2-fluorophenyl)-3-(1-{[4-methoxy-3-(methoxymethyl)phenyl]methyl}piperidin-3-yl)propanamide
N-methyl-2-(2-oxo-1,3-oxazolidin-3-yl)-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]acetamide
2-(2-chloro-5-methylphenyl)-2-{methyl[(3-methyl-1,2-oxazol-5-yl)methyl]amino}acetic acid
N-{2-[(dimethylcarbamoyl)methyl]phenyl}-3-(morpholin-4-yl)azetidine-1-carboxamide
7-(propan-2-yl)-2-[4-(1H-1,2,4-triazol-1-yl)butanoyl]-2,7-diazaspiro[4.5]decan-6-one
N-(2,1,3-benzoxadiazol-5-ylmethyl)-N-methyl-2-(2-methyl-1,3-thiazol-4-yl)acetamide
N,N-dimethyl-5-(5-methyl-1H-indol-3-yl)furan-2-carboxamide
3-cyclopropyl-N-methyl-N-{[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}-1H-pyrazole-5-carboxamide
N-cyclopropyl-4-fluoro-N-{[5,6,7-trimethoxy-2-(2-methylphenyl)quinolin-3-yl]methyl}benzamide
1-[(3S,4S)-3-hydroxy-4-(4-methylpiperazin-1-yl)pyrrolidin-1-yl]-3-methylbut-2-en-1-one
N-[(3-methoxyphenyl)methyl]-N-(prop-2-en-1-yl)-2-[(propan-2-yl)amino]pyrimidine-5-carboxamide
2-ethyl-9-(4-methylpyrimidine-5-carbonyl)-4-phenyl-2,9-diazaspiro[5.5]undecane
N-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-5-fluoro-4-(morpholin-4-yl)pyrimidin-2-amine
9-[2-(morpholin-4-yl)ethyl]-2-(2-phenylethyl)-2,9-diazaspiro[5.5]undecan-3-one
2-(3-methoxypropyl)-9-[4-(2-methylpropyl)benzoyl]-2,9-diazaspiro[5.5]undecan-3-one
2-ethyl-6-methyl-5-{2-[(1R,5R)-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]-2-oxoethyl}-3,4-dihydropyrimidin-4-one
1-[3-(3-methylbutyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-2-(2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethan-1-one
2-methoxy-N-{1-[1-(3-methyl-5,6-dihydro-1,4-dioxine-2-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}-2-phenylacetamide
1-(3-chlorobenzoyl)-4-phenoxypiperidine-4-carboxylic acid
1-ethyl-N-{1-[(2-methylphenyl)methyl]cyclopropyl}-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
(3S,4R)-1-(3-ethyl-5-methyl-1,2-oxazole-4-carbonyl)-4-(3-methoxyphenyl)pyrrolidine-3-carboxylic acid
(3aR,6aR)-2-cyclopentanecarbonyl-5-(5-methyl-1,3,4-thiadiazol-2-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N,N-dimethyl-6-{4-[1-(pyrrolidin-1-yl)ethyl]piperidin-1-yl}pyrimidin-4-amine
2-(dimethylamino)-7-[5-methyl-2-(methylamino)benzoyl]-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
4-(3,4-dimethoxybenzoyl)-2-(naphthalen-1-ylmethyl)morpholine
1-(1,3-benzoxazol-2-yl)-4-(2-methyl-1H-imidazol-1-yl)piperidine-4-carboxylic acid
[(3,4-dimethoxypyridin-2-yl)methyl][1-(dimethyl-1,3-thiazol-4-yl)ethyl]methylamine
1-phenyl-N-{2-[2-(pyridin-3-yl)-1,3-thiazol-4-yl]ethyl}-1H-1,2,3-triazole-4-carboxamide
1,5-dimethyl-2-phenyl-4-(1-{[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl}-1H-imidazol-2-yl)-2,3-dihydro-1H-pyrazol-3-one
1-{3-[3-({[(3,4-difluorophenyl)methyl]amino}methyl)phenoxy]-2-hydroxypropyl}piperidin-4-ol
N,6-dimethyl-N-(oxan-2-ylmethyl)-2-(pyridin-3-yl)pyrimidin-4-amine
3-(4-chloro-1H-pyrazol-1-yl)-N-[(1-methylpyrrolidin-3-yl)methyl]propanamide
propan-2-yl 3-oxo-2-[(2E)-3-phenylprop-2-en-1-yl]-2,8-diazaspiro[4.5]decane-8-carboxylate
N'-(3-chloro-4-methylphenyl)-N-[3-(1H-imidazol-1-yl)propyl]propanediamide
4-({4-[3-(thiophene-2-carbonyl)piperidine-1-carbonyl]furan-2-yl}methyl)morpholine