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N-{[5-(dimethylcarbamoyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}-1-ethylpiperidine-2-carboxamide
3-(2-fluorophenoxy)-1-(oxolan-3-ylmethyl)azetidine
8-(3-hydroxy-4-methoxybenzoyl)-3-(3-methylbutyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
{2-[3-(1-benzyl-1H-imidazol-2-yl)piperidin-1-yl]-1,3-thiazol-4-yl}methanol
[4-(2-phenoxyethyl)-1-{[2-(trifluoromethyl)phenyl]methyl}piperidin-4-yl]methanol
7-fluoro-2-methyl-4-[4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazine-1-carbonyl]quinoline
1-methyl-4-(2-methyl-1H-1,3-benzodiazole-4-carbonyl)piperazine-2-carboxylic acid
(1R,3S)-N1,N1,2,2,3-pentamethyl-N3-[(6-methylquinolin-5-yl)methyl]cyclopentane-1,3-dicarboxamide
1-{2-[1-({7-methylimidazo[1,2-a]pyridin-2-yl}methyl)piperidin-2-yl]ethyl}pyrrolidin-2-one
N,4-dimethyl-5-[4-(2-methylphenyl)-1,4-diazepane-1-carbonyl]-1,3-thiazol-2-amine
methyl (2S,4S,5R)-5-(4-chlorophenyl)-1,2-dimethyl-4-[(1,2-oxazol-3-ylmethyl)carbamoyl]pyrrolidine-2-carboxylate
(3R,4R)-3-cyclopropyl-4-methyl-1-{5-methyl-6-[(2-methylpyridin-3-yl)oxy]pyrimidin-4-yl}pyrrolidin-3-ol
2-{4-[3-(morpholine-4-carbonyl)piperidin-1-yl]piperidin-1-yl}pyrimidin-4-amine
N-benzyl-4-[(3-methylpyridin-2-yl)methyl]piperazine-1-sulfonamide
1-[(4-fluorophenyl)methyl]-4-[(3-propyl-1,2,4-oxadiazol-5-yl)methyl]-1,4-diazepane
1-cyclohexyl-N-cyclopropyl-5-(2-methylpiperidine-1-carbonyl)-4-oxo-1,4-dihydropyridine-3-carboxamide
4-{4-[(2-methylprop-2-en-1-yl)oxy]benzoyl}-3-propylmorpholine
2-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)-1-{4-[2-(oxolan-2-yl)-5-(trifluoromethyl)-1H-1,3-benzodiazol-1-yl]piperidin-1-yl}ethan-1-one
N-[4-(furan-2-yl)butan-2-yl]-2-(phenylamino)pyrimidine-5-carboxamide
4-methyl-1-{[2-(piperidin-1-yl)pyrimidin-5-yl]methyl}-1,4-diazepan-5-one
4-(piperidin-1-ylmethyl)-N-[(1-propyl-1H-imidazol-2-yl)methyl]benzamide
4-{[1-(cyclopropylmethyl)piperidin-4-yl]oxy}-N-(2-phenylethyl)benzamide
(3R,5S)-1-benzyl-N-[(3,5-dimethylphenyl)methyl]-5-(morpholin-4-ylmethyl)piperidine-3-carboxamide
N-ethyl-5-({4-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl}methyl)pyrimidin-2-amine
N-(1-hydroxybutan-2-yl)-1-methyl-2-oxo-N-(pyridin-4-ylmethyl)-1,2-dihydropyridine-3-carboxamide
1-(2-methyl-1-benzofuran-5-yl)-3-[2-(2-methylpropanesulfonyl)ethyl]urea
1-[(3R,4R)-4-ethyl-3,4-dihydroxypiperidin-1-yl]-2-(pyridin-4-ylsulfanyl)ethan-1-one
6-{1-[2-(piperazin-1-yl)ethyl]-1H-1,2,3-triazole-4-carbonyl}-1H,2H,3H,4H,5H,6H,7H,8H-pyrazolo[3,4-d]azepin-3-one
5-ethyl-N-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]pyrazolo[1,5-a]pyrimidin-7-amine
1-{2-[3-(3-chlorophenyl)propanamido]ethyl}piperidine-3-carboxamide
1-benzyl-N-cyclopropyl-4-oxo-5-(3-phenylpiperidine-1-carbonyl)-1,4-dihydropyridine-3-carboxamide
N,N-dimethyl-6-{3-[1-(1,3-thiazol-2-ylmethyl)-1H-pyrazol-3-yl]phenyl}pyridazin-3-amine
1-ethyl-5-[ethyl(2-methylprop-2-en-1-yl)amino]-N-methyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
(2S,4S,5R)-5-(4-chlorophenyl)-1,2-dimethyl-4-[(pyridin-3-ylmethyl)carbamoyl]pyrrolidine-2-carboxylic acid
2-({5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl}methyl)-7-(2-phenylethyl)-2,7-diazaspiro[4.5]decane
N-[2-(cyclohexylsulfanyl)ethyl]-5-oxo-1-(pyridin-4-ylmethyl)pyrrolidine-3-carboxamide
2-ethyl-9-(2-methyl-6-oxo-1,6-dihydropyrimidine-5-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
N-{[4-(1H-1,3-benzodiazol-2-yl)cyclohexyl]methyl}-1-(methoxymethyl)cyclobutane-1-carboxamide
1-[3-(3-hydroxyphenyl)propanoyl]-4-methylpiperidine-4-carbonitrile
1-[7-(cyclohexylmethyl)-2,7-diazaspiro[4.5]decan-2-yl]-3-(1-methyl-1H-pyrazol-4-yl)propan-1-one
N-[(1-ethyl-1H-imidazol-2-yl)methyl]-N-methyl-1-(2-phenylethyl)piperidin-3-amine
6-(hydroxymethyl)-N-[3-(pyridin-3-yl)phenyl]-1,4-oxazepane-4-carboxamide
N-[(5-{[(2-fluorophenyl)methyl]sulfanyl}-4-(2-methylpropyl)-4H-1,2,4-triazol-3-yl)methyl]-2,3,4-trimethoxybenzamide
2-(3-cyano-2-methoxypyridin-4-yl)benzamide
13-(2-hydroxy-7-methylquinolin-3-yl)-5-thia-2,7,10-triazatricyclo[6.5.0.02,6]trideca-1(8),3,6-trien-11-one
1-[(3-chlorophenyl)methyl]-5-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-3-(2-methoxyethyl)-1H-1,2,4-triazole
2-(2-methoxyphenyl)-5-{1-propyl-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}-1,3-thiazole
2-cyclopropyl-4-methyl-5-{4-[(2-methylphenyl)sulfanyl]piperidine-1-carbonyl}pyrimidine
3-(1H-pyrazol-1-yl)-N-[2,2,2-trifluoro-1-(pyridin-3-yl)ethyl]benzamide
4-{2,3-dimethyl-5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}-1λ6-thiomorpholine-1,1-dione