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3-[({1-[2-(2-methoxyphenyl)ethyl]piperidin-4-yl}methyl)(methyl)amino]propane-1,2-diol
N-({5-[(4-methoxy-2-methylphenyl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)cyclobutanecarboxamide
1-[1-(propan-2-yl)piperidin-4-yl]-3-[4-(trifluoromethyl)benzoyl]piperidine
2-(3-methylbutyl)-8-[3-(methylsulfanyl)propanoyl]-2,8-diazaspiro[5.5]undecan-3-one
5-[(2E)-but-2-en-1-yl]-N-methyl-N-(2-phenylethyl)-1,3,4-oxadiazole-2-carboxamide
N-[1-(3-fluorophenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]-1-methyl-1H-imidazole-4-sulfonamide
5-[2-chloro-4-(1H-pyrazol-1-yl)benzoyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxylic acid
methyl 4-(5-methyl-4-{[methyl(oxan-4-yl)amino]methyl}-1,3-oxazol-2-yl)benzoate
5-[2-(3-hydroxy-4-methoxyphenyl)-1H-imidazol-1-yl]-1,3,6-trimethyl-2,3-dihydro-1H-1,3-benzodiazol-2-one
3-(4-ethylphenyl)-5-{pyrazolo[1,5-a]pyridine-3-carbonyl}-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
(2S,4R)-1-[(3-chlorophenyl)methyl]-4-{[(2,4-dimethoxy-3-methylphenyl)methyl]amino}-N-(propan-2-yl)pyrrolidine-2-carboxamide
1-{[2-(4-methoxy-2,3-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidine-3-carboxamide
2-(2-amino-4,6-dimethylpyrimidin-5-yl)-N-methyl-N-{[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}acetamide
4-{[(1R,3S,3aS,6aR)-3-(3-ethoxyphenyl)-1-(hydroxymethyl)-5-methyl-octahydropyrrolo[3,4-c]pyrrol-1-yl]methyl}phenol
3-(5-{1-[(2-methyl-2,3-dihydro-1-benzofuran-5-yl)methyl]-1H-imidazol-2-yl}thiophen-2-yl)prop-2-yn-1-ol
2-(methylamino)-N-[3-(2-oxopyrrolidin-1-yl)propyl]pyridine-4-carboxamide
2-[2-(ethylsulfanyl)-1,3-thiazol-4-yl]-1-[2-(3-methyl-1,2,4-oxadiazol-5-yl)piperidin-1-yl]ethan-1-one
N-cyclohexyl-N-ethyl-1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
N-{2-[(2R)-5-oxopyrrolidine-2-carbonyl]-1,2,3,4-tetrahydroisoquinolin-7-yl}-1-phenylcyclopropane-1-carboxamide
2-(morpholin-3-yl)-N-(quinolin-8-yl)acetamide
4-{[3-(3-chlorobenzoyl)piperidin-1-yl]methyl}-2-ethoxyphenol
methyl 4-{[methyl({[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl})amino]methyl}-1H-pyrazole-3-carboxylate
N-[2-(4-fluorobenzenesulfonyl)ethyl]-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-amine
5,6-dimethyl-N4-{2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]ethyl}pyrimidine-2,4-diamine
(3S,4R)-1-{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}-4-(pyridin-4-yl)pyrrolidine-3-carboxylic acid
2-(3-chloro-4-methoxyphenyl)-2-[4-hydroxy-4-(pyridin-3-yl)piperidin-1-yl]acetic acid
methyl 6-[({1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}carbamoyl)amino]-1,2,3,4-tetrahydroquinoline-1-carboxylate
3-(3,4-dimethylbenzoyl)-9-methoxy-N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
1-[(2E)-3-phenylprop-2-en-1-yl]-4-(2-propyl-1,3-thiazole-4-carbonyl)piperazine
6-fluoro-2-{[2-(piperidin-1-ylmethyl)-1,4-oxazepan-4-yl]methyl}quinoline
2-[(3-methoxyphenyl)methyl]-8-(3-methoxypropyl)-2,8-diazaspiro[4.5]decan-3-one
N-[1-(1H-indol-5-yl)ethyl]-1H,4H,6H,7H-pyrano[4,3-c]pyrazole-3-carboxamide
2-[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl]-7-(propan-2-yl)-2,7-diazaspiro[4.5]decan-6-one
(3aS,6aR)-5-[(4-hydroxyphenyl)methyl]-3-[3-(morpholin-4-yl)propyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
5-{5H,6H,7H,8H-imidazo[1,5-a]pyrazine-7-carbonyl}-1-(prop-2-en-1-yl)piperidin-2-one
N-(9H-fluoren-2-yl)-2-(morpholin-3-yl)acetamide
1-[2-({[(4-fluorophenyl)methyl](methyl)amino}methyl)-5-methoxyphenoxy]-3-(4-methylpiperazin-1-yl)propan-2-ol
6-methyl-3-[3-(1H-pyrazol-3-yl)phenyl]pyridin-2-amine
2-{4-[3-hydroxy-3-(2-methylphenyl)pyrrolidin-1-yl]pyrimidin-5-yl}acetic acid
7-{6-azaspiro[2.5]octane-1-carbonyl}-2-phenyl-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
5-[4-(1H-indole-6-carbonyl)piperazin-1-yl]-2-methyl-2,3-dihydropyridazin-3-one
2-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)-N-{[2-(2-fluorophenyl)-3-methyl-1H-indol-5-yl]methyl}acetamide
6-methyl-5-[5-(2-methylbutan-2-yl)-1,2,4-oxadiazol-3-yl]-2-(pyridin-4-ylmethyl)-1,2,3,4-tetrahydro-2,7-naphthyridine
N-{3-[bis(2-hydroxyethyl)amino]propyl}-2,8-dimethylquinoline-4-carboxamide
(4S)-1-[(1-cyclohexyl-1H-imidazol-5-yl)methyl]-3,3,4-trimethylpiperidin-4-ol
2-[methyl(phenyl)amino]-1-{4-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
3-[(3R,4S)-1-(2-methyl-5-propylpyrimidin-4-yl)-4-(morpholin-4-yl)piperidin-3-yl]propanoic acid
3-hydroxy-N-[1-(pyridin-2-yl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]pyridine-2-carboxamide
{1-[(2-fluorophenyl)methanesulfonyl]-3-(prop-2-en-1-yl)piperidin-3-yl}methanol
N-({1-[2-(4-chlorophenyl)ethyl]piperidin-3-yl}methyl)-N-methylbenzamide