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2-(4-propanoylphenoxy)-N-[3-(1H-1,2,4-triazol-1-yl)propyl]acetamide
3-(3-fluorophenyl)-5-{5-[(methylsulfanyl)methyl]furan-2-carbonyl}-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
1-{3-[3-(hydroxymethyl)-3-(3-methylbut-2-en-1-yl)piperidin-1-yl]-3-oxopropyl}azepan-2-one
4-{[4-(1,3-benzoxazol-2-yl)piperazin-1-yl]methyl}-2-fluoro-6-methoxyphenol
{1-[(1-cyclopropyl-1H-imidazol-5-yl)methyl]-3-(3-methoxypropyl)piperidin-3-yl}methanol
5-ethyl-2-{1-[(1-methylpiperidin-2-yl)methyl]-1H-imidazol-2-yl}pyridine
2-[4-methyl-6-(4-{[2-(1H-pyrazol-1-yl)ethyl]amino}piperidin-1-yl)pyrimidin-2-yl]phenol
methyl(oxan-4-ylmethyl){[5-(1H-pyrazol-3-yl)thiophen-2-yl]methyl}amine
4-fluoro-N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-N-(oxolan-2-ylmethyl)benzamide
3-benzyl-5-[5-(2-methylpropyl)-1,2-oxazol-3-yl]-1H-1,2,4-triazole
2-(1-cyclopentyl-4-{[2-(difluoromethoxy)phenyl]methyl}piperazin-2-yl)ethan-1-ol
2-[1-(furan-3-ylmethyl)-4-(1-methyl-1H-indole-6-carbonyl)piperazin-2-yl]ethan-1-ol
2-{2-[1-({4-oxo-3H,4H-thieno[3,2-d]pyrimidin-2-yl}methyl)piperidin-3-yl]-1H-imidazol-1-yl}acetamide
1-ethyl-N-(furan-3-ylmethyl)-N-methyl-5-[methyl(2-methylpropyl)amino]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N-({1-[(3-methylthiophen-2-yl)sulfonyl]piperidin-3-yl}methyl)-1-phenylmethanesulfonamide
(1s,4s)-N-[3-(3,4-diethoxyphenyl)propyl]-4-hydroxycyclohexane-1-carboxamide
2-methyl-N-[1-(3-methylpyridin-2-yl)ethyl]-6-(piperidin-4-yl)pyrimidin-4-amine
{[6-chloro-2-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}(methyl)(1H-pyrazol-5-ylmethyl)amine
4-[(2-fluorophenyl)methyl]-1-[2-(phenylsulfanyl)acetyl]-1,4-diazepan-5-one
1-[(1R,2R,6S,7S)-4-azatricyclo[5.2.1.02,6]decan-4-yl]-4-(2-methyl-1H-imidazol-1-yl)butan-1-one
4-(4-phenoxyphenyl)-1H-pyrazolo[3,4-d]pyrimidin-6-amine
ethyl 1-[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]-4-oxo-5-phenoxy-1,4-dihydropyridine-3-carboxylate
N-[(3,4-difluorophenyl)methyl]-3-{1-[(3-hydroxyphenyl)methyl]piperidin-3-yl}propanamide
3-{[3-cyclopropyl-1-(2-fluorophenyl)-1H-1,2,4-triazol-5-yl]methyl}-3,4-dihydroquinazolin-4-one
ethyl 4-{6-[(3-phenyl-1H-pyrazol-4-yl)methyl]-6-azaspiro[2.5]octane-1-carbonyl}piperazine-1-carboxylate
2-[({1-[1-(naphthalen-1-ylmethyl)-1H-1,2,3-triazole-4-carbonyl]piperidin-4-yl}oxy)methyl]pyridine
N-[(3S,7S,8aS)-1,4-dioxo-3-(propan-2-yl)-octahydropyrrolo[1,2-a]piperazin-7-yl]-4-ethylbenzamide
1-(3-methylpyridin-2-yl)-4-(2-propyl-1,3-thiazole-4-carbonyl)piperazine
2-amino-8-[2-(pyridin-2-yl)pyrimidin-5-yl]-4H,5H,6H,7H,8H-[1,3]thiazolo[4,5-c]azepin-6-one
N-cyclopropyl-2-{4-[(4-ethyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)methyl]piperidin-1-yl}pyridine-4-carboxamide
4-{1-[(3-methoxyphenyl)methyl]-5-(oxolan-3-yl)-1H-1,2,4-triazol-3-yl}benzamide
4-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]-1-({2-methylimidazo[1,2-a]pyridin-3-yl}methyl)piperidine
4-[(4-{2-[1-(2-cyclopentylacetyl)piperidin-2-yl]ethoxy}phenyl)methyl]piperazine-1-carbaldehyde
4-[3-(propoxymethyl)pyrrolidin-1-yl]pyrimidine-5-carboxylic acid
1-{4-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl}-2-[2-(propan-2-yl)-1H-imidazol-1-yl]propan-1-one
1-[1-ethyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-4-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}piperidine
1-(3-fluorophenyl)-5-[(5-methyl-1H-pyrazol-1-yl)methyl]-3-(oxan-4-yl)-1H-1,2,4-triazole
3-(4-methyl-1,3-thiazol-5-yl)-N-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}propanamide
1-{[2-(2H-1,3-benzodioxol-5-yl)phenyl]methyl}piperazine
N2,N4,N4,5-tetramethyl-N2-[2-(pyridin-4-yl)ethyl]pyrimidine-2,4-diamine
N,N-dimethyl-2-[(1S,5R)-6-[(1-methyl-1H-indol-2-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-3-yl]acetamide
(1S,5R)-6-(cyclobutylmethyl)-3-[2-(2-methyl-1,3-thiazol-4-yl)acetyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
1-methyl-8-(4-methylquinolin-2-yl)-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
N-[(3R,4R)-3-hydroxypiperidin-4-yl]-5-(1H-indol-1-ylmethyl)furan-2-carboxamide
N-cyclobutyl-4-{[(5-methylpyrazin-2-yl)methyl]sulfamoyl}benzamide
N-[2-(3,4-dimethylphenyl)ethyl]-4-hydroxy-1-methylpiperidine-4-carboxamide
4-[(3,4-dimethoxyphenyl)methyl]-3-[2-(4-hydroxypiperidin-1-yl)-2-oxoethyl]piperazin-2-one
3-ethyl-6-(4-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}piperidine-1-carbonyl)-3H-imidazo[4,5-b]pyridin-2-amine
2-{1-[(3-ethyl-1H-pyrazol-5-yl)methyl]piperidin-4-yl}-1H-1,3-benzodiazole
{[2-(4-methoxy-2,5-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]amine