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N-[3-(1H-imidazol-1-yl)propyl]-3-(2-methylpyrrolidine-1-carbonyl)benzene-1-sulfonamide
N-{[2-(4-methyl-1,4-diazepan-1-yl)pyridin-3-yl]methyl}-4-(1H-1,2,4-triazol-1-yl)butanamide
2-{5,7-dimethylpyrido[2,3-d]pyrimidin-4-yl}-7-methyl-2,7-diazaspiro[4.4]nonane
N-{[2-(diethylamino)pyridin-3-yl]methyl}-4,4,4-trifluorobutanamide
2-(piperazin-1-yl)-1-{spiro[azepane-4,2'-chromene]-1-yl}ethan-1-one
1-{4-[(1-methylpiperidin-4-yl)oxy]phenyl}-3-[1-(pyrazin-2-yl)propan-2-yl]urea
N-methyl-4-[3-methyl-5-(pyrrolidin-1-ylmethyl)phenyl]-1H-pyrrolo[2,3-b]pyridin-6-amine
N,6-dimethyl-N-{[5-(propan-2-yl)-1,2-oxazol-3-yl]methyl}-2-(pyridin-3-yl)pyrimidin-4-amine
1-(furan-2-carbonyl)-4-{pyrazolo[1,5-a]pyrimidin-3-ylmethyl}piperazine
N-{2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]ethyl}-3-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanamide
(2S,4R)-4-amino-N-ethyl-1-({5-[(4-methylphenyl)sulfanyl]furan-2-yl}methyl)pyrrolidine-2-carboxamide
4-({3-[(2-chlorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)morpholine
N-(1-carbamoylcyclopentyl)-2-(1H-imidazol-2-yl)benzamide
7-(7-methoxy-4-methylquinazolin-2-yl)-2-methyl-2,7-diazaspiro[4.5]decane
N-[2-(5-cyclobutyl-1,2,4-oxadiazol-3-yl)ethyl]-3-phenoxypropanamide
7-methyl-2-[1-(2-methylphenyl)piperidin-4-yl]-2,7-diazaspiro[4.5]decan-6-one
2-[methyl(piperidin-4-yl)amino]-N-[(1-phenylcyclohexyl)methyl]acetamide
4-(2-methylphenoxy)-1-[3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]piperidine
(3S,4S)-1-[4-(4-fluorophenyl)-4-oxobutanoyl]-4-propylpyrrolidine-3-carboxylic acid
4-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-1-[(2-methyl-1,3-thiazol-4-yl)methyl]-6-(pyridin-4-ylmethoxy)-1,4-diazepan-2-one
(1S,5R)-6-(1-ethyl-1H-pyrazole-3-carbonyl)-3-[(4-methoxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane
4-(cyclopropylmethyl)-1-[(1-phenyl-1H-pyrazol-4-yl)methyl]-1,4-diazepan-5-one
N-[2-(4-fluorophenyl)ethyl]-4-hydroxy-4-(5-methylpyridin-2-yl)piperidine-1-carboxamide
3-[1-(1H-imidazol-1-yl)butan-2-yl]-5-methyl-3H,4H-thieno[2,3-d]pyrimidin-4-one
(2S)-1-[(4-{[2-(2-methoxyphenyl)ethyl]amino}quinazolin-2-yl)methyl]pyrrolidine-2-carboxamide
1'-{[2-(2-hydroxyethoxy)phenyl]methyl}-1-methyl-1,2-dihydrospiro[indole-3,3'-piperidine]-2-one
3-(azepane-1-sulfonyl)-N-[1-(1H-pyrazol-1-yl)propan-2-yl]benzamide
2-(4-methyl-2-phenyl-1H-imidazol-1-yl)-N-{1,4,6-trimethyl-1H-pyrazolo[3,4-b]pyridin-3-yl}acetamide
2-(3-chloro-4-hydroxyphenyl)-1-[4-hydroxy-4-(5-methylpyridin-2-yl)piperidin-1-yl]ethan-1-one
7-(cyclobutylmethyl)-2-[2-(2-oxo-1,2-dihydropyrimidin-1-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one
2-[(4S)-4-hydroxy-4-(methoxymethyl)-3,3-dimethylpiperidin-1-yl]-N-(2-phenylethyl)acetamide
N-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}-1-(propan-2-yl)-1H-pyrazole-4-carboxamide
N-[1-(3,5-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-(1H-indazol-3-yl)acetamide
4-{5-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-3-(thiophen-2-ylmethyl)-1H-1,2,4-triazol-1-yl}-1-methylpiperidine
2-amino-6-cyclopropanecarbonyl-4-[3,5-dimethyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
N-methyl-N-(oxolan-3-yl)-1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidine-4-carboxamide
[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl][3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl]methylamine
2-(azepan-1-yl)-1-{4-[4-(morpholine-4-carbonyl)piperidin-1-yl]piperidin-1-yl}ethan-1-one
(4aR,8aR)-4a-hydroxy-7-{[4-methoxy-3-(methoxymethyl)phenyl]methyl}-N,N-dimethyl-decahydro-2,7-naphthyridine-2-carboxamide
1-[(3R,4R)-3-[(dimethylamino)methyl]-4-(hydroxymethyl)pyrrolidin-1-yl]-4-(4-methoxyphenyl)butane-1,4-dione
3-chloro-5-fluoro-N-{1-[(3-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}benzamide
1-(furan-2-ylmethyl)-N-[2-(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)ethyl]piperidine-3-carboxamide
3,5-dimethoxy-2-[(3,3,4-trimethylpiperazin-1-yl)methyl]benzoic acid
[(3R,4R)-1-(5-methoxy-1H-indole-2-carbonyl)-4-{[(2-methoxyethyl)(methyl)amino]methyl}pyrrolidin-3-yl]methanol
3-({[5-methyl-6-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)thieno[2,3-d]pyrimidin-4-yl]amino}methyl)-1λ6-thiolane-1,1-dione
7-[(3-chloro-5-fluoro-4-methoxyphenyl)methyl]-5H,6H,7H,8H-imidazo[1,5-a]pyrazine
2-[(4-{4-[(2R,6R)-6-methyl-2-(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridine-1-carbonyl]phenoxy}piperidin-1-yl)methyl]pyridine
N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-2-(4-methyl-1,2,5-oxadiazol-3-yl)acetamide
2-[1-oxo-1-(pyrrolidin-1-yl)propan-2-yl]-5-(piperazin-1-yl)-2,3-dihydropyridazin-3-one
3-{[ethyl({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)amino]methyl}phenol