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1'-(5-chloropyridin-2-yl)-5-ethyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
5-[(dimethylamino)methyl]-N-(1-hydroxybutan-2-yl)-N-[(2-methylphenyl)methyl]furan-2-carboxamide
1-[3-(morpholin-4-yl)propyl]-6-oxo-N-(2-phenoxyethyl)piperidine-3-carboxamide
[(5-cyclopropyl-1H-pyrazol-3-yl)methyl](methyl){[5-(1H-pyrazol-3-yl)thiophen-2-yl]methyl}amine
(1-{[1-(2-phenylethyl)-2-(propane-2-sulfonyl)-1H-imidazol-5-yl]methyl}piperidin-2-yl)methanol
N-[1-(naphthalen-1-ylmethyl)-5-oxopyrrolidin-3-yl]pent-4-enamide
1-{[4-(benzyloxy)phenyl]methyl}-4-methyl-1,4-diazepan-5-one
N-[4-(3-methoxyphenyl)phenyl]-1-(thian-4-yl)pyrrolidine-2-carboxamide
3-({3-oxo-2-[2-(pyridin-2-yl)ethyl]-2,9-diazaspiro[5.5]undecan-9-yl}methyl)benzonitrile
2-(dimethyl-1,2-oxazole-4-carbonyl)-7-[(2-fluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
1-(4-methoxyphenyl)-4-[1-(pyridin-2-yl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]butane-1,4-dione
1-{2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}-4-(2-methoxyethyl)piperazine
2-[4-methoxy-3-(pyrrolidin-1-ylmethyl)phenoxy]-3-(trifluoromethyl)pyridine
N-[1-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-yl]-1H-pyrrolo[2,3-b]pyridin-6-amine
methyl 1-[3-(2-phenylethyl)-1,2-oxazole-5-carbonyl]piperidine-2-carboxylate
(2S)-2-amino-3-(1H-imidazol-4-yl)-1-{4-[(3-methylphenyl)sulfanyl]piperidin-1-yl}propan-1-one
[2-(4-methoxy-3-methylphenyl)-1,3-thiazol-4-yl]methanol
N-[3-(dimethylamino)propyl]-5-(4-phenylazepane-1-carbonyl)pyridin-2-amine
1-(2-ethoxyethyl)-5-(4-methyl-1,4-diazepane-1-carbonyl)-2,3-dihydro-1H-1,3-benzodiazol-2-one
3-(1-butyl-1H-imidazol-2-yl)-1-{[4-(1H-pyrazol-1-yl)phenyl]methyl}piperidine
5-(1,3-dimethyl-1H-pyrazole-5-carbonyl)-1-(2-phenylethyl)-N-(pyridin-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
8-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-2-(propan-2-yl)-2,8-diazaspiro[5.5]undecan-3-one
N-{[4-(cyclobutylmethoxy)phenyl]methyl}-N-cyclopropyl-2-(3-oxo-2,3-dihydro-1H-isoindol-1-yl)acetamide
3-(3-methoxyphenyl)-1-{2-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-1-yl}propan-1-one
N-[2-methoxy-1-(pyridin-2-yl)ethyl]-N,1,5-trimethyl-1H-indole-2-carboxamide
N-{[2-(2-methoxyphenoxy)pyridin-3-yl]methyl}-2-(2-methyl-1H-imidazol-1-yl)acetamide
(3R,4R)-3-hydroxy-N-(2-methylphenyl)-4-{[(5-methylpyrazin-2-yl)methyl]amino}pyrrolidine-1-carboxamide
4-{[4-methoxy-3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}piperazine-2-carboxylic acid
4,5-dimethyl-6-[3-(pyridin-2-yl)azetidin-1-yl]-2-(trifluoromethyl)pyrimidine
(2S,4S)-1-[(4-chlorophenyl)methyl]-N-(pyridin-3-ylmethyl)-4-({[2-(trifluoromethyl)phenyl]methyl}amino)pyrrolidine-2-carboxamide
N-(2-chlorophenyl)-3-(1-{[4-(propan-2-yl)-1,3-thiazol-2-yl]methyl}piperidin-4-yl)propanamide
2-methoxy-4-{2-[2-(pyrrolidine-1-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl]propyl}phenol
(benzylsulfamoyl)[(2-ethoxypyridin-3-yl)methyl]amine
ethyl 3-{[2-(3-phenylpropyl)-1,3-benzoxazol-5-yl]formamido}propanoate
1-(1,4-dioxane-2-carbonyl)-4-[3-(trifluoromethyl)phenyl]piperidin-4-ol
3-({2-[1-(3-fluoro-4-methylbenzoyl)piperidin-4-yl]-1H-imidazol-1-yl}methyl)pyridine
N-[(1R,2R)-1-({5-ethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)-2,3-dihydro-1H-inden-2-yl]acetamide
N-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}-1-(4-fluorophenyl)-N-methylcyclopropane-1-carboxamide
2-{[1-(2-hydroxypropanoyl)piperidin-4-yl]oxy}-4-methoxy-N-(2-methoxyethyl)benzamide
N-(2-cyclooctylethyl)-1-cyclopentyl-6-oxopiperidine-3-carboxamide
8-fluoro-3-{3-[(2-methyl-1H-imidazol-1-yl)methyl]piperidine-1-carbonyl}-1,4-dihydroquinolin-4-one
1-(furan-2-ylmethyl)-4-[2-(1,3-thiazol-2-yl)pyrrolidine-1-carbonyl]piperidine
N-{1-[4-(3-methoxypropyl)-4H-1,2,4-triazol-3-yl]ethyl}-2,6-dimethylpyridine-4-carboxamide
2-(4-{[3,5-dimethyl-1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-1-(thiophen-3-ylmethyl)piperazin-2-yl)ethan-1-ol
7-(4-chloro-1-methyl-1H-pyrazole-3-carbonyl)-1-oxa-7-azaspiro[3.5]nonane
3-{[2-(2-butyl-1H-imidazol-4-yl)-1H-imidazol-1-yl]methyl}-7-fluoro-1,2-dihydroquinolin-2-one
2,7-dimethyl-N-(1H-1,2,3,4-tetrazol-5-ylmethyl)pyrazolo[1,5-a]pyrimidine-5-carboxamide
3-(2-hydroxyphenyl)-N-methyl-N-[3-(1-methyl-1H-pyrazol-4-yl)propyl]-1H-pyrazole-5-carboxamide
6-ethyl-3-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}-1,5-dimethyl-1,2-dihydropyridin-2-one
4-(2-methoxyphenoxy)-1-(2-methylpyridin-4-yl)piperidine-4-carboxylic acid