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4-[1-methyl-6-(2-phenylethyl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]piperazin-2-one
4-[4-(4-cyclopentylpiperazine-1-carbonyl)phenyl]-2-methylbutan-2-ol
2-{2-[6-hydroxy-4-(pyridin-4-yl)-1,4-diazepan-1-yl]-2-oxoethoxy}acetamide
N-(2,1,3-benzothiadiazol-5-ylmethyl)-3-(dimethyl-1H-1,2,4-triazol-1-yl)-N,2-dimethylpropanamide
8-[(4-methoxy-2-methylphenyl)methyl]-2-(3-methoxypropyl)-2,8-diazaspiro[5.5]undecan-3-one
N3-methyl-N3-(2-methylpropyl)-4-oxo-1-(propan-2-yl)-N5-[2,2,2-trifluoro-1-(furan-2-yl)ethyl]-1,4-dihydropyridine-3,5-dicarboxamide
5-methoxy-N-{[5-(2-methylpropyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}furan-2-carboxamide
4-hydroxy-2-(3-methylphenyl)-N-[2-(pyridin-2-yl)ethyl]pyrimidine-5-carboxamide
3-{4-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}-2-methylphenol
2-(ethylamino)-N-{[3-(trifluoromethoxy)phenyl]methyl}pyrimidine-5-carboxamide
4-{2-[(1-methyl-1H-indol-3-yl)sulfanyl]acetyl}-1λ6-thiomorpholine-1,1-dione
3-[(6-chloro-2-methylquinolin-4-yl)formamido]-N-cyclohexylpropanamide
N-[3-(2-methoxyphenyl)-3-methylpentyl]-1-methyl-2-oxo-1,2-dihydropyridine-3-carboxamide
1-[(4-methoxyphenyl)methyl]-3-{[5-(2-methylpropyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}urea
N-methyl-2-{[(2-methyl-1,3-benzothiazol-5-yl)oxy]methyl}-N-[(5-methylfuran-2-yl)methyl]-1,3-oxazole-4-carboxamide
(5S,9aS,9bS)-2-(2,3-dihydro-1H-inden-2-yl)-5-[2-(morpholin-4-yl)-1,3-thiazol-5-yl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
5-[2-(benzyloxy)ethyl]-4-(furan-3-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
3-{4-[(3-fluorophenyl)methyl]piperazine-1-carbonyl}-1-methyl-1,2-dihydropyridin-2-one
N-methyl-N-(1-methylpyrrolidin-3-yl)-2-[3-(trifluoromethyl)phenoxymethyl]-1,3-oxazole-4-carboxamide
2-(3-methoxyphenyl)-5-(oxane-4-carbonyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
14-[3-(1H-pyrazol-1-ylmethyl)phenyl]-2,8,11-triazatricyclo[7.5.0.02,7]tetradeca-1(9),3,5,7-tetraen-12-one
4,4,4-trifluoro-N-methyl-N-[(1-phenylpyrrolidin-3-yl)methyl]butanamide
1-(2,2-dimethylpropyl)-3-hydroxy-3-{[(2-methylpropyl)amino]methyl}piperidin-2-one
1-cyclopropyl-N-(2,2-diphenylpropyl)-6-oxopiperidine-3-carboxamide
1-(1-{[4-(piperidin-1-ylmethyl)thiophen-2-yl]methyl}piperidin-4-yl)-N-(propan-2-yl)piperidine-4-carboxamide
1-[(1R,5R)-6-(cyclopropylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]-2-[5-(4-fluorophenyl)-2H-1,2,3,4-tetrazol-2-yl]ethan-1-one
4-methyl-N-[(4-sulfamoylphenyl)methyl]-1H-imidazole-5-carboxamide
N-({5-cyclobutanecarbonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-5-hydroxypyrazine-2-carboxamide
(3S,9aR)-8-[(2-fluorophenyl)methyl]-3-(1H-indol-3-ylmethyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
1-[3-carboxy-5-(thiomorpholine-4-sulfonyl)phenyl]-1H-pyrazole-4-carboxylic acid
2-ethyl-4-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl]pyridine
N-[(3,4-difluorophenyl)methyl]-3-[1-(2,6-dimethylpyrimidine-4-carbonyl)piperidin-3-yl]propanamide
methyl 3-{2-[(2,4-dimethylphenyl)carbamoyl]acetamido}propanoate
1-[4-(2H-1,3-benzodioxol-5-yl)pyrimidin-2-yl]-N-[2-(diethylamino)ethyl]-5-(furan-2-yl)-N-methyl-1H-pyrazole-4-carboxamide
N-{1-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]ethyl}-2-(trimethyl-1H-pyrazol-1-yl)acetamide
2-{[1-(6-methylpyridazin-3-yl)piperidin-3-yl]methyl}-1H-1,3-benzodiazole
N-[(3R,7S,8aS)-3-[(4-hydroxyphenyl)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]thiophene-2-carboxamide
4-[4-ethyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(3-methylbut-2-en-1-yl)piperidine
(2S,4S)-4-(4-cyanobenzamido)-N-[(2-fluorophenyl)methyl]-1-methylpyrrolidine-2-carboxamide
6-cyclopentyl-N-{[4-(dimethylamino)oxan-4-yl]methyl}-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
({5-[1-(5-methoxy-1H-indole-2-carbonyl)piperidin-4-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methyl)dimethylamine
1-methyl-N-(3-{[(3-methylphenyl)methyl]sulfanyl}propyl)azepane-2-carboxamide
N-(cyclohexylmethyl)-1-cyclopropyl-4-oxo-5-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-1,4-dihydropyridine-3-carboxamide
1-[(1,4-dimethyl-1H-pyrazol-5-yl)methyl]-4-(2-ethoxyethyl)-1,4-diazepan-6-ol
1-{1-[(2-chlorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}-4-(methoxymethyl)piperidine
1-[3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)phenyl]-3-{2-[(trifluoromethyl)sulfanyl]ethyl}urea
2-{2-cyclopropyl-3-oxo-4-phenyl-2,9-diazaspiro[5.5]undecan-9-yl}-N-methylacetamide
1-[3-(naphthalene-2-carbonyl)piperidin-1-yl]-3-(1H-pyrazol-1-yl)propan-1-one
1-{8-methyl-2,8-diazaspiro[4.5]decan-2-yl}-3-[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]propan-1-one
2-[4-methyl-6-({[3-(pyrimidin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}amino)pyrimidin-2-yl]phenol