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2-[5-(2H-indazol-2-ylmethyl)-3-(pyridin-4-yl)-1H-1,2,4-triazol-1-yl]ethan-1-ol
3-{3-[(4-fluorophenyl)amino]piperidin-1-yl}propanamide
1-ethyl-3-methyl-8-({6-methylimidazo[2,1-b][1,3]thiazol-5-yl}methyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-{[4-(1H-imidazol-1-yl)phenyl]methyl}-4-(3-methylpyridin-4-yl)-1,4-diazepane
[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl](methyl){[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}amine
{5-[(1-{[2-(furan-2-yl)pyrimidin-5-yl]methyl}piperidin-4-yl)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}methanol
4-[(3-methylpyridin-2-yl)methyl]-2-(naphthalen-1-ylmethyl)morpholine
(2S)-1-(5-ethyl-1,3-oxazole-4-carbonyl)-N-[4-(1,3-thiazol-4-yl)phenyl]pyrrolidine-2-carboxamide
3-[(3S,5S,9S)-2,8-dioxo-1,7-diazatricyclo[7.3.0.03,7]dodecan-5-yl]-1-[3-(trifluoromethyl)phenyl]urea
2-{1-[(4-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]acetamide
1-{2-[4-(2,5-dihydro-1H-pyrrol-1-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl]-2-oxoethyl}imidazolidine-2,4-dione
4-(3-methylfuran-2-carbonyl)-2-{[3-(trifluoromethyl)phenyl]methyl}morpholine
N-[(3-methoxyphenyl)methyl]-3-[1-(pyrazine-2-carbonyl)piperidin-3-yl]propanamide
9-methoxy-3-[2-(phenylsulfanyl)acetyl]-10-(thiomorpholine-4-carbonyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepin-7-one
3-(2-hydroxyphenyl)-N-[(2-methylphenyl)methyl]-N-(prop-2-en-1-yl)propanamide
3-{2-[2,2-bis(prop-2-en-1-yl)piperidin-1-yl]-2-oxoethyl}-4-[(2-methoxyphenyl)methyl]piperazin-2-one
1-{4-[(4,4-difluoropiperidin-1-yl)methyl]-2-methoxyphenoxy}-3-(morpholin-4-yl)propan-2-ol
4-[7-(2-cyclohexylethyl)-2,7-diazaspiro[4.5]decan-2-yl]-N,N-dimethyl-4-oxobutanamide
(4aR,8aS)-6-(3-fluorobenzoyl)-1-(oxolane-2-carbonyl)-decahydro-1,6-naphthyridine
N-[2-(5-amino-1,3,4-thiadiazol-2-yl)propan-2-yl]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
ethyl 5-(2H-1,3-benzodioxol-4-ylmethyl)-1-(2-phenylethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-1-(2-hydroxyethyl)-1H-1,3-benzodiazole-5-carboxamide
N-(6,6-dimethyl-1-phenyl-4,5,6,7-tetrahydro-1H-indazol-4-yl)-1-ethyl-1H-pyrazole-4-carboxamide
2-{4-[2-(3-hydroxyphenyl)acetyl]morpholin-3-yl}-N-(pyrimidin-4-ylmethyl)acetamide
[(3R,4R)-1-(5-chloro-2-methoxybenzoyl)-4-(piperidin-1-ylmethyl)pyrrolidin-3-yl]methanol
2-{[3-(difluoromethoxy)phenyl]methyl}-1H,2H-pyrrolo[1,2-d][1,2,4]triazin-1-one
2-[(propan-2-yl)amino]-N-(2,2,2-trifluoroethyl)pyrimidine-5-carboxamide
2-propoxy-1-{3-[4-(trifluoromethyl)phenyl]-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl}ethan-1-one
[(1-cyclohexylpiperidin-3-yl)methyl][3-(1H-pyrazol-1-yl)propyl](pyridin-3-ylmethyl)amine
2-(2,5-dimethoxyphenyl)-2-[4-(pyridin-2-ylmethyl)piperazin-1-yl]acetic acid
2-cyclohexyl-N-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]-1,3-benzoxazole-6-carboxamide
4-(benzyloxy)-1-{[5-methyl-2-(thiophen-3-yl)-1,3-oxazol-4-yl]methyl}piperidine
2-[(2-butyl-5-chloro-1H-imidazol-4-yl)methyl]-2,8-diazaspiro[4.5]decane
(2S,4R)-4-amino-N-methyl-1-[3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)propanoyl]pyrrolidine-2-carboxamide
5-[(1R,2S,4R)-bicyclo[2.2.1]hept-5-ene-2-carbonyl]-N-phenyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
[(4-fluoro-3-methoxyphenyl)methyl](methyl)[1-(pyridin-2-yl)ethyl]amine
(4aR,7aS)-1-methyl-4-{[5-(2-methylpropyl)-1H-pyrazol-3-yl]methyl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-{4-fluoro-3-[3-(pyridin-3-yl)propyl]phenyl}ethan-1-one
2-oxo-6-phenyl-N-{[1-(propan-2-yl)pyrrolidin-3-yl]methyl}-1,2-dihydropyridine-3-carboxamide
1-{2-[(2S,4R)-4-(dimethylamino)-2-(hydroxymethyl)pyrrolidin-1-yl]-2-oxoethyl}-4-methyl-1,2-dihydroquinolin-2-one
3-[1-(5-carbamoylthiophen-3-yl)-1H-1,3-benzodiazol-2-yl]propanoic acid
2-(2,3-dimethoxyphenyl)-1-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]-1H-imidazole
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-1-methyl-2-oxo-6-(propan-2-yl)-1,2-dihydropyridine-3-carboxamide
[(3R,4R)-1-(1-methyl-1H-indole-4-carbonyl)-4-[(4-methylpiperazin-1-yl)methyl]pyrrolidin-3-yl]methanol
5-{3-[4-(4-fluorophenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}-4-methylpyrimidin-2-amine
3-methanesulfonyl-1-{2-methyl-4-phenyl-2,9-diazaspiro[5.5]undecan-9-yl}propan-1-one
5-[(2S)-2-amino-2-cyclohexylacetyl]-N-cyclopropyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
(3R,4S)-1-[(2-fluoro-4,5-dimethoxyphenyl)methyl]-3,4-dimethylpiperidin-4-ol
[2-(azepan-1-yl)ethyl](ethyl)(1,3-thiazol-4-ylmethyl)amine
3-[5-(3-benzyl-1,2,4-oxadiazol-5-yl)pyridin-2-yl]phenol