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N-[2-(1-methanesulfonylpiperidin-2-yl)ethyl]-1,3-benzothiazole-6-carboxamide
N-cyclopropyl-4-{[1-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}piperazine-2-carboxamide
[(3R,4R)-4-({[2-(dimethylamino)ethyl](methyl)amino}methyl)-1-(5-methyl-1H-indole-2-carbonyl)pyrrolidin-3-yl]methanol
1-(4-methyl-1,2,5-oxadiazole-3-carbonyl)-3-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
1-(6-methoxypyrimidin-4-yl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
1-methyl-1'-(oxolan-2-ylmethyl)-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
2-[2-methoxy-5-({3-oxo-2,9-diazaspiro[5.5]undecan-9-yl}methyl)phenoxy]acetic acid
4-({[2-(phenylamino)pyrimidin-5-yl]formamido}methyl)benzoic acid
2-{[(5-cyclopropyl-1H-pyrazol-3-yl)methyl](methyl)amino}-2-(2,3-dihydro-1-benzofuran-7-yl)acetic acid
2-phenyl-1-{2-phenylimidazo[1,2-a]pyridine-6-carbonyl}azetidine
(2R,4S)-4-hydroxy-1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]piperidine-2-carboxylic acid
1-[(3-ethyl-4,5-dihydro-1,2-oxazol-5-yl)methyl]-6-(ethylamino)-1H,4H,5H,8H-imidazo[4,5-e][1,3]diazepine-4,8-dione
N-cyclopropyl-2-methoxy-N-({3-[2-(piperidin-1-yl)ethoxy]phenyl}methyl)benzamide
N-(4-methoxyphenyl)-1-[4-(trifluoromethyl)pyridin-2-yl]piperidin-3-amine
1-[(2,3-difluorophenyl)methyl]-3-hydroxy-3-{[methyl(1,2-oxazol-3-ylmethyl)amino]methyl}piperidin-2-one
[(3R,4R)-1-[5-chloro-3-(trifluoromethyl)pyridin-2-yl]-4-(morpholin-4-ylmethyl)pyrrolidin-3-yl]methanol
4-[2-amino-3-cyano-5-ethyl-6-(propan-2-yl)pyridin-4-yl]benzamide
1-{5-[3-(3-chlorophenyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}azetidin-3-ol
5-[(2H-1,3-benzodioxol-5-yloxy)methyl]-N-[(4-methyl-1,3-thiazol-2-yl)methyl]-1H-pyrazole-3-carboxamide
(1R,7S)-3-cycloheptyl-N-methyl-N-[(3-methylpyridin-2-yl)methyl]-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
2-(4-acetyl-1,4-diazepan-1-yl)-2-[2-(trifluoromethoxy)phenyl]acetic acid
(2R,6S)-2,6-dimethyl-4-{[3-(4-phenylphenyl)-1H-pyrazol-4-yl]methyl}morpholine
(1S,5R)-6-benzyl-3-[2-(pyridin-3-yl)acetyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
methyl 6-[2-(3,5-difluorophenyl)acetyl]-2-(piperidine-1-sulfonyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
2-(2,3-dihydro-1H-inden-1-yl)-N-[(2-ethoxypyridin-3-yl)methyl]acetamide
N-{[6-(dimethylamino)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl}-3-(2-methoxyphenyl)-N-(oxolan-2-ylmethyl)propanamide
6-(3,6-dimethyl-1-benzofuran-2-carbonyl)-N,1-dimethyl-1H,4H,5H,6H,7H-pyrrolo[2,3-c]pyridine-2-carboxamide
5-{2-[1-(2-chlorophenyl)-1H-1,2,4-triazol-5-yl]ethyl}-4,6-dimethylpyrimidin-2-ol
6-[(1S,5R)-7-oxo-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]pyridine-2-carbonitrile
3-(2-methyl-1H-1,3-benzodiazol-6-yl)-1-[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)ethyl]urea
N-[3-(4-methylphenyl)propyl]-3-(1-methylpiperidin-2-yl)propanamide
2-(1H-indol-4-yl)-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
1-methyl-5-{[2-(propan-2-yloxy)ethyl]amino}-N-(thiophen-2-ylmethyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
1-[5-({2-methylimidazo[1,2-a]pyridin-3-yl}methyl)-3-(propan-2-yl)-1H-1,2,4-triazol-1-yl]butan-2-ol
5-[4-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidine-1-carbonyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
(2S)-N-[4-(1,3-benzoxazol-2-yl)phenyl]-1-(1,3-thiazol-4-ylmethyl)pyrrolidine-2-carboxamide
N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-3-(3-hydroxy-3-methylbutyl)-N-methylbenzamide
1-(diethylamino)-3-(2-methoxy-4-{[(3-methoxypropyl)amino]methyl}phenoxy)propan-2-ol
N-[(2R,3R)-2-hydroxy-1'-[(8-methoxyquinolin-2-yl)methyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]benzamide
1-{3-[5-phenyl-2-(pyridin-4-yl)pyrimidin-4-yl]piperidin-1-yl}ethan-1-one
[(5-chloro-2,4-dimethoxyphenyl)methyl](ethyl)[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]amine
2-[3,5-bis(trifluoromethyl)phenyl]-5-(pyrrolidine-1-carbonyl)pyrimidin-4-ol
N-cyclopropyl-N-[(2-methoxyphenyl)methyl]-2-(1H-pyrazol-1-yl)butanamide
1'-(1,4-dioxane-2-carbonyl)spiro[indene-1,4'-piperidine]
(4aS,8aR)-6-(4-fluorobenzoyl)-1-(4-hydroxybutyl)-decahydro-1,6-naphthyridin-2-one
ethyl 4-(6-methyl-3-{[(2-phenylpropyl)amino]methyl}quinolin-2-yl)piperazine-1-carboxylate
1-[5-(propan-2-yl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carbonyl]-1,4-diazepan-5-one
N-{3-[(2R,3R,6R)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]propyl}methanesulfonamide
(1S,5R)-3-(3,5-difluoropyridine-2-carbonyl)-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
3-{4-[4-ethyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}-5-fluoropyridine