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(3R,9aR)-3-benzyl-8-{[4-(4-fluorophenyl)-1,3-thiazol-2-yl]methyl}-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
1-(2,3-dihydro-1H-inden-2-yl)-4-{4H,5H,6H,7H-pyrazolo[1,5-a]pyridine-3-carbonyl}-1,4-diazepane
(3ar,6ar)-N-(2,1,3-benzothiadiazol-5-ylmethyl)-N-methyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
9-{5-[(diethylamino)methyl]-2-methylfuran-3-carbonyl}-2-methyl-2,9-diazaspiro[5.5]undecan-3-one
8-{[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]methyl}-1-methyl-3-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[(5-ethylpyridin-2-yl)methyl]-3-fluoro-4-hydroxy-N-methylbenzamide
2-phenyl-1-{3-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
N-(2H-1,3-benzodioxol-5-ylmethyl)-3-(4-methyl-4H-1,2,4-triazol-3-yl)-N-(pyridin-3-ylmethyl)propanamide
2-methyl-4-[4-({methyl[(5-methyl-1,2-oxazol-3-yl)methyl]amino}methyl)phenyl]butan-2-ol
5-methoxy-1-methyl-N-{pyrazolo[1,5-a]pyrimidin-3-ylmethyl}-1H-indole-2-carboxamide
1-[(1-methyl-1H-imidazol-2-yl)methyl]-4-{1-[(2-methylphenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}piperazine
6-chloro-N-methyl-N-(pyrazin-2-ylmethyl)-2-(1H-pyrazol-4-yl)quinoline-4-carboxamide
3-cyclopropyl-5-[2-(1H-imidazol-4-yl)-1-(1H-pyrrol-1-yl)ethyl]-1-phenyl-1H-1,2,4-triazole
3-({2-[1-(ethanesulfonyl)piperidin-3-yl]-1H-imidazol-1-yl}methyl)pyridine
N-[(5-methyl-1,2-oxazol-3-yl)methyl]-3-(4-methylpiperazine-1-carbonyl)benzene-1-sulfonamide
2-amino-1-(4-{5-[(4-hydroxypiperidin-1-yl)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-2-methylpropan-1-one
(2R)-N-{[4-(3-fluorophenyl)-5-(pyridin-2-yl)-1H-imidazol-2-yl]methyl}-5-oxopyrrolidine-2-carboxamide
4-[3-(4-chlorophenyl)-2-(methoxymethyl)-7-oxo-4H,7H-pyrazolo[1,5-a]pyrimidin-5-yl]pyrrolidin-2-one
2-{3-[2-(2,6-difluorophenyl)ethyl]piperidin-1-yl}-N,N-dimethylacetamide
4-benzyl-3-[1-(4-methylpyrimidin-2-yl)piperidin-4-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one
1-methyl-N-[1-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-yl]-1H-indole-6-carboxamide
N-methyl-N-(2-phenylethyl)-1-(1-propyl-1H-pyrazole-5-carbonyl)piperidin-3-amine
(2R,6R)-11-methoxy-4-(1H-pyrrole-3-carbonyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl](1-methoxypropan-2-yl)amine
N-[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]-2-{1-[(5-methylfuran-2-yl)methyl]-3-oxopiperazin-2-yl}acetamide
2-chloro-5-methyl-N-{[1-(propan-2-yl)piperidin-4-yl]methyl}benzamide
2-(5-{1-[2-(1H-imidazol-4-yl)ethyl]-1H-imidazol-2-yl}furan-2-yl)-1-methyl-1H-1,3-benzodiazole
4-[7-(dimethyl-1,3-thiazole-5-carbonyl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl]morpholine
8-benzyl-3-[3-(dimethylamino)propyl]-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
8-[(3-chloro-4-hydroxyphenyl)methyl]-2-cyclopropanecarbonyl-2,8-diazaspiro[4.5]decane-3-carboxylic acid
1-methyl-5-[2-(trifluoromethoxy)phenyl]-1H,4H-pyrazolo[3,4-d]imidazole
(2S,3R)-2-amino-3-hydroxy-N-{[2-(2-methoxyphenoxy)pyridin-3-yl]methyl}butanamide
(4aS,8aR)-1-(2-aminoethyl)-6-[(2,3-difluorophenyl)methyl]-decahydro-1,6-naphthyridine-4a-carboxylic acid
N-{2-ethyl-7-[3-(2-methylphenyl)piperidine-1-carbonyl]-1-(pyridin-3-ylmethyl)-1H-1,3-benzodiazol-5-yl}acetamide
2-[3-(1H-pyrazol-3-yl)phenyl]-4-(pyrrolidine-1-carbonyl)pyridine
4-({1-[(7-methyl-2,3-dihydro-1,4-benzodioxin-6-yl)methyl]piperidin-2-yl}methyl)morpholine
2-[(1E)-pent-1-en-1-yl]-N-(propan-2-yl)pyrimidin-4-amine
1-{[4-(methylamino)pyrimidin-2-yl]amino}-3-phenylpropan-2-ol
N-{2-[(1S,2S,4S)-bicyclo[2.2.1]hept-5-en-2-yl]ethyl}-3-(4H-1,2,4-triazol-4-yl)benzamide
1-[4-(1-benzofuran-2-yl)pyrimidin-2-yl]-5-cyclopropyl-N-[2-(diethylamino)ethyl]-1H-pyrazole-4-carboxamide
4-ethyl-3-({1-[1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]piperidin-4-yl}methyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
2-ethyl-1-[(4-methoxyphenyl)methyl]-6-methyl-3-(4-phenylazepane-1-carbonyl)-1,4-dihydropyridin-4-one
6-tert-butyl-1-methyl-N-[2-(4-methyl-1H-pyrazol-1-yl)propyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
7-(cyclopentylmethyl)-N4-(1,3-thiazol-2-ylmethyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine
2-[4-(2-fluoro-5-methoxyphenyl)-3,5-dimethyl-1H-pyrazol-1-yl]acetic acid
2-(5-chloro-2-methoxyphenyl)-2-[4-(pyrrolidine-1-carbonyl)piperidin-1-yl]acetic acid
(2R)-2-amino-4-methyl-N-({2-[3-(trifluoromethyl)phenoxy]pyridin-3-yl}methyl)pentanamide
5-(2-methoxypyridin-3-yl)-4-methyl-2-(4H-1,2,4-triazol-4-yl)pyridine
N-({5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}methyl)-3,4-dihydro-2H-1-benzopyran-3-amine
4-{pyrazolo[1,5-a]pyrimidin-3-yl}-N-(pyridin-2-ylmethyl)-1H-pyrrolo[2,3-b]pyridin-6-amine