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3-(4-{[2-(2-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methoxy}phenyl)-1,3-oxazolidin-2-one
[(5-{[(1R,5R)-3-benzoyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}thiophen-3-yl)methyl]dimethylamine
5,6-dimethyl-N-[2-(pyridin-3-yloxy)propyl]pyrimidin-4-amine
N-[(4-benzyl-5-{[(2-chlorophenyl)methyl]sulfanyl}-4H-1,2,4-triazol-3-yl)methyl]-2-(3-methyl-1H-pyrazol-1-yl)acetamide
1-[1-(dimethylsulfamoyl)piperidin-4-yl]-N-(pyridin-2-ylmethyl)piperidine-3-carboxamide
4-(4-methylphenoxy)-1-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperidine
2-amino-4-[2-(ethylsulfanyl)pyrimidin-5-yl]-6-(4-hydroxyphenyl)pyridine-3-carbonitrile
1-[(3S,4R)-3-benzyl-4-hydroxy-4-methylpiperidin-1-yl]-2-(4-methyl-1H-pyrazol-1-yl)ethan-1-one
1-(1H-indazol-6-yl)-4-[2-(4-methylphenoxy)acetyl]piperazin-2-one
N-(1-methyl-1H-indazol-5-yl)-4-(pyrimidin-2-yl)-1,4-diazepane-1-carboxamide
N-[(6-fluoro-1H-1,3-benzodiazol-2-yl)methyl]-N-methyl-2-[1-(3-methylbutyl)-3-oxopiperazin-2-yl]acetamide
1-(oxan-4-yl)-N-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}piperidine-3-carboxamide
1-(furan-2-yl)-2-[(2R,3R,6R)-3-(4-methylphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]ethane-1,2-dione
(2S,4R)-4-(3-cyanobenzamido)-N-ethyl-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]pyrrolidine-2-carboxamide
(3S,4S)-1-[5-(3-methyl-1,2,4-oxadiazol-5-yl)pyridin-2-yl]-4-(naphthalen-2-yl)piperidin-3-ol
1-(2-chlorophenyl)-4-[(3R)-3-hydroxy-3-phenylpropyl]piperazin-2-one
N-(2-methoxyethyl)-N-propyl-2-(pyridin-3-yl)pyrimidine-5-carboxamide
1-(4-aminopyrimidin-2-yl)-4-(2-methoxyphenoxy)piperidine-4-carboxylic acid
(2R,3S,6R)-3-(2-methoxyphenyl)-5-(3-methylfuran-2-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
6-(4-fluorophenyl)-N-[(2S)-1-hydroxypropan-2-yl]-8-oxo-7-(prop-2-en-1-yl)-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
2-[(3R)-3-hydroxy-3-phenylpropyl]-5-(1,2,3,4-tetrahydroisoquinolin-2-yl)-2,3-dihydropyridazin-3-one
[(3R,4R)-4-({[2-(dimethylamino)ethyl](methyl)amino}methyl)-1-(2,5-dimethylfuran-3-carbonyl)pyrrolidin-3-yl]methanol
[1-(2,6-difluoro-3-methoxybenzoyl)-3-propylpiperidin-3-yl]methanol
N-[(2,4-dichloro-6-methylphenyl)methyl]-2-(piperidin-4-yl)acetamide
N-(cyclohex-1-en-1-ylmethyl)-4-(piperidin-1-yl)butanamide
(1-{4-[4-(2-chlorophenyl)piperidin-4-yl]pyrimidin-2-yl}piperidin-4-yl)methanol
3-(1H-pyrazol-1-ylmethyl)-N-[2-(pyridin-3-ylformamido)ethyl]benzamide
1-(2-chloro-5-methylbenzoyl)-4-(cyclopropylmethyl)-3-(propan-2-yl)-1,4-diazepan-5-one
ethyl 1-benzyl-5-[(3-hydroxyphenyl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
3-(4-methoxyphenyl)-N-[(3-methylpyridin-2-yl)methyl]-3-phenylpropanamide
2-(1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}pyrrolidin-2-yl)-1,3-thiazole
methyl (2S)-2-[methyl({2-methyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl})amino]propanoate
4-(2-benzyl-1,3-thiazole-4-carbonyl)-2-(1H-pyrazol-1-ylmethyl)-1,4-oxazepane
N-[2-(1H-imidazol-4-yl)ethyl]-6-methoxy-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
[(3R,4R)-1-(2-methyl-5-propylpyrimidin-4-yl)-4-(pyrrolidin-1-ylmethyl)pyrrolidin-3-yl]methanol
1-{3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-(2-methylphenyl)ethan-1-one
2-[3-(3-chlorophenyl)-1-methyl-1H-pyrazol-4-yl]-5-methyl-1H-1,3-benzodiazole
N-[(1S,3aS,6aS)-octahydropentalen-1-yl]-2,4-dioxo-1,2,3,4-tetrahydropyrimidine-5-carboxamide
N-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-(3-methyl-5,6-dihydro-1,4-dioxine-2-carbonyl)piperidin-3-amine
N-[(5-{[5-(4-methylphenyl)furan-2-yl]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl)methyl]acetamide
1-{2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}-4-(pyridin-3-ylmethyl)-1,4-diazepane
2-methyl-6-{1-[2-(2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)acetyl]piperidin-4-yl}-3,4-dihydropyrimidin-4-one
2-{3-[5-(4-methyl-1H-imidazol-5-yl)-4-phenyl-1H-imidazol-1-yl]propyl}phenol
5-{4-[(4-cyclopentyl-1H-1,2,3-triazol-1-yl)methyl]piperidine-1-carbonyl}-2-methylpyrimidine
4-[7-(cyclobutylmethyl)-6-oxo-2,7-diazaspiro[4.5]decane-2-carbonyl]-1λ6-thiane-1,1-dione
2-[(4aS,7aS)-octahydro-1H-pyrrolo[3,4-b]pyridine-6-carbonyl]-3-ethyl-1H-indole
4-{[2-(4-fluorophenyl)azetidin-1-yl]methyl}-1H-pyrazole-3-carboxylic acid
(1S,3R)-3-amino-N-[3-(2-ethyl-2H-1,2,3,4-tetrazol-5-yl)phenyl]cyclopentane-1-carboxamide
(2S,4S)-4-amino-1-[(2S)-2-methoxy-2-phenylacetyl]-N-methylpyrrolidine-2-carboxamide
4-phenyl-N-[1-(1-{[4-(propan-2-yl)-1,3-thiazol-2-yl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]butanamide