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4-{[4-methoxy-3-(methoxymethyl)phenyl]methyl}-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
4-methyl-2-{1-[3-(1H-1,2,3,4-tetrazol-1-yl)-1H-pyrazole-4-carbonyl]piperidin-3-yl}-1H-1,3-benzodiazole
N-[(3S,4R)-1-[2-(1-methyl-1H-pyrrol-2-yl)-2-oxoacetyl]-4-(5-methylfuran-2-yl)pyrrolidin-3-yl]acetamide
1-[3-(2-chlorophenyl)propyl]-4-(pyridin-2-yl)piperidin-4-ol
1-{5-[(cyclobutylamino)methyl]-2-methoxyphenoxy}-3-(4-methyl-1,4-diazepan-1-yl)propan-2-ol
{[3-(1-benzofuran-2-yl)-1-benzyl-1H-pyrazol-4-yl]methyl}(methyl)[2-(2-methyl-1H-imidazol-1-yl)ethyl]amine
1-[1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]-3-propylpiperidine-3-carboxylic acid
N-[(3,5-dimethyl-2-phenyl-1H-indol-7-yl)methyl]-2-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)acetamide
1-(2-methoxyphenyl)-4-[1-(2-phenylethyl)piperidin-3-yl]piperazine
7-chloro-4-(1,4-diazepane-1-carbonyl)-2-(furan-2-yl)-8-methylquinoline
N-(adamantan-1-yl)-1-(piperidin-3-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
1-[1-(1-benzothiophene-5-carbonyl)azetidin-3-yl]-3,5-dimethyl-1H-pyrazole
4-[(3-ethyl-1H-pyrazol-5-yl)methyl]-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-({8-[(3,5-dimethoxyphenyl)methyl]-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)pyridine-3-carboxamide
5-methyl-1-(4-methylphenyl)-4-[3-(1-methylpiperidin-4-yl)propanoyl]piperazin-2-one
1-[(3R,4R)-3-[(dimethylamino)methyl]-4-(hydroxymethyl)pyrrolidin-1-yl]-3-[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]propan-1-one
2-(3-hydroxypropyl)-9-(5-phenyl-1,2,4-oxadiazol-3-yl)-2,9-diazaspiro[5.5]undecan-3-one
1-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-N-[3-(1,3-thiazol-4-yl)phenyl]piperidine-4-carboxamide
3-(2,5-dimethoxyphenyl)-1-{pyrazolo[1,5-a]pyridine-3-carbonyl}pyrrolidine
1-(5-{4H,5H,6H,7H-thieno[3,2-c]pyridin-5-ylmethyl}imidazo[2,1-b][1,3]thiazole-6-carbonyl)piperidine
1-[1-(2-hydroxyethyl)-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-5-yl]-3-phenoxypropan-1-one
5-methyl-N-{2-[1-(pyridin-4-ylmethyl)piperidin-3-yl]ethyl}pyridine-3-carboxamide
2-(1H-pyrazol-1-yl)-N-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)butanamide
1-{[2-methyl-4-(1H-pyrazol-1-yl)phenyl]methyl}-4-(pyridin-4-ylmethyl)-1,4-diazepane
1-{2-[4-(2-phenylpropyl)piperazin-1-yl]ethyl}-N-(propan-2-yl)-1H-1,2,3-triazole-4-carboxamide
4-[(2,6-difluorophenyl)methyl]-7-(3,6-dimethylpyrazin-2-yl)-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-{2-[3-cyclopropyl-1-(3,4-dimethylphenyl)-1H-1,2,4-triazol-5-yl]ethyl}methanesulfonamide
N-methyl-N-[1-(3-phenylpropyl)piperidin-3-yl]-1H-1,2,3-benzotriazole-5-carboxamide
3-{[4-(5-chloropyrimidin-2-yl)piperazin-1-yl]methyl}quinolin-7-ol
2-chloro-5-acetamido-N-methyl-N-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]benzamide
N-{[2-(1H-imidazol-1-yl)phenyl]methyl}-3-methanesulfonylbenzamide
2-(morpholin-3-yl)-1-{4-[(pyridin-2-yl)amino]piperidin-1-yl}ethan-1-one
1-(4-methoxyphenyl)-4-{1-[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]piperidin-3-yl}piperazine
4-[1-(1-{[4-(1H-imidazol-1-yl)phenyl]methyl}piperidin-4-yl)ethyl]morpholine
3-(2-{4-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2-oxoethyl)-1,3-oxazolidin-2-one
1-(4-{[3-(oxolan-3-yl)-1H-1,2,4-triazol-5-yl]methyl}phenyl)-1H-1,2,3,4-tetrazole
N-[(3-methoxyphenyl)methyl]-2-[methyl(pyridin-3-ylmethyl)amino]-N-(prop-2-en-1-yl)acetamide
N-{[2-(dimethylamino)pyridin-3-yl]methyl}-1-ethyl-3-methyl-1H-pyrazole-5-carboxamide
2-(1,3-dimethyl-2,5-dioxoimidazolidin-4-yl)-N-[3-(1-methyl-1H-1,3-benzodiazol-2-yl)propyl]acetamide
2-ethyl-N-[2-(pyridin-3-yl)ethyl]-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
1-({3-[3-(1H-imidazol-1-yl)propoxy]phenyl}methyl)-N,N-dimethylpiperidin-3-amine
1-methyl-3-(propan-2-yl)-N-[1-(thian-4-yl)piperidin-4-yl]-1H-pyrazole-5-carboxamide
(1R,9S)-5-amino-3-[5-(3-hydroxy-3-methylbut-1-yn-1-yl)thiophen-2-yl]-6,12-diazatricyclo[7.2.1.02,7]dodeca-2(7),3,5-triene-4-carbonitrile
1,4,6-trimethyl-2-oxo-N-(2-{5H,6H,7H-[1,3]thiazolo[3,2-a]pyrimidin-3-yl}ethyl)-1,2-dihydropyridine-3-carboxamide
1-{2-[(2H-1,3-benzodioxol-5-ylmethyl)amino]ethyl}-N-(2-methylphenyl)-1H-1,2,3-triazole-4-carboxamide
2-(3-fluoro-4-methoxyphenyl)-N-(propan-2-yl)benzamide
3-{2-[(2-methylphenyl)sulfanyl]acetyl}-3,9-diazaspiro[5.6]dodecan-10-one
4-(2-butyl-1H-imidazol-4-yl)-3-cyclobutyl-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
2-methoxy-1-{1'-[(3-methyl-1,2-oxazol-5-yl)methyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}ethan-1-one
N,2-dimethyl-6-(2-methylpropyl)-N-[2-(pyridin-4-yl)ethyl]pyrimidine-4-carboxamide