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N-(1,3-benzoxazol-2-ylmethyl)-N-methyl-1-(oxolan-2-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
N-{[2-(4-acetylpiperazin-1-yl)-6-methylquinolin-3-yl]methyl}-N-[2-(cyclohex-1-en-1-yl)ethyl]cyclopropanecarboxamide
{2-[3-(3-methoxypropyl)piperidin-1-yl]-1,3-thiazol-4-yl}methanol
1-(5-ethyl-2-methylpyrimidin-4-yl)-N-[3-(4-methyl-1,3-thiazol-2-yl)propyl]piperidin-4-amine
2-(2-methyl-1,3-thiazol-4-yl)-5-[(1S,5R)-1,3,3-trimethyl-6-azabicyclo[3.2.1]octane-6-carbonyl]pyrimidin-4-ol
N-({2-[4-(pyridin-2-yl)piperazin-1-yl]pyridin-3-yl}methyl)-3-(1H-1,2,4-triazol-1-yl)propanamide
N-[1-(3-ethyl-1,2,4-oxadiazol-5-yl)ethyl]-5-(propan-2-yl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
3-phenyl-3-{[5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]amino}propan-1-ol
(1S,5R)-3-(pyridin-4-ylmethyl)-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N,N-dimethyl-7-(3-methylbenzoyl)-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
N-(1-{[4-(2-methylpropyl)phenyl]methyl}piperidin-3-yl)-3-(1H-1,2,3,4-tetrazol-1-yl)propanamide
3-{2-[(5-tert-butyl-1,3,4-oxadiazol-2-yl)amino]ethyl}-1,3-oxazinan-2-one
N-[(3R,5S)-5-(diethylcarbamoyl)-1-methylpyrrolidin-3-yl]-2-oxo-1,2-dihydroquinoline-4-carboxamide
N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-N-(propan-2-yl)-2-(pyrrolidin-1-yl)benzamide
[1-(2-{[2-(trifluoromethyl)pyrimidin-4-yl]amino}ethyl)piperidin-2-yl]methanol
3-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}-3-methyl-1-[4-(2-methyl-1H-imidazol-1-yl)phenyl]urea
5-amino-N-(2,3-dihydro-1-benzofuran-2-ylmethyl)-N-methyl-4-phenyl-1H-pyrazole-3-carboxamide
2-[(6-chloro-2-fluoro-3-methoxyphenyl)methyl]-2,7-diazaspiro[4.5]decane
4-[2-(2-hydroxyphenoxy)acetyl]-5-methyl-1-(4-methylphenyl)piperazin-2-one
N-{1-[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]ethyl}-3-(5-methylfuran-2-yl)-1H-pyrazole-5-carboxamide
(3S,4S)-1-[4-(3-hydroxy-3-methylbutyl)benzoyl]-4-(pyrrolidin-1-yl)pyrrolidin-3-ol
8-[(dimethyl-1H-1,2,4-triazol-5-yl)methyl]-8-azaspiro[4.5]decane-7,9-dione
3-methyl-N-[2-(2-methylpropanesulfonyl)ethyl]-[1,2]oxazolo[5,4-d]pyrimidin-4-amine
(1R,2S)-1-({6-cyclopentyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)-2,3-dihydro-1H-inden-2-ol
N-methyl-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-2-(2,5,7-trimethyl-1H-indol-3-yl)acetamide
5-[3-(diethylcarbamoyl)phenyl]thiophene-2-carboxamide
3-(2H-1,3-benzodioxol-5-yl)-N-[2-(1H-imidazol-4-yl)ethyl]-3-phenylpropanamide
{[3-(4-fluorophenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}[2-(pyridin-4-yl)ethyl]amine
N-[(1,5-dimethyl-1H-indazol-3-yl)methyl]-1,9-dioxaspiro[5.5]undecan-4-amine
4-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}-1-(4-methylphenyl)piperazin-2-one
3-(4-fluorophenyl)-4-{6-methyl-4-oxo-4H-pyrido[1,2-a]pyrimidine-3-carbonyl}piperazin-2-one
methyl 3-[({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)(oxolan-2-ylmethyl)carbamoyl]propanoate
5-cyclohexaneamido-1-(2-methoxyethyl)-N-[2-(pyridin-3-yl)ethyl]-1H-1,3-benzodiazole-7-carboxamide
N-(2-hydroxypropyl)-4-{[1-(2-phenylethyl)piperidin-4-yl]oxy}benzamide
2-(1-{[5-methyl-2-(5-methylfuran-2-yl)-1,3-oxazol-4-yl]methyl}piperidin-3-yl)-1,3-benzoxazole
5-[methyl(2-phenylethyl)amino]-2-{[2-(methylamino)-1,3-thiazol-4-yl]methyl}-2,3-dihydropyridazin-3-one
4-(2,3-dihydro-1H-indene-5-carbonyl)-1-[(2-fluorophenyl)methyl]piperazin-2-one
3-methoxy-6-{[1-(pyrrolidin-1-yl)hex-5-en-2-yl]oxy}pyridazine
N-benzyl-3-[(3-hydroxyazetidin-1-yl)methyl]-N-methylimidazo[1,2-a]pyridine-2-carboxamide
1-(carbamoylmethyl)-N-[1-(4-ethoxy-3-fluorophenyl)ethyl]piperidine-4-carboxamide
N-(furan-3-ylmethyl)-N,1-dimethyl-2-oxo-1,2,5,6,7,8-hexahydroquinoline-3-carboxamide
N-[1-(methoxymethyl)cyclopentyl]-1-methyl-5-phenyl-1H-pyrazole-3-carboxamide
N,N-dimethyl-6-[4-(propan-2-yloxy)phenyl]pyridine-3-carboxamide
(2R)-1-({4-[(2,3-dihydro-1H-inden-4-yl)carbamoyl]phenyl}methyl)pyrrolidine-2-carboxamide
N-{4-[({[(1R,2R)-2-hydroxycyclohexyl]methyl}carbamoyl)methyl]phenyl}butanamide
2-(3,4-dimethylphenoxy)-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]acetamide
(2E)-N-({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)-4-methyl-N-(oxolan-2-ylmethyl)pent-2-enamide
{[5-(1,5-dimethyl-1H-pyrrol-2-yl)-1,3,4-oxadiazol-2-yl]methyl}({[2-(1H-1,2,4-triazol-1-yl)pyridin-3-yl]methyl})amine
N-(2,1,3-benzoxadiazol-5-ylmethyl)-3-(4-hydroxyphenyl)-N-methyl-1H-pyrazole-5-carboxamide
(4aR,8aR)-2-cyclobutanecarbonyl-7-[(2,5-difluorophenyl)methyl]-decahydro-2,7-naphthyridin-4a-ol