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N-(2-methoxyethyl)-N-[(5-methylthiophen-2-yl)methyl]-1-oxo-1,2-dihydroisoquinoline-4-carboxamide
methyl 4-[4-(1-methyl-6-oxo-1,6-dihydropyridine-3-carbonyl)piperazin-1-yl]benzoate
[2-(1H-1,2,3-benzotriazol-1-yl)ethyl]({[2-(naphthalen-2-yl)pyrimidin-5-yl]methyl})amine
4-[3-({1-[6-methyl-2-(propan-2-yl)pyrimidin-4-yl]piperidin-4-yl}amino)propyl]phenol
N-[(3S,4R)-4-(5-methylfuran-2-yl)-1-[3-(pyridin-3-yl)propanoyl]pyrrolidin-3-yl]acetamide
(1R,2S)-2-[3-(carbamoylmethyl)-1-(3,4-dimethylphenyl)-1H-1,2,4-triazol-5-yl]-N-methylcyclohexane-1-carboxamide
[(4-fluoro-3-methoxyphenyl)methyl]({[1-(2-methoxyethyl)piperidin-4-yl]methyl})(pyridin-4-ylmethyl)amine
2-(1-{5H,6H-benzo[h]quinazolin-2-yl}-5-cyclopropyl-1H-pyrazole-4-carbonyl)-7-methyl-2,7-diazaspiro[4.4]nonane
3-(5-fluoro-1H-1,3-benzodiazol-2-yl)-1-(1,2-oxazinan-2-yl)propan-1-one
N-[(4-fluorophenyl)methyl]-3-(4-methylpiperazine-1-carbonyl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
2-(2-{[5-methyl-4-(1-methyl-1H-1,2,4-triazol-5-yl)pyrimidin-2-yl]amino}ethyl)-3,4-dihydroquinazolin-4-one
N-phenyl-3-[1-(thiophene-3-sulfonyl)piperidin-4-yl]propanamide
2-benzyl-8-[2-(methylamino)pyrimidine-5-carbonyl]-2,8-diazaspiro[4.5]decan-3-one
2-fluoro-6-methoxy-4-({methyl[(3-methylthiophen-2-yl)methyl]amino}methyl)phenol
4-(5-methylpyrazine-2-carbonyl)-3,4-dihydro-2H-1,4-benzoxazine
2-{1-[(3,4-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-(3-hydroxy-2,2-dimethylpropyl)acetamide
(3S,4S)-1-{1-methyl-6-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-4-(4-methylpiperazin-1-yl)pyrrolidin-3-ol
N-[(4-fluorophenyl)methyl]-3-{imidazo[1,2-a]pyridin-2-yl}propanamide
4-[3-({5-methylpyrazolo[1,5-a]pyrimidin-7-yl}amino)propyl]-1,3-thiazol-2-amine
2-{methyl[2-(4-methyl-1,3-thiazol-5-yl)ethyl]amino}-2-[6-(piperidin-1-yl)pyridin-3-yl]acetic acid
6-methyl-N-[(2-methyl-1,3-thiazol-4-yl)methyl]-2-(4-methylphenoxymethyl)-1-[2-(morpholin-4-yl)ethyl]-4-oxo-1,4-dihydropyridine-3-carboxamide
(1S,5R)-3-[(4-fluorophenyl)methyl]-6-(2-methoxypyridine-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
3-methyl-N-{[2-(morpholin-4-yl)-6H,7H,8H-cyclopenta[g]quinolin-3-yl]methyl}-N-[3-(2-oxopyrrolidin-1-yl)propyl]thiophene-2-carboxamide
2-[4-(3-phenylpropyl)morpholin-3-yl]acetic acid
1-{4-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2-(3-fluorophenyl)ethan-1-one
8-fluoro-2-{[4-(3-methylpyridin-2-yl)piperazin-1-yl]methyl}quinolin-4-ol
7-fluoro-N-{2-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]ethyl}-2-methylquinoline-4-carboxamide
1-methyl-8-{5-[(methylsulfanyl)methyl]furan-2-carbonyl}-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
2-(3,4-dimethoxyphenyl)-N-methyl-N-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}acetamide
N-[4-(1H-1,3-benzodiazol-2-yl)phenyl]-1-[(2-methyl-1,3-thiazol-5-yl)methyl]piperidine-4-carboxamide
1-[4-(4-methoxybenzoyl)piperazin-1-yl]-3-(3-methyl-1H-pyrazol-1-yl)propan-1-one
N-[3-(4-chloro-3,5-dimethyl-1H-pyrazol-1-yl)propyl]-5-methanesulfonyl-2-methylpyrimidin-4-amine
3-(1-benzyl-5-oxopyrrolidin-3-yl)-4-[(3-methylphenyl)methyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
2-fluoro-N-({3-methyl-7-[2-(1H-pyrazol-1-yl)benzoyl]-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)benzamide
N-[3-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]-1-[(3-methyl-1H-1,2,4-triazol-5-yl)methyl]piperidine-4-carboxamide
1-{imidazo[2,1-b][1,3]thiazole-6-amido}-1,2,3,4-tetrahydronaphthalene-1-carboxylic acid
2-(3-{[methyl({[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl})amino]methyl}phenoxy)acetamide
[({4-[4-(2-methoxyphenyl)piperazin-1-yl]quinazolin-2-yl}methyl)sulfamoyl]dimethylamine
4-[1-(2-methyl-1H-1,3-benzodiazol-6-yl)-1H-imidazol-2-yl]-2,1,3-benzoxadiazole
6-{[3-(1H-pyrazol-1-yl)propyl]amino}-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3(8),6,12,14-pentaen-4-one
2-[(1,1-dioxo-1λ6-thian-3-yl)methyl]benzene-1-sulfonamide
2-{[3-(pyridin-3-yl)azetidin-1-yl]methyl}-1H-1,3-benzodiazole
3-chloro-N-methyl-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}thiophene-2-carboxamide
4-[4-(4-fluorophenyl)-1,2,3,6-tetrahydropyridine-1-carbonyl]-N-methylpyridin-2-amine
(2S,3R)-3-hydroxy-2-[(2-{[(2-methyl-1,3-benzothiazol-5-yl)oxy]methyl}-1,3-oxazol-4-yl)formamido]butanamide
6-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-N-propylpyridine-3-carboxamide
N-{2H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-3-[(4-fluorophenyl)formamido]-N-methylpropanamide
1-[2-methoxy-4-({[2-(pyridin-4-yl)ethyl]amino}methyl)phenoxy]-3-(morpholin-4-yl)propan-2-ol
(1R,3S)-3-methoxy-7-(5-propylthiophene-3-carbonyl)-7-azaspiro[3.5]nonan-1-ol
1-[2-({[(6-fluoro-1H-1,3-benzodiazol-2-yl)methyl](methyl)amino}methyl)phenoxy]-3-(piperidin-1-yl)propan-2-ol