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[1-(cyclohexylmethyl)-4-[(4-methoxyphenyl)methyl]piperidin-4-yl]methanol
N-[(4-chlorophenyl)methyl]-2-(2-hydroxypropanoyl)-1,2,3,4-tetrahydroisoquinoline-6-sulfonamide
2-({[(3-ethoxyphenyl)methyl](2-hydroxyethyl)amino}methyl)-6-methylpyridin-3-ol
{[1-butyl-2-(4-methylpentanesulfonyl)-1H-imidazol-5-yl]methyl}(methyl)[3-(morpholin-4-yl)propyl]amine
3-[3-(2-methoxyphenyl)phenyl]-1-methyl-1H-pyrazole
8-(2H-1,3-benzodioxol-5-ylmethyl)-2-cyclopropanecarbonyl-2,8-diazaspiro[4.5]decane-3-carboxylic acid
5-chloro-2-methoxy-4-[({1-[5-methyl-1-(naphthalen-1-yl)-1H-pyrazol-4-yl]ethyl}amino)methyl]phenol
(3R)-3,4,4-trimethyl-1-(2-methyl-1H-pyrrole-3-carbonyl)pyrrolidin-3-ol
1-cyclopropyl-4-{3-[(2-methylphenyl)methoxy]azetidine-1-carbonyl}pyrrolidin-2-one
3-acetyl-N-[1-(2,3-dihydro-1H-inden-2-yl)-2-methylpropan-2-yl]-1H-pyrazole-5-carboxamide
N-(4-methoxy-2-methylphenyl)-3-{1-[(3-methylpyridin-4-yl)methyl]piperidin-3-yl}propanamide
3-[(2-fluorophenyl)formamido]-N-[(5-methoxy-1,3-benzoxazol-2-yl)methyl]propanamide
1-(1-cyclopropyl-1H-pyrrole-2-carbonyl)-4-[2-(dimethylamino)ethyl]-1,4-diazepan-5-one
1-[3-(2,5-dimethoxyphenyl)pyrrolidin-1-yl]-3-(furan-2-yl)propan-1-one
3-[(3R,7S,8aS)-3-(2-methylpropyl)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-[(3-fluorophenyl)methyl]urea
3-{[benzyl(methyl)amino]methyl}-1-[(3,4-difluorophenyl)methyl]-3-hydroxypiperidin-2-one
[(3-cyclohexyl-1,2,4-oxadiazol-5-yl)methyl][1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]amine
{[2-(2-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]methylamine
2-(2-oxopyrrolidin-1-yl)-N-{[2-(pyrrolidin-1-yl)-1,3-thiazol-4-yl]methyl}propanamide
(2S)-2-amino-3-methoxy-N-[(2-methoxyphenyl)methyl]-N-(prop-2-en-1-yl)propanamide
N-[(3S,4S)-4-hydroxy-1-(propan-2-yl)pyrrolidin-3-yl]-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
2-{1-[(2-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]acetamide
N-[2-(4-ethylphenoxy)ethyl]-N-methyl-1H-pyrazole-3-carboxamide
2-(2-methyl-4-phenylpyridine-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
9-[(2-chloro-4-fluorophenyl)methyl]-2-(2-hydroxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
5-[(1S,5R)-3-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-1H-1,3-benzodiazole
N3-butyl-N5-[(3,4-difluorophenyl)methyl]-1-(furan-2-ylmethyl)-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
(4aS,8aR)-6-[6-methyl-2-(methylsulfanyl)pyrimidin-4-yl]-1-[2-(methylamino)ethyl]-decahydro-1,6-naphthyridin-2-one
2-(4-{[4-(methylsulfanyl)phenyl]methyl}piperazin-1-yl)pyrazine
4-(2,1,3-benzothiadiazol-4-yl)-1-methyl-3-(pyridin-2-yl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
N-(2,1,3-benzoxadiazol-5-ylmethyl)-2-[(propan-2-yl)amino]pyrimidine-5-carboxamide
1-(2,4-difluorobenzenesulfonyl)-2-[2-(1H-pyrazol-1-yl)ethyl]piperidine
2-(4-ethyl-3,5-dimethyl-1H-pyrazol-1-yl)-1-[2-(morpholine-4-carbonyl)piperazin-1-yl]ethan-1-one
5-[(2E)-3,7-dimethylocta-2,6-dien-1-yl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxylic acid
methyl (2S)-2-{[5-ethyl-4-(pyrrolidin-1-ylmethyl)furan-2-yl]formamido}-3-phenylpropanoate
4-(2,8-dimethylquinoline-4-carbonyl)-3-(1H-imidazol-4-ylmethyl)piperazin-2-one
2-{4-[3-(3-methylpiperidin-1-yl)-3-oxopropyl]piperazin-1-yl}pyridine-3-carbonitrile
N-ethyl-N-[2-(5-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-3-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanamide
3-(3,5-dimethyl-1H-pyrazol-1-yl)-N-[4-(furan-2-ylmethoxy)phenyl]azetidine-1-carboxamide
2-{1-[(4-fluorophenyl)methyl]-4-[(2-methoxyphenyl)methyl]piperazin-2-yl}ethan-1-ol
7-oxo-N-[(3R)-piperidin-3-yl]-7H-[1,3]thiazolo[3,2-a]pyrimidine-5-carboxamide
1-methyl-8-(2-phenylethyl)-3-(propan-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-(2,3-dihydro-1,4-benzodioxin-6-yl)-3-[2-(4-ethyl-3,5-dimethyl-1H-pyrazol-1-yl)ethyl]urea
N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-3-(2-methyl-1H-1,3-benzodiazol-1-yl)propanamide
4-(furan-2-yl)-N-methyl-N-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}benzamide
2-(2-{3-[1-(2-methoxyethyl)-1H-pyrazol-3-yl]phenyl}phenyl)-5-methyl-1,3,4-oxadiazole
3-(3-hydroxy-3-methylbut-1-yn-1-yl)-N-{2-[2-(thiophen-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]ethyl}benzamide
3-{1-[(1-methyl-1H-imidazol-2-yl)methyl]piperidin-3-yl}benzoic acid
2-(3-ethyl-4-methyl-1H-pyrazole-5-carbonyl)-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
1-{4-[(3-chlorophenyl)methyl]piperazin-1-yl}-2-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]ethan-1-one