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(3R,4R)-N-cyclohexyl-3-(hydroxymethyl)-4-{[(2-methoxyethyl)(methyl)amino]methyl}pyrrolidine-1-carboxamide
3-{1-[3-chloro-4-(pyrrolidin-1-yl)benzoyl]piperidin-3-yl}propanamide
1-[1-(2-hydroxyacetyl)piperidin-4-yl]-N-(oxolan-2-ylmethyl)piperidine-4-carboxamide
4-(2-methoxy-4-methylbenzoyl)-2-(6-methoxynaphthalen-2-yl)morpholine
3-[5-(1-benzofuran-3-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]propanoic acid
N-(2,5-dimethylphenyl)-3-[2-(3-methoxyphenyl)azetidin-1-yl]propanamide
N-cyclopentyl-4-oxo-4-[4-(pyridin-4-ylmethyl)-1,4-diazepan-1-yl]butanamide
5-{2-[(4aR,8aR)-octahydro-2H-1,4-benzoxazin-4-yl]-2-oxoethyl}-6-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-methyl-4-{2-[3-(2-methylpiperidin-1-yl)azetidin-1-yl]pyridine-4-carbonyl}piperazine
1-(1-methyl-1H-imidazole-2-carbonyl)-4-(4-propyl-1H-1,2,3-triazol-1-yl)piperidine
(3R,4S)-1-{3,6-dimethyl-[1,2]oxazolo[5,4-b]pyridine-4-carbonyl}-4-phenylpyrrolidin-3-amine
2-{1-[(dimethyl-1,2-oxazol-4-yl)sulfonyl]pyrrolidin-2-yl}pyridine
1-{[1,2,4]triazolo[1,5-a]pyrimidin-2-ylmethyl}-3-(trifluoromethyl)-1,2-dihydropyridin-2-one
5-[4-(5-chloro-2-methylphenyl)piperazine-1-carbonyl]-N-cyclohexyl-1-cyclopropyl-4-oxo-1,4-dihydropyridine-3-carboxamide
2-({1-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]piperidin-3-yl}formamido)acetamide
ethyl 1-(1-carbamoylcyclopropanecarbonyl)-3-(3-phenylpropyl)piperidine-3-carboxylate
2,4-dichloro-3-{[2-(2-hydroxyethyl)morpholin-4-yl]methyl}phenol
5-(oxolan-2-yl)-N-{[2-(pyrazin-2-yl)-1,3-thiazol-4-yl]methyl}thiophene-2-carboxamide
1-(4-fluorophenyl)-4-(5-methyl-1-propyl-1H-pyrazole-4-carbonyl)-1,4-diazepane
1-[1-(2-fluorobenzoyl)piperidin-4-yl]-N-(2-methylpropyl)-1H-1,2,3-triazole-4-carboxamide
4-[4-ethyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-[(4-methylphenyl)methyl]piperidine
8-(7-fluoro-2-oxo-1,2-dihydroquinoline-4-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
3-(isoquinolin-4-yl)-4H-chromen-4-one
1-[(4-methanesulfonylmorpholin-2-yl)methyl]-3-(2-methyl-1-benzofuran-7-yl)urea
N-[3-(azepane-1-carbonyl)phenyl]-4-methyl-1,4-diazepane-1-carboxamide
1-[(3R,4R)-4-[2-(3,5-dimethyl-1-benzofuran-2-yl)-1H-imidazol-1-yl]oxolan-3-yl]-4-methylpiperazine
(4aR,8aR)-2-cyclobutanecarbonyl-7-(furan-2-ylmethyl)-decahydro-2,7-naphthyridin-4a-ol
8-(5-cyano-4-methyl-6-oxo-1,6-dihydropyridine-3-carbonyl)-2-methyl-2,8-diazaspiro[4.5]decane-3-carboxylic acid
7-fluoro-2-methyl-4-(3-phenylpiperazine-1-carbonyl)quinoline
2-methyl-6-({3-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)pyridine
3-[(4-methoxyphenyl)methyl]-1-methyl-8-({4-[methyl(phenyl)amino]phenyl}methyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-[5-(pyridin-4-yl)pyrazolo[1,5-a]pyrimidin-7-yl]thiomorpholine
1-({4-methyl-5-[1-(pyrimidin-2-yl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)azepane
5-{[3-(2-hydroxyethyl)-4-[(4-methoxy-3-methylphenyl)methyl]piperazin-1-yl]methyl}-2-methoxyphenol
1-[4-(1,3-benzothiazol-2-yl)piperazin-1-yl]-2-(2-methoxyphenyl)ethan-1-one
1-[4-(benzenesulfonyl)piperazin-1-yl]-4-(1H-pyrazol-4-yl)butan-1-one
N-[(3,4-difluorophenyl)methyl]-4-(1H-pyrazol-4-yl)butanamide
4-methyl-N-[(2S)-3-methylbutan-2-yl]-3-(2-oxoimidazolidin-1-yl)benzamide
N-(2-methyl-1-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}propyl)-2-(5-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)acetamide
[(3R,4R)-1-(5-chloro-2-methoxybenzoyl)-4-(morpholin-4-ylmethyl)pyrrolidin-3-yl]methanol
2-[4-(methanesulfonamidomethyl)phenyl]-N-methylbenzamide
1-{[2-(3-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-3,5-dimethyl-1H-1,2,4-triazole
{[2-(2,4-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl){[4-(trifluoromethyl)phenyl]methyl}amine
2-methyl-3-[(4-{1-methyl-octahydropyrrolo[1,2-a]piperazine-2-carbonyl}piperidin-4-yl)oxy]pyridine
3-hydroxy-3-({[(4-hydroxy-1-methylpiperidin-4-yl)methyl]amino}methyl)-1-(2-phenylethyl)piperidin-2-one
N-cyclopentyl-N'-(2-methoxyethyl)-N'-(1-methylpiperidin-4-yl)butanediamide
2-{4-[(2-phenylpyrimidin-5-yl)methyl]piperazin-1-yl}pyridine-3-carboxamide
6-chloro-3-fluoro-N-[2-(pyrrolidin-1-yl)ethyl]imidazo[1,2-a]pyridine-2-carboxamide
(3aS,6aS)-2-cyclopentanecarbonyl-5-[2-(6-methylpyridin-2-yl)ethyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-(3,4-dihydro-2H-1-benzopyran-6-ylmethyl)-1-(propan-2-yl)-1H-pyrazole-4-carboxamide