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N-{1-[1-(5-methylhex-5-en-2-yl)piperidin-4-yl]-1H-pyrazol-5-yl}-3-phenoxypropanamide
2-(2-{4-[4-(piperidin-3-yl)benzoyl]piperazin-1-yl}ethoxy)ethan-1-ol
2-[1-(propan-2-yl)piperidin-4-yl]-N-[2,2,2-trifluoro-1-(pyridin-3-yl)ethyl]acetamide
1,8-dibenzyl-3-(2-methoxyethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-8-(6-methylpyridin-2-yl)-1,8-diazaspiro[4.5]decane
2,6-dimethyl-3-[3-(4-phenyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]-1,4-dihydropyridin-4-one
1-[(3R,4R)-3-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-4-(hydroxymethyl)pyrrolidin-1-yl]-2-[methyl(phenyl)amino]ethan-1-one
5-(5-methylfuran-2-yl)-N-({2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl}methyl)-1,2,4-triazin-3-amine
N-cyclopropyl-N-{[2-(2,3-dimethoxyphenyl)-6H,7H,8H-cyclopenta[g]quinolin-3-yl]methyl}-3-(3,5-dimethyl-1H-pyrazol-1-yl)propanamide
2-(pyridin-4-yl)-N-(thiophen-3-ylmethyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
N-(1-{7-[2-(4-chlorophenoxy)acetyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-3-methylbutyl)-2-(dimethylamino)acetamide
1-(4,4-difluoropiperidin-1-yl)-2-(dimethylamino)-2-(4-methylphenyl)ethan-1-one
2-(3-{[3-(2,3-dimethoxyphenyl)pyrrolidin-1-yl]methyl}phenoxy)acetamide
3-(5-fluoro-1H-1,3-benzodiazol-2-yl)-N-[(4-{[(2-fluorophenyl)methyl]amino}-8-methylquinazolin-2-yl)methyl]propanamide
1-{2-[7-(1-benzothiophen-3-yl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]ethyl}pyrrolidin-2-one
N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-N-(oxolan-2-ylmethyl)-1,3-benzoxazole-2-carboxamide
4-(4-{[4-(trifluoromethoxy)phenyl]methyl}piperazin-1-yl)-2-[(3,4,5-trimethoxyphenyl)methyl]-2,3-dihydro-1H-isoindole-1,3-dione
7-propyl-2-(pyridin-4-yl)-2,7-diazaspiro[4.5]decan-6-one
1-[(4-methyl-1H-imidazol-5-yl)methyl]-4-[1-(2-phenylethyl)pyrrolidin-3-yl]piperidine
(4aS,8aR)-6-[5-(3-methyl-1,2,4-oxadiazol-5-yl)pyridin-2-yl]-1-propyl-decahydro-1,6-naphthyridin-2-one
1-[(1S,5R)-3-(2,3-dihydro-1H-inden-2-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-(5-methyl-1H-pyrazol-1-yl)ethan-1-one
9-hydroxy-4-oxo-N-(oxolan-2-ylmethyl)-N-(thiophen-3-ylmethyl)-4H-pyrido[1,2-a]pyrimidine-3-carboxamide
N-[(5-methylpyrazin-2-yl)methyl]-2-[3-(trifluoromethyl)phenoxymethyl]-1,3-oxazole-4-carboxamide
2-(1-methyl-1H-pyrazol-3-yl)-1-(4,5,6,7-tetrahydro-1-benzothiophene-2-carbonyl)piperidine
2-ethyl-4-{1-[(4-fluorophenyl)methyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-5-yl}-6-methylpyrimidine
5-(5-ethylfuran-2-yl)-1H,5H,6H,7H,8H-pyrido[3,2-f]indazol-7-one
N-{1-[6-amino-2-(diethylamino)pyrimidin-4-yl]pyrrolidin-3-yl}acetamide
4-[1-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)piperidin-4-yl]pyridine
1-{1-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperidin-4-yl}-N-(2-phenylethyl)piperidine-3-carboxamide
2-[4-(6,8-dimethylquinolin-4-yl)-1-(1-methylpiperidin-4-yl)piperazin-2-yl]ethan-1-ol
1-(pyridin-4-yl)-4-[4-(trimethyl-1H-pyrazol-4-yl)pyrimidin-2-yl]-1,4-diazepane
4-[1-(2-fluorophenyl)-3-(1-phenylcyclopropyl)-1H-1,2,4-triazol-5-yl]butanamide
1-methyl-9-{[2-(3-methylphenyl)pyrimidin-5-yl]methyl}-1,4,9-triazaspiro[5.5]undecan-5-one
1-(2-fluorophenyl)-4-[(3-{[1-(1,3-thiazole-5-carbonyl)piperidin-3-yl]methoxy}phenyl)methyl]piperazine
(1-methyl-1H-imidazol-2-yl)({1-[5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]piperidin-4-yl})methanol
1-(2-cyclohexylethyl)-3-hydroxy-3-{[methyl(propan-2-yl)amino]methyl}piperidin-2-one
N-(2,1,3-benzoxadiazol-5-ylmethyl)-N-methyl-3-{5-[(3-methylphenyl)methyl]-1,3,4-oxadiazol-2-yl}propanamide
2-[4-(3,3,3-trifluoro-2-methylpropyl)piperazin-1-yl]pyrazine
1-[(3S)-3-(dimethylamino)pyrrolidin-1-yl]-3-{[(4-fluorophenyl)methyl]sulfanyl}propan-1-one
N-[2-(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)ethyl]-1-[2-(piperidin-2-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
1-{[2-(2,5-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-3-(3-fluorophenoxymethyl)piperidine
N-{3-[2-(3-chlorophenyl)-1H-imidazol-1-yl]phenyl}methanesulfonamide
3-amino-N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}benzamide
2-ethyl-4-methyl-5-[2-(1H-pyrazol-4-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]-1,3-oxazole
3-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]-1-{1H-pyrrolo[2,3-b]pyridin-6-yl}piperidine
N-[(4-methyl-1,3-thiazol-2-yl)methyl]-2-(pyridin-4-yl)quinoline-4-carboxamide
1-{[3-(4-cyclohexylphenyl)-1-methyl-1H-pyrazol-4-yl]methyl}-4-(furan-2-carbonyl)-1,4-diazepane
2-(2-hydroxyphenyl)-N-[(2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)methyl]acetamide
(3aS,6aS)-5-[(2-aminopyridin-3-yl)methyl]-1-oxo-2-(prop-2-en-1-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
[(3R,4R)-1-(2-chloro-5-fluorobenzoyl)-4-(piperidin-1-ylmethyl)pyrrolidin-3-yl]methanol