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(2R,3R,6R)-3-(4-methoxyphenyl)-5-[(2-methyl-1H-imidazol-4-yl)methyl]-1,5-diazatricyclo[5.2.2.02,6]undecane
N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-5,7-dimethyl-[1,2,4]triazolo[4,3-a]pyrimidine-3-carboxamide
4-(3-{imidazo[1,2-a]pyridin-2-yl}-1,2,4-oxadiazol-5-yl)-1-(pyridin-3-ylmethyl)pyrrolidin-2-one
1-(1H-1,3-benzodiazole-5-carbonyl)-3-(3-phenylpropyl)piperidine-3-carboxylic acid
1-(2,3-dimethylphenyl)-N-[(3-methyl-1H-pyrazol-5-yl)methyl]-4,5,6,7-tetrahydro-1H-indazol-4-amine
N-(1,4-dioxan-2-ylmethyl)-3-sulfamoylbenzamide
N-[(4-methylphenyl)methyl]-4-oxo-N-(propan-2-yl)-4H-pyrido[1,2-a]pyrimidine-3-carboxamide
(1R,5R)-N,N-dimethyl-6-[(3-methylthiophen-2-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
6-methoxy-N-[1-(methoxymethyl)cyclopentyl]-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
N-[(2-methoxyphenyl)methyl]-1-methyl-N-[(3-methylphenyl)methyl]-1H-imidazole-5-carboxamide
2-(3-methyl-1H-1,2,4-triazol-5-yl)-N-{3-[(trifluoromethyl)sulfanyl]phenyl}pyrrolidine-1-carboxamide
2-({[(3-tert-butyl-1H-pyrazol-5-yl)methyl](methyl)amino}methyl)-4-hydroxyquinoline-6-carboxamide
N-[(1R,3R)-3-aminocyclopentyl]-6-(2-hydroxyethyl)pyrazolo[1,5-a]pyrimidine-2-carboxamide
1-[(3-methoxyphenyl)methyl]-4-[(3R)-1,2,3,4-tetrahydroisoquinoline-3-carbonyl]piperazin-2-one
N-{2-[(3,5-dimethyl-1H-pyrazol-4-yl)sulfanyl]phenyl}-2-(1,2,3,6-tetrahydropyridin-4-yl)acetamide
1-{1-[(4-fluoro-2-methylphenyl)methyl]piperidin-4-yl}-N-(2-methoxyethyl)piperidine-3-carboxamide
4-{3'-oxo-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-4'-yl}butanamide
1-[(1S,5R)-3-acetyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-3-(4,5,6,7-tetrahydro-1H-indazol-3-yl)propan-1-one
3-[4-(2-phenylethyl)-1H-1,2,3-triazol-1-yl]propane-1,2-diol
1-(azepan-1-yl)-2-[(3R,4R)-4-hydroxy-3-methyl-4-(oxan-4-yl)piperidin-1-yl]ethan-1-one
3-[(3R,4S)-1-(3-chloro-5-fluorobenzoyl)-4-(morpholin-4-yl)piperidin-3-yl]propanoic acid
2-{7-methyl-6-oxo-2,7-diazaspiro[4.5]decan-2-yl}pyridine-3-carboxylic acid
4-{2-[(4-fluorophenyl)methyl]-3H-imidazo[4,5-b]pyridin-3-yl}-1-(3-methylbut-2-en-1-yl)piperidine
3-(2-ethyl-1H-imidazol-1-yl)-1-{2-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-1-yl}propan-1-one
(3R,4R)-1-[(2-butyl-5-chloro-1H-imidazol-4-yl)methyl]-3-methyl-4-(oxan-4-yl)piperidin-4-ol
N-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-N-methyl-3-(1,2-oxazinan-2-yl)propanamide
(2S,4R)-4-amino-N-methyl-1-[2-(4-methylphenoxymethyl)furan-3-carbonyl]pyrrolidine-2-carboxamide
4-({[1-(2,3-dihydro-1,4-benzodioxin-6-yl)-3-ethyl-1H-1,2,4-triazol-5-yl]methyl}sulfanyl)pyridine
1-{3-[(1R,5R)-6-(cyclobutylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]-3-oxopropyl}-6-methyl-1,2-dihydropyridin-2-one
propyl 4-{4-methyl-5-[(4-methylpiperazin-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidine-1-carboxylate
(2S,4S,5R)-4-[(carboxymethyl)(methyl)carbamoyl]-1,2-dimethyl-5-(2-methylphenyl)pyrrolidine-2-carboxylic acid
(1S,5R)-3-[(2-methyl-1,3-oxazol-4-yl)methyl]-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonane
(2E)-3-(3-fluorophenyl)-N-[1-(4-methyl-5-{[(2-methylphenyl)methyl]sulfanyl}-4H-1,2,4-triazol-3-yl)ethyl]prop-2-enamide
5-[1-(cyclopentylmethyl)pyrrolidin-2-yl]-N-(1-methyl-1H-pyrazol-4-yl)thiophene-2-carboxamide
7-[6-(4-methoxyphenyl)-2-oxo-1,2-dihydropyridine-3-carbonyl]-2,7-diazaspiro[4.4]nonane-1,3-dione
2-{2-[1-(9H-purin-6-yl)piperidin-3-yl]-1H-imidazol-1-yl}acetamide
5-[(1R,5S)-3-benzyl-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-4-methylpyrimidin-2-amine
4-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl]-2-(propan-2-yl)-1,3-thiazole
2-{4-cyclobutyl-1-[(2-ethoxyphenyl)methyl]piperazin-2-yl}ethan-1-ol
2-[4-(1H-indol-3-ylmethyl)-1-(2-methylpropyl)piperazin-2-yl]ethan-1-ol
N-[2-(dimethylsulfamoyl)ethyl]-2,6-dimethylpyridine-4-carboxamide
N-[(3S,4R)-1-[(5-cyano-1-ethyl-1H-pyrrol-3-yl)methyl]-4-(5-methylfuran-2-yl)pyrrolidin-3-yl]acetamide
2-[4-(dimethyl-1,3-oxazole-4-carbonyl)piperazin-1-yl]-1,3-benzothiazole
6-[4-(2-benzyl-1,3-thiazole-4-carbonyl)piperazin-1-yl]pyridine-3-carbonitrile
(1,4-dioxan-2-ylmethyl)(methyl){[5-methyl-2-(2-methylphenyl)-1,3-oxazol-4-yl]methyl}amine
2-(morpholin-4-yl)-2-(pyridin-3-yl)-N-{[7-(pyrimidin-5-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}acetamide
ethyl 2-[1-(2-benzyl-1-methyl-5-propanamido-1H-1,3-benzodiazole-7-carbonyl)piperidin-2-yl]acetate
methyl 2-chloro-4-[({[(2S,4S)-4-fluoropyrrolidin-2-yl]methyl}carbamoyl)amino]benzoate
1-(4-chloro-3-methylphenoxy)-3-[(pyrimidin-4-yl)amino]propan-2-ol
7-(pyridin-2-ylmethyl)-1-oxa-3,7-diazaspiro[4.5]decan-2-one