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1-methyl-2-oxo-N-[2-(3-phenylpyrrolidin-1-yl)ethyl]-1,2,5,6,7,8-hexahydroquinoline-3-carboxamide
2-(4-fluorophenyl)-1-(thiophene-3-carbonyl)piperidine
2-cyclopentyl-8-(9H-purin-6-yl)-1,3,8-triazaspiro[4.5]dec-1-en-4-one
(2S,4R)-4-acetamido-N,N-diethyl-1-[(2-fluoro-4-methoxyphenyl)methyl]pyrrolidine-2-carboxamide
1-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-6-methyl-4-(trifluoromethyl)-1,2-dihydropyridin-2-one
1-methyl-4-[(5-{1-[(2-methylphenyl)methyl]-1H-1,2,3-triazol-4-yl}-1,2,4-oxadiazol-3-yl)methyl]piperidine
1-[(4-fluoro-3-methylphenyl)methyl]-4-[(2-methyl-1H-imidazol-1-yl)methyl]piperidine
2-[(2S,4S)-2-(diethylcarbamoyl)-4-(1-methyl-1H-pyrazole-5-amido)pyrrolidin-1-yl]acetic acid
(1R,5R)-N,N-dimethyl-6-(2-methyl-1H-pyrrole-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
(3-{2-[1-(4-fluoro-2-methylbenzoyl)piperidin-4-yl]-1H-imidazol-1-yl}propyl)dimethylamine
5-methyl-N4-[1-(thiophene-2-carbonyl)piperidin-3-yl]pyrimidine-2,4-diamine
4-[(4-fluorophenyl)methyl]-1-{[5-(hydroxymethyl)furan-2-yl]methyl}-3-(propan-2-yl)-1,4-diazepan-5-one
N-(4-phenylbutan-2-yl)-7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carboxamide
N-methyl-N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-1H-1,2,4-triazole-5-carboxamide
5-amino-3-[3-(4-fluorophenyl)-1H-pyrazol-4-yl]-1,6-diazatricyclo[6.2.2.02,7]dodeca-2,4,6-triene-4-carbonitrile
dimethyl({2-[3-(3-{pyrazolo[1,5-a]pyrimidin-3-yl}phenyl)-1H-pyrazol-1-yl]ethyl})amine
1-(1-{4-[(3-methylphenyl)sulfanyl]piperidin-1-yl}-1-oxopropan-2-yl)pyrrolidin-2-one
2-[ethyl({[(3R,4R)-4-(hydroxymethyl)-1-[3-(5-methylfuran-2-yl)-1H-pyrazole-5-carbonyl]pyrrolidin-3-yl]methyl})amino]ethan-1-ol
1-[3-(5-methyl-1H-pyrazol-1-yl)propyl]-4-(1H-pyrazol-1-ylmethyl)piperidine
N,N-dimethyl-3-{1-[2-(pyridin-2-yl)pyrimidine-5-carbonyl]piperidin-3-yl}propanamide
2-{[6-(1,2,3,4-tetrahydroisoquinolin-5-yl)quinazolin-4-yl]amino}ethan-1-ol
3-(1-{1-[2-(diethylamino)acetyl]piperidin-4-yl}-1H-pyrazol-5-yl)-1-(2-methylphenyl)urea
1-[2-(3-chlorophenyl)ethyl]-3-[4-(2-ethoxyphenyl)piperazine-1-carbonyl]-2-(methoxymethyl)-6-methyl-1,4-dihydropyridin-4-one
1-{[1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}pyrrolidin-3-amine
1-(3-tert-butyl-1-methyl-1H-pyrazol-5-yl)-3-(2-methyl-4,5,6,7-tetrahydro-1,3-benzothiazol-4-yl)urea
1-(1-methyl-5-{[(oxolan-2-ylmethyl)(propyl)amino]methyl}-1H-pyrrol-3-yl)ethan-1-one
1-methyl-2-oxo-3-(pentan-3-yl)-1H,2H,3H-imidazo[4,5-b]pyridine-6-carboxylic acid
(4aS,8aR)-1-[2-(1H-imidazol-4-yl)ethyl]-6-[(2E)-3-phenylprop-2-en-1-yl]-decahydro-1,6-naphthyridin-2-one
4-(1,3-dimethyl-1H-pyrazol-4-yl)-N-methyl-N-(1,2-oxazol-3-ylmethyl)pyrimidin-2-amine
methyl 2-(oxan-2-ylmethyl)-1-oxo-1,2-dihydroisoquinoline-7-carboxylate
1-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-3-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
6-tert-butyl-1-methyl-N-(2-phenoxyethyl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-[1-(1H-imidazol-1-yl)-3,3-dimethylbutan-2-yl]-5,6,7,8-tetrahydroquinoline-3-carboxamide
1-(3,5-dimethylphenyl)-4-(7-fluoroquinazolin-4-yl)piperazin-2-one
2-chloro-N-[2-(1-methylpiperidine-2-carbonyl)-1,2,3,4-tetrahydroisoquinolin-7-yl]benzamide
(3S,4S)-1-(1-cyclobutanecarbonylpiperidin-4-yl)-4-cyclopropylpyrrolidine-3-carboxylic acid
2-(2,2-dimethylpropanamido)-N-[2-(3-hydroxypiperidin-1-yl)ethyl]-5-methylthiophene-3-carboxamide
5-(2,3-difluoro-4-methoxyphenyl)-1-(thiophen-2-ylmethyl)-1H,4H-pyrazolo[3,4-d]imidazole
2-methoxy-N-(2-methoxy-5-{[(thiolan-3-yl)carbamoyl]amino}phenyl)acetamide
(3S,4S)-1-[(5-cyclohexylthiophen-2-yl)methyl]-4-(morpholin-4-yl)pyrrolidin-3-ol
4-[2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-benzyl-N-butyl-1-methyl-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
1,3,6-trimethyl-N-(2-propoxypropyl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
1-(4-ethylpiperazin-1-yl)-3-(3-{[methyl(2-methylpropyl)amino]methyl}phenoxy)propan-2-ol
N-ethyl-2-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]pyridine-4-carboxamide
methyl(pyrazin-2-ylmethyl){[5-(pyrrolidin-1-ylmethyl)thiophen-2-yl]methyl}amine
2-{1-[(3,5-dimethoxyphenyl)methyl]-4-(1,3-thiazol-2-ylmethyl)piperazin-2-yl}ethan-1-ol
methyl 6-(4-methylpentanoyl)-2-[(3-methylphenyl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
2-methoxy-3-{4-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyrazine
4-chloro-2-methoxy-N-[2-(1-methylpiperidin-3-yl)ethyl]benzamide