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3-[1-(4-fluorobenzenesulfonyl)piperidin-3-yl]-N-(4-methoxy-2-methylphenyl)propanamide
3-[(1,4-dimethylpiperazin-2-yl)methyl]-1-[2-(2-fluorophenoxy)phenyl]urea
[3-(3-methoxypropyl)-1-[2-(pyridin-2-yl)ethyl]piperidin-3-yl]methanol
2-[2-({[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}amino)pyrimidin-4-yl]pyridine-4-carboxylic acid
N-[(3S,4R)-1-{[2-(furan-2-yl)pyrimidin-5-yl]methyl}-4-(5-methylfuran-2-yl)pyrrolidin-3-yl]acetamide
({3-[(2-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)[2-(morpholin-4-yl)ethyl]amine
1-methyl-4-(1-{1-[4-(pyrrolidine-1-carbonyl)pyridin-2-yl]piperidin-4-yl}ethyl)piperazine
N-[5-oxo-1-(3-phenylpropyl)pyrrolidin-3-yl]isoquinoline-5-carboxamide
1-(3-chlorophenyl)-4-[2-methyl-2-(4-methylphenoxy)propanoyl]piperazin-2-one
N-{1-[5-(trifluoromethyl)pyridin-2-yl]piperidin-3-yl}quinoxaline-5-carboxamide
1-(2-aminoethyl)-N-[(1-benzyl-1H-imidazol-2-yl)methyl]-N-methyl-1H-1,2,3-triazole-4-carboxamide
2-{[5-(4-fluorophenyl)pyrazolo[1,5-a]pyrimidin-7-yl]amino}-N,N-dimethylethane-1-sulfonamide
2-butoxy-N-{1-[5-methyl-1-(2-methylphenyl)-1H-pyrazol-4-yl]ethyl}acetamide
5-(4-chloro-2-methylbenzoyl)-1-[(4-fluorophenyl)methyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazole
N,3,6-trimethyl-N-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-[1,2]oxazolo[5,4-d]pyrimidin-4-amine
2-(1H-pyrazol-1-yl)-N-{[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)pyridin-3-yl]methyl}propanamide
1-[(4-fluorophenyl)methyl]-N-[(2-phenylphenyl)methyl]-1H-1,2,3-triazole-4-carboxamide
1,1-dioxo-N-(2,3,4,9-tetrahydro-1H-carbazol-6-ylmethyl)-1λ6-thiane-4-carboxamide
1-[(2R,3R,6R)-3-(2,3-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]pentane-1,4-dione
3-hydroxy-1-(3-phenylpropyl)-3-{[(thiophen-2-ylmethyl)amino]methyl}piperidin-2-one
methyl (2S)-2-{2-[(3-ethyl-1H-1,2,4-triazol-5-yl)sulfanyl]acetamido}-3-(4-hydroxyphenyl)propanoate
2-(adamantan-1-yl)-N-[3-(dimethylamino)butyl]-4-hydroxypyrimidine-5-carboxamide
3-{ethyl[3-(2-methoxyphenoxy)propyl]amino}-1λ6-thiolane-1,1-dione
1-(3-{[3-(methoxymethyl)pyrrolidin-1-yl]sulfonyl}benzoyl)-1,4-diazepane
2-({6-chloroimidazo[2,1-b][1,3]thiazol-5-yl}sulfonyl)-7-methyl-2,7-diazaspiro[4.5]decan-6-one
2-{5-[(2S,4R)-4-hydroxypyrrolidin-2-yl]-3-(1-phenylcyclopropyl)-1H-1,2,4-triazol-1-yl}acetic acid
1,4-dimethyl-9-{[1-(2-methylpropyl)-1H-1,3-benzodiazol-2-yl]methyl}-1,4,9-triazaspiro[5.5]undecane
1-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]-3-(3-methylphenoxymethyl)piperidine
3-[5-(2,6-difluoro-4-methoxyphenyl)-3-methyl-1H-1,2,4-triazol-1-yl]-1λ6-thiolane-1,1-dione
4-hydroxy-1-methyl-N-[2-(4-phenylpiperidin-1-yl)ethyl]piperidine-4-carboxamide
1'-[2-(3-chloro-4-hydroxyphenyl)acetyl]-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
3-benzoyl-1-(4-methyl-1,3-thiazol-2-yl)piperidine
ethyl 4-(2-methoxyethyl)piperidine-4-carboxylate
dimethyl[(5-{[4-(pyridin-3-ylmethyl)-1,4-diazepan-1-yl]methyl}thiophen-3-yl)methyl]amine
3-[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]-N-[3-(pyridin-3-yloxy)propyl]propanamide
(cyclohex-3-en-1-ylmethyl)({2-[4-(pyridin-2-yl)piperazin-1-yl]pyridin-3-yl}methyl)amine
6-{2-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidine-1-carbonyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
(3S,4R)-N,N-dimethyl-1-{2-methylimidazo[1,2-a]pyrimidine-3-carbonyl}-4-(4-methylphenyl)pyrrolidin-3-amine
1-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]-N-(piperidin-4-yl)piperidine-3-carboxamide
N-(1H-indazol-5-yl)-4-methoxy-4-phenylpiperidine-1-carboxamide
N-(2,6-dimethylpyridin-3-yl)-4-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carboxamide
N-[3-(4-chloro-3-methylphenoxy)-2-hydroxypropyl]-5-propyl-1,2-oxazole-3-carboxamide
N1,N1-dimethyl-N3-(2-{[(2-methylphenyl)methyl]sulfanyl}ethyl)piperidine-1,3-dicarboxamide
2-ethoxy-5-(2-{[(1-methyl-1H-imidazol-2-yl)methyl]amino}pyrimidin-4-yl)benzoic acid
2-ethyl-9-{2-[methyl(pyridin-3-ylmethyl)amino]acetyl}-2,9-diazaspiro[5.5]undecan-3-one
1-(cyclopentylmethyl)-4-[(2-phenyl-1H-imidazol-4-yl)methyl]piperazine
3-[(3S,4S)-3-hydroxy-4-(naphthalen-2-yl)piperidine-1-carbonyl]-6-methyl-1,2-dihydropyridin-2-one
N-{[2-(dimethylamino)pyridin-3-yl]methyl}-2-(5-ethyl-1-benzofuran-3-yl)acetamide
2,5-dimethyl-N-[2-(thiophen-2-yl)ethyl]-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
N-[(3R,5S)-1-[(2E)-but-2-en-1-yl]-5-[(propan-2-yl)carbamoyl]pyrrolidin-3-yl]-2,4-dimethylpyrimidine-5-carboxamide