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2-(4-oxo-3,4-dihydroquinazolin-3-yl)-N-[2-(3-phenyl-1,2,4-oxadiazol-5-yl)ethyl]acetamide
2-[(1S,4R)-2-azabicyclo[2.2.1]heptan-2-yl]-1-{2-benzyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl}ethan-1-one
1-benzyl-5-[2-(dimethyl-1,2-oxazol-4-yl)ethyl]-3-(oxolan-3-yl)-1H-1,2,4-triazole
2-(4-{5-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl}piperazin-1-yl)-1,3-benzothiazole
N-{[2-(3-hydroxypiperidin-1-yl)pyridin-3-yl]methyl}-2-(phenylsulfanyl)acetamide
2-[4-(dimethylamino)-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]-4-methylphenol
4-{[3-(3-fluoro-4-methoxyphenyl)-1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}-1,4-oxazepane
[3-(cyclopropylmethyl)-1-[3-(dimethylamino)pyrazin-2-yl]piperidin-3-yl]methanol
(butan-2-yl)({[4-(1H-imidazol-1-yl)phenyl]methyl})(pyridin-3-ylmethyl)amine
7-[(2,3-difluorophenyl)methyl]-2-(oxane-4-carbonyl)-2,7-diazaspiro[4.5]decane
3-(4-methylphenyl)-1-[(1S,5R)-3-(pyridin-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]propan-1-one
4-(3-tert-butyl-1H-pyrazol-1-yl)-1-(3-methylpyrazin-2-yl)piperidine-4-carboxylic acid
1-[(1S,5R)-3-[(dimethyl-1,2-oxazol-4-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]-3-(thiophen-3-yl)propan-1-one
(3R,5S)-N-[3-(dimethylamino)propyl]-5-(3-fluorophenoxymethyl)-1-(pyridin-4-ylmethyl)piperidine-3-carboxamide
3-[(3R,4S)-1-[3-(hydroxymethyl)quinolin-2-yl]-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propan-1-ol
4-(hydroxymethyl)-5-methyl-N-{2-[4-(propan-2-yl)-1,3-thiazol-2-yl]ethyl}-1,2-oxazole-3-carboxamide
N-[(4-ethoxyphenyl)methyl]-N-ethyl-3,5-dimethyl-1H-indole-2-carboxamide
4-phenyl-2-[(3-propyl-1,2,4-oxadiazol-5-yl)methyl]-1,2-dihydrophthalazin-1-one
1-(oxolan-2-ylmethyl)-N-[2-(1-phenyl-1H-pyrazol-4-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
[1-(1-{[4-(methylsulfanyl)phenyl]methyl}piperidin-3-yl)piperidin-4-yl]methanol
2,5-dimethyl-4-(4-{[3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}piperazin-1-yl)pyrimidine
methyl 1-benzyl-5-{[(2-methoxyphenyl)methyl]amino}-3-(pyridine-3-amido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
N-(2-hydroxyethyl)-1,3-dimethyl-N-(thiophen-2-ylmethyl)-1H-indole-2-carboxamide
N-[2-(azepan-1-yl)ethyl]-N-ethyl-3-propanamidobenzamide
1-ethyl-4-{[(1-methylpiperidin-4-yl)(pyridin-3-ylmethyl)amino]methyl}-1H-pyrrole-2-carbonitrile
2-{3-oxo-1-[(3-phenoxyphenyl)methyl]piperazin-2-yl}-N-[2-(pyridin-4-yl)ethyl]acetamide
[(3R,4R)-4-[(4-methylpiperazin-1-yl)methyl]-1-(quinoline-6-carbonyl)pyrrolidin-3-yl]methanol
5-{4-[(3-fluorophenyl)methyl]piperazine-1-carbonyl}-N-methyl-1-(3-methylbutyl)-4-oxo-1,4-dihydropyridine-3-carboxamide
3,5-dimethyl-1-{1-[(3-phenyloxolan-3-yl)methyl]azetidin-3-yl}-1H-pyrazole
3,3,3-trifluoro-N-({1-[(3-fluoro-4-methylphenyl)methyl]pyrrolidin-3-yl}methyl)propanamide
3-{[3-(3-hydroxypropyl)piperidin-1-yl]methyl}-6-methoxy-1,2-dihydroquinolin-2-one
1-{4-[4-(3-methoxyphenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}cyclopropane-1-carboxamide
[(3R,4R)-4-{[(2-methoxyethyl)(methyl)amino]methyl}-1-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]pyrrolidin-3-yl]methanol
N-(butan-2-yl)-N-(pyridin-3-ylmethyl)-2,3-dihydro-1,4-benzodioxine-5-carboxamide
[(3R,4R)-4-({[2-(dimethylamino)ethyl](methyl)amino}methyl)-1-[(2,4,5-trifluorophenyl)methyl]pyrrolidin-3-yl]methanol
ethyl 2-{3'-oxo-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-1-yl}pentanoate
methyl 6-[(2E)-3-(3-chlorophenyl)prop-2-enoyl]-2-[(prop-2-en-1-yl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
ethyl 1-(5-{[2-(propan-2-yl)-1H-imidazol-1-yl]methyl}-1H-pyrazole-3-carbonyl)piperidine-3-carboxylate
N-methyl-5-(3-methyl-1,2,4-oxadiazol-5-yl)-N-(thiophen-3-ylmethyl)pyridin-2-amine
2,3-dimethyl-N-{2-[3-({methyl[(1-methyl-1H-pyrazol-4-yl)methyl]amino}methyl)phenoxy]propyl}-1H-indole-7-carboxamide
2-[2-(azepan-1-ylmethyl)phenyl]-6-cyclopropyl-3,4-dihydropyrimidin-4-one
6-chloro-4-(1,2,3,4-tetrahydroisoquinolin-5-yl)quinoline
N-cyclopropyl-5-(5-ethylpyrimidin-2-yl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
3-{[(4-fluorophenyl)methyl]sulfanyl}-N-[3-(oxolan-3-yl)propyl]propanamide
3-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-1-(4-methyl-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-6-yl)urea
2-(5-acetylthiophen-3-yl)-N-[(4-chlorophenyl)methyl]acetamide
4-benzyl-3-ethyl-1-[4-(hydroxymethyl)-5-methyl-1,2-oxazole-3-carbonyl]-1,4-diazepan-5-one
1-{[2-(3-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-3-methylpiperazine
N-(2-fluorophenyl)-3-[(oxan-4-yl)sulfamoyl]benzamide
2-(3-cyano-2-methyl-1H-indol-1-yl)-N-[(1-ethyl-1H-pyrazol-4-yl)methyl]acetamide