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8-fluoro-2-({[3-(furan-2-yl)propyl]amino}methyl)quinolin-4-ol
N-[(2-chlorophenyl)methyl]-3-{1-[(3-methylpyridin-4-yl)methyl]piperidin-3-yl}propanamide
N-({4-[(3-fluorophenyl)methoxy]phenyl}methyl)-N-(oxolan-2-ylmethyl)pyridine-4-carboxamide
3-(cyclopropylmethyl)-1-[2-(2-oxopyrrolidin-1-yl)ethyl]piperidine-3-carboxylic acid
N-(6-ethylpyridin-2-yl)-5-{1-[(3-methyl-1H-pyrazol-5-yl)methyl]pyrrolidin-2-yl}thiophene-2-carboxamide
(3aR,6aR)-N-[(8-methoxyquinolin-5-yl)methyl]-N,2-dimethyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
2-{1-[(3,4-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-methylacetamide
N-[(3S,4R)-1-(dimethyl-1,3-thiazole-5-carbonyl)-4-(4-methylphenyl)pyrrolidin-3-yl]cyclopropanecarboxamide
{[2-(cyclopentanesulfonyl)-1-(3-methoxypropyl)-1H-imidazol-5-yl]methyl}(methyl)(2-phenoxyethyl)amine
2-[({5-cyclobutanecarbonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)amino]pyridine-3-carbonitrile
1-(4-benzyl-6-hydroxy-1,4-diazepan-1-yl)-2-(pyridin-2-ylsulfanyl)ethan-1-one
6-methoxy-N-methyl-N-[3-(1-methyl-1H-imidazol-2-yl)propyl]pyrimidin-4-amine
(5-fluoro-7-{4-[2-(pyrrolidin-1-yl)ethoxy]phenyl}-2,3-dihydro-1-benzofuran-2-yl)methanamine
(2S,4S)-4-(4-{[(2-methoxyphenyl)formamido]methyl}-1H-1,2,3-triazol-1-yl)-N-methylpyrrolidine-2-carboxamide
{[5-chloro-1-methyl-3-(5-methyl-1,2-oxazol-3-yl)-1H-pyrazol-4-yl]methyl}(methyl)[(2-methyl-1,3-thiazol-4-yl)methyl]amine
N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-N-(propan-2-yl)-6-(4H-1,2,4-triazol-4-yl)pyridine-3-carboxamide
(3aR,6aR)-2-benzyl-N-[2-(pyridin-4-yl)ethyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
7-(cyclobutylmethyl)-2-(3-phenyl-1,2-oxazole-5-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
2-[2-({3-phenyl-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl}methyl)-1H-pyrrol-1-yl]-1,3-thiazole
2-(2-fluorophenyl)-N-[2-(pyrrolidine-1-sulfonyl)-1,2,3,4-tetrahydroisoquinolin-7-yl]acetamide
2-({[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}amino)-1-(1-methyl-1H-imidazol-2-yl)ethan-1-ol
(3S,5S)-1-[3-(2H-1,3-benzodioxol-5-yl)propanoyl]-5-(cyclopropylcarbamoyl)piperidine-3-carboxylic acid
N-[3-(5-amino-1,3,4-thiadiazol-2-yl)propyl]-1-cyclohexylpiperidine-3-carboxamide
(3R,5S)-N-butyl-5-[(pyridin-3-yloxy)methyl]-1-(pyridin-4-ylmethyl)piperidine-3-carboxamide
N-[2-(6-hydroxypyrimidin-4-yl)ethyl]-5,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
4-cyclobutaneamido-N-methyl-N-(3-phenylpropyl)benzamide
(3aS,6aR)-5-(1-benzofuran-2-carbonyl)-3-(pyridin-2-ylmethyl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
methyl (2S,4S,5R)-2-ethyl-5-(4-fluorophenyl)-4-[(3-hydroxy-2,2-dimethylpropyl)carbamoyl]-1-methylpyrrolidine-2-carboxylate
[1-(dimethyl-1,3-thiazol-4-yl)ethyl]({[2-(7-methoxy-2H-1,3-benzodioxol-5-yl)-5-methyl-1,3-oxazol-4-yl]methyl})methylamine
N-[(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)methyl]-2-oxo-1-phenylpyrrolidine-3-carboxamide
N-{[1-tert-butyl-3-(4-chlorophenyl)-1H-1,2,4-triazol-5-yl]methyl}acetamide
7-{[3-(4-chlorophenoxy)phenyl]methyl}-3-methyl-1-oxa-3,7-diazaspiro[4.5]decan-2-one
N-({1-[2-(2-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-N-methyl-3-(1H-1,2,3,4-tetrazol-1-yl)propanamide
N-(1-methyl-1H-indazol-3-yl)-2-[5-(pyridin-3-yl)-1H-indazol-1-yl]acetamide
ethyl 1-{[3-benzamido-2-(methoxycarbonyl)thieno[2,3-b]pyridin-6-yl]methyl}piperidine-4-carboxylate
1-ethyl-4-[(2-phenyl-1H-imidazol-4-yl)methyl]piperazine
N-[2-(5-amino-1,3,4-thiadiazol-2-yl)ethyl]-1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
3-(1,5-dimethyl-1H-pyrazol-4-yl)-7-thia-2,4,5-triazatricyclo[6.4.0.02,6]dodeca-1(12),3,5,8,10-pentaene
3-{[4-(1-hydroxypropyl)piperidin-1-yl]methyl}-N,8-dimethyl-N-(2-phenylethyl)imidazo[1,2-a]pyridine-2-carboxamide
ethyl 1-{[4-(ethoxycarbonyl)-1-(1-methyl-2-oxo-1,2-dihydroquinolin-4-yl)-1H-pyrazol-5-yl]methyl}piperidine-3-carboxylate
1-{[3-(trifluoromethoxy)phenyl]methyl}imidazolidin-2-one
(1R,5R)-N,N-dimethyl-6-[3-(pyridin-4-yl)propanoyl]-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
4-[(1E)-1-(5-chloro-2-hydroxyphenyl)prop-1-en-2-yl]-7-hydroxy-6-methoxy-1,2,3,4-tetrahydroquinolin-2-one
1-[2-(cyclopent-2-en-1-yl)acetyl]-4-(4-methylphenoxy)piperidine-4-carboxylic acid
N-ethyl-3-(5-phenyl-1,3,4-oxadiazol-2-yl)-N-[2-(1H-pyrazol-1-yl)ethyl]propanamide
3-(4-methoxy-3,5-dimethylbenzoyl)-1-(1H-pyrazol-3-ylmethyl)piperidine
5-methyl-3-[4-(1,3,4-oxadiazol-2-yl)phenyl]-1H-indole
5-acetyl-6-methyl-3-[4-(3-methylpyridin-4-yl)-1,4-diazepane-1-carbonyl]-1,2-dihydropyridin-2-one
N-(butan-2-yl)-2-(methylamino)-N-(thiophen-3-ylmethyl)pyridine-3-carboxamide
2-(4-{[2-(3,4-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazin-1-yl)pyrazine