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2-(1-benzyl-3-oxopiperazin-2-yl)-N-{[5-methyl-2-(thiophen-2-yl)-1,3-oxazol-4-yl]methyl}acetamide
2-{2-[(E)-2-phenylethenyl]phenoxy}propanamide
N-[1-(furan-2-yl)ethyl]-1-(methoxymethyl)cyclobutane-1-carboxamide
N-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N-methyl-2-oxo-1,2,5,6,7,8-hexahydroquinoline-3-carboxamide
2-[(4-{[1-(pyridine-3-carbonyl)piperidin-3-yl]methoxy}phenyl)methyl]-1,2,3,4-tetrahydroisoquinoline
N-[(2R,3R)-1'-[(2E)-3-(furan-2-yl)-2-methylprop-2-en-1-yl]-2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-phenoxyacetamide
4-[4-ethyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-methylpiperidine
3-cyclopropyl-5-(2-methoxyethyl)-1-[4-(trifluoromethyl)phenyl]-1H-1,2,4-triazole
5-methyl-3-[1-(pyrazin-2-yl)propan-2-yl]-3,4-dihydroquinazolin-4-one
1'-[3-(4,5-dimethyl-1H-pyrazol-3-yl)propanoyl]-1,2-dihydrospiro[indole-3,3'-piperidine]-2-one
1-{[4-(hydroxymethyl)oxan-4-yl]methyl}-1-methyl-3-[2-methyl-5-(4H-1,2,4-triazol-4-yl)phenyl]urea
N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl}-N-(oxolan-2-ylmethyl)butanamide
4-({3-ethoxy-4-[(3-methylbut-2-en-1-yl)oxy]phenyl}methyl)-1,4-oxazepan-6-ol
2-(1,3-benzoxazol-2-yl)-N-[(1,3-dimethyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)methyl]acetamide
N-[cyclopropyl(1-methyl-1H-1,2,4-triazol-5-yl)methyl]-6-ethyl-2-methylquinoline-4-carboxamide
2-[(1-acetylpiperidin-4-yl)oxy]-5-methoxy-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}benzamide
4-(2-{1-[5-(1H-pyrazol-1-ylmethyl)furan-2-carbonyl]piperidin-2-yl}ethyl)phenol
8-[(2E)-3-(furan-2-yl)-2-methylprop-2-en-1-yl]-1-methyl-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-[2-(1-methylpiperidin-2-yl)ethyl]-1,2-dihydroquinolin-2-one
(2S,4S)-N-ethyl-1-(thiophen-2-ylmethyl)-4-(thiophene-3-amido)pyrrolidine-2-carboxamide
N,N-diethyl-1-{[1-(4-methoxybenzoyl)piperidin-3-yl]methyl}-1H-1,2,3-triazole-4-carboxamide
N-(4-methoxy-2-methylphenyl)-3-{1-[2-(methylsulfanyl)acetyl]piperidin-3-yl}propanamide
5-methoxy-1-methyl-2-[4-(1H-1,2,4-triazole-3-carbonyl)piperazine-1-carbonyl]-1H-indole
N2-[1-(1-ethyl-1H-1,2,4-triazol-5-yl)ethyl]-N4,N4,5-trimethylpyrimidine-2,4-diamine
4-methyl-2-(2-{2-methyl-4-oxo-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl}-2-oxoethyl)-1,2-dihydrophthalazin-1-one
1-(3-acetamidopropanoyl)-3-(3-methoxypropyl)piperidine-3-carboxylic acid
N-({1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}methyl)-2-(trimethyl-1H-pyrazol-1-yl)acetamide
(5S,9aS,9bS)-5-(2,1,3-benzoxadiazol-4-yl)-2-(pyridin-3-ylmethyl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
N-methyl-4-[4-(1,2,3,4-tetrahydroisoquinolin-2-yl)piperidine-1-carbonyl]-1,3-thiazol-2-amine
(2S)-2-amino-1-(4-{[4-(4-methylphenyl)-1H-1,2,3-triazol-1-yl]methyl}piperidin-1-yl)butan-1-one
(3R,4R)-1-(3,4-dihydro-2H-1-benzopyran-6-carbonyl)-4-methyl-3-(propan-2-yl)pyrrolidin-3-ol
2-(1H-indazol-3-yl)-N-{[1-(2-methylpropyl)pyrrolidin-3-yl]methyl}acetamide
1-[(3-methylphenyl)methyl]-4-{[2-(pyrrolidin-1-yl)pyrimidin-5-yl]methyl}piperazin-2-one
4-{1-[1-(1-methyl-5-phenyl-1H-pyrazole-3-carbonyl)piperidin-4-yl]ethyl}morpholine
methyl({4-methyl-5-[(2-phenoxyethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)[(5-methylfuran-2-yl)methyl]amine
1-{4-[(furan-2-ylmethyl)sulfanyl]phenyl}-3-{2-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}urea
N-{[2-(azocan-1-yl)pyridin-3-yl]methyl}-5-hydroxy-4-oxo-4H-pyran-2-carboxamide
2-[(3-ethyl-1H-1,2,4-triazol-5-yl)sulfanyl]-N-{2-[3-(pyridin-3-yl)-1H-1,2,4-triazol-5-yl]ethyl}acetamide
1-{1-[5-(2-fluorophenyl)-1,2,4-triazin-3-yl]-4-phenylpiperidin-4-yl}ethan-1-one
1-[2-(4-methylpentyl)morpholin-4-yl]but-3-en-1-one
N-(butan-2-yl)-2-[3-(furan-2-yl)-1-(2-methoxyphenyl)-5-oxo-4,5-dihydro-1H-1,2,4-triazol-4-yl]acetamide
1-{3-[3-(2H-1,3-benzodioxol-5-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]butyl}-1H-pyrazole
N-cyclohexyl-3-[2-methyl-4-(4-methylphenyl)-5-oxopiperazin-1-yl]propanamide
N-cyclohexyl-N-ethyl-2-[4-(1H-1,2,4-triazole-5-carbonyl)morpholin-3-yl]acetamide
(3S,4S)-3-hydroxy-4-(piperidin-1-yl)-N-(2,4,6-triethylphenyl)pyrrolidine-1-carboxamide
2-[1-(1-benzothiophene-5-carbonyl)pyrrolidin-2-yl]-6-chloro-1H-1,3-benzodiazole
(3S,4R)-4-(3-fluorophenyl)-1-(4-methoxy-2-methylbenzoyl)pyrrolidine-3-carboxylic acid
2-({[(3R,4R)-4-(hydroxymethyl)-1-[2-methyl-5-(propan-2-yl)furan-3-carbonyl]pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
N-[3-(1H-imidazol-2-yl)propyl]-2,3,4,5-tetrahydro-1-benzoxepine-4-carboxamide
methyl 3-[(3-ethyl-1,2-oxazol-5-yl)methyl]-1-(2-methoxyethyl)-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxylate