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1,9-dimethyl-4-[(2E)-3-phenylprop-2-en-1-yl]-1,4,9-triazaspiro[5.6]dodecan-10-one
N-{2-[5-(oxolan-3-yl)-4-phenyl-1H-imidazol-1-yl]ethyl}aniline
9-(cyclopropylmethyl)-4-[(3-hydroxyphenyl)methyl]-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
4-{1-[1-(3-chlorobenzoyl)piperidin-4-yl]piperidine-4-carbonyl}morpholine
methyl 1-methoxy-8-{2-[4-(methylsulfanyl)phenyl]acetyl}-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylate
2-[2-(1-{[3-(2H-1,3-benzodioxol-5-yl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-2-yl)ethyl]pyridine
1-(3-fluorophenyl)-3-{1-[1-(2-methylfuran-3-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}urea
2-(2,4-difluorophenyl)-2-[(2-methyl-1-benzofuran-5-yl)formamido]acetic acid
2-(5-{1-[(2R,6S)-2,6-dimethylmorpholin-4-yl]ethyl}-1-(4-fluorophenyl)-1H-1,2,4-triazol-3-yl)acetamide
(5S,9aS,9bS)-2-(2-methoxyphenyl)-5-[3-(methylsulfanyl)phenyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
(2S)-N-(3-cyano-4-methoxyphenyl)-2-(methoxymethyl)pyrrolidine-1-carboxamide
1-(2-{4-[(2-ethoxyphenyl)methyl]piperazin-1-yl}ethyl)-N-(propan-2-yl)-1H-1,2,3-triazole-4-carboxamide
1-(ethanesulfonyl)-4-(2,3,5,6-tetramethylbenzoyl)piperazine
2-(5-chloro-2-ethoxyphenyl)-5-(piperidine-1-carbonyl)pyridine
1-(4-chlorobenzenesulfonyl)-4-[2-(propan-2-yl)-3H-imidazo[4,5-b]pyridin-3-yl]piperidine
1-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]-3-[3-(trifluoromethyl)benzoyl]piperidine
1-methyl-N-{2-[(pyridin-2-ylmethyl)carbamoyl]phenyl}piperidine-3-carboxamide
(4aR,7aS)-1-cyclobutanecarbonyl-4-[(2-fluorophenyl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-(1-phenylethyl)-4-{4-[(pyridin-3-ylmethyl)amino]piperidin-1-yl}benzamide
N-[(2-methylphenyl)(pyridin-4-yl)methyl]-3-propyl-1H-pyrazole-5-carboxamide
3-chloro-6-methyl-N-[3-(2-oxopyrrolidin-1-yl)propyl]pyrazolo[1,5-a]pyrimidine-2-carboxamide
4-{1-[3-(4-methylphenyl)phenyl]piperidin-4-yl}-1,4-diazepan-2-one
3-(azocane-1-sulfonyl)-N-(oxolan-3-yl)benzamide
2-[2-fluoro-4-(pyrrolidin-1-ylmethyl)phenoxy]-5-(piperidine-1-carbonyl)pyridine
1-[(3-methylquinoxalin-2-yl)methyl]-N-[4-(1H-pyrazol-1-yl)phenyl]piperidine-4-carboxamide
3-(2,6-difluorophenyl)-1-(1-methoxypropan-2-yl)-1-{[4-(methylsulfanyl)phenyl]methyl}urea
3-({3-[2-(3,4-difluorophenyl)ethyl]piperidin-1-yl}sulfonyl)pyridine
[1-(furan-3-carbonyl)-3-(2-phenoxyethyl)piperidin-3-yl]methanol
3-(2-amino-1,3-thiazol-4-yl)-1-{4-[(2-methylphenyl)sulfanyl]piperidin-1-yl}propan-1-one
2-cyclopropanecarbonyl-8-(3,6-dimethylpyrazin-2-yl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
2-({3-azaspiro[5.5]undecan-9-yl}amino)-N-ethylpropanamide
1-cyclopentanecarbonyl-4-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine
5-({1-[(4-methoxypiperidin-1-yl)sulfonyl]pyrrolidin-3-yl}methyl)-1,2-dihydropyridin-2-one
3-(3-methoxyquinoxalin-2-yl)-N-[(6-oxo-1,6-dihydropyrimidin-4-yl)methyl]propanamide
9-{[5-(3-fluorophenyl)-1,3,4-oxadiazol-2-yl]methyl}-2-methyl-2,9-diazaspiro[5.5]undecan-3-one
methyl 6-(cyclohex-3-ene-1-carbonyl)-2-{[(3-fluorophenyl)methyl]sulfamoyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
3-(3-hydroxy-3-methylbutyl)-N-methyl-N-{[3-(methylsulfanyl)phenyl]methyl}benzamide
9-(2-methoxyethyl)-1-methyl-4-{[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-1,4,9-triazaspiro[5.6]dodecan-10-one
N-(cyclopropylmethyl)-3-{[(3-ethyl-1,2-oxazol-5-yl)methyl](methyl)sulfamoyl}benzamide
5-propyl-N-({5-propyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)pyrimidin-4-amine
7-[2-(7-fluoro-2-methyl-1H-indol-3-yl)acetyl]-2,7-diazaspiro[4.4]nonane-1,3-dione
1-{2-[1-(pyridin-4-yl)piperidin-4-yl]ethyl}pyrrolidin-2-one
7-(2-methyl-1,3-benzothiazole-5-carbonyl)-2,7-diazaspiro[4.4]nonane-1,3-dione
4-({[(2-methyl-1,3-thiazol-4-yl)methyl]carbamoyl}amino)-N-(oxolan-2-ylmethyl)benzamide
2-[ethyl({[(3R,4R)-1-(5-ethyl-2,6-dimethylpyrimidin-4-yl)-4-(hydroxymethyl)pyrrolidin-3-yl]methyl})amino]ethan-1-ol
7-[2-(methylsulfanyl)pyrimidin-4-yl]-2-oxa-7-azaspiro[4.5]decane
(4S)-3-[(1-cyclopropyl-1H-imidazol-2-yl)methyl]-4-(propan-2-yl)-1,3-oxazolidin-2-one
5-[({1-[(2-chloro-6-fluorophenyl)methyl]-1H-1,2,4-triazol-5-yl}methyl)sulfanyl]-1,3,4-thiadiazol-2-amine
1-(4-{5-[(dimethylamino)methyl]-4-ethyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-2-(2-methyl-1,3-thiazol-4-yl)ethan-1-one
N-methyl-N-[(3-phenyl-1H-pyrazol-5-yl)methyl]-3-(1H-pyrazol-1-ylmethyl)benzamide