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2-methoxy-1-(3-{4-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]piperidine-1-carbonyl}piperidin-1-yl)ethan-1-one
methyl 4-[5-({2-[2-(pyridin-2-yl)ethyl]piperidin-1-yl}methyl)-1,2,4-oxadiazol-3-yl]benzoate
1-[9-(but-3-yn-1-yloxy)-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(4-fluorophenyl)ethan-1-one
N-[(4,6-dimethylpyridin-2-yl)methyl]-N-methyl-2-(phenylamino)pyrimidine-5-carboxamide
4-[(3,3-diphenylpiperidin-1-yl)sulfonyl]morpholine
(1R,2R,6S,7S)-N-[2-(benzyloxy)phenyl]-10-oxa-4-azatricyclo[5.2.1.02,6]decane-4-carboxamide
1-(3-methoxypropyl)-3-(naphthalen-2-ylmethyl)-8-(propan-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
3,3-dimethyl-1-[(3S,4R)-4-(propan-2-yl)-1-(2-{5H,6H,7H-[1,3]thiazolo[3,2-a]pyrimidin-3-yl}acetyl)pyrrolidin-3-yl]urea
2-[4-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)phenyl]-N-[2-(pyridin-2-yl)ethyl]acetamide
3-phenyl-N-(4-{4-[4-(pyrimidin-2-yl)-1,4-diazepan-1-yl]piperidin-1-yl}phenyl)propanamide
3-[(3R,4S)-4-(dimethylamino)-1-(3-methoxybenzenesulfonyl)piperidin-3-yl]propanoic acid
(2S,4S,5R)-2-ethyl-4-[(2-methoxy-2-methylpropyl)carbamoyl]-5-(4-methoxyphenyl)-1-methylpyrrolidine-2-carboxylic acid
(4aR,8aR)-2-[(3,5-difluorophenyl)methyl]-7-(pyrrolidine-1-carbonyl)-decahydro-2,7-naphthyridin-4a-ol
2-(2,5-dioxoimidazolidin-4-yl)-N-[2-(4-phenyl-1,3-thiazol-2-yl)ethyl]acetamide
2-{3-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}phenol
4-(4-chlorophenoxy)-1-(pyrrolidin-3-ylmethyl)piperidine
N-[4-(1H-1,2,3,4-tetrazol-5-yloxy)phenyl]-1,4-dithiepan-6-amine
5-propyl-N-[1-(pyridin-2-ylmethyl)piperidin-4-yl]-1,2-oxazole-3-carboxamide
2-(2,5-dioxoimidazolidin-1-yl)-N-[3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)propyl]acetamide
2-butyl-1-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}-2,5-dihydro-1H-pyrrole
2-cyano-N-methyl-N-[(4-phenoxyphenyl)methyl]benzamide
5-methyl-4-(3,4,5-trimethoxyphenyl)thieno[2,3-d]pyrimidine
N-[(5-cyclopropyl-1H-pyrazol-3-yl)methyl]-N-methyl-4-[5-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]butanamide
3-benzyl-8-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-1-methyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-{5-[({imidazo[1,2-a]pyridin-3-ylmethyl}amino)methyl]-2-methoxyphenoxy}-3-[methyl(propan-2-yl)amino]propan-2-ol
1-(cyclobutylmethyl)-4-(pyrazin-2-yl)-1,4-diazepane-6-carboxylic acid
(3S,4R)-4-(2H-1,3-benzodioxol-5-yl)-1-(5-methylthiophene-2-carbonyl)pyrrolidine-3-carboxylic acid
5-({3-[(3-methoxyphenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)pyrrolidin-2-one
1-[(4-acetamidophenyl)methyl]-N-[4-(1H-pyrazol-5-yl)phenyl]piperidine-3-carboxamide
3-{[1-(3-fluoro-4-methylbenzoyl)piperidin-4-yl]methyl}benzoic acid
N-[4-(furan-2-yl)phenyl]-1-[3-(2-oxoazepan-1-yl)propanoyl]piperidine-3-carboxamide
2-[({2-[(6-methylpyridin-3-yl)oxy]pyridin-3-yl}methyl)amino]pyridine-4-carboxamide
4-{2-chloro-4-[3-(methoxymethyl)pyrrolidine-1-carbonyl]phenoxy}-1-methanesulfonylpiperidine
5-methyl-1'-[1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
dimethyl[(4-methyl-5-{1-[(4-methyl-1H-imidazol-5-yl)methyl]piperidin-3-yl}-4H-1,2,4-triazol-3-yl)methyl]amine
1-[3-(2-ethoxyethoxy)phenyl]-2-(1H-imidazol-4-yl)-1H-imidazole
N-(2-methanesulfonylethyl)-2-(4-propanoylphenoxy)acetamide
N-[(5-cyclopropyl-1H-pyrazol-3-yl)methyl]-N'-(2-fluoro-5-methylphenyl)-N-methylbutanediamide
(2,1,3-benzothiadiazol-5-ylmethyl)(methyl){[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}amine
2-{9-[(2-chloro-5-fluorophenyl)methyl]-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl}acetamide
(3aR,7aS)-2-(3-cyclohexyl-1H-pyrazole-4-carbonyl)-2,3,3a,4,7,7a-hexahydro-1H-isoindole
(1H-indazol-3-ylmethyl)(methyl)[(5-methyl-1H-pyrazol-3-yl)methyl]amine
5-[1-(cyclohexylmethyl)-4-hydroxypiperidin-4-yl]-N-(thiophen-2-ylmethyl)-1-benzofuran-2-carboxamide
N-[(1-methyl-3-phenyl-1H-pyrazol-4-yl)methyl]-1-(pyrimidin-2-yl)piperidin-3-amine
1-(4-acetyl-4-phenylpiperidin-1-yl)-3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)propan-1-one
5-(2-ethylpiperidine-1-carbonyl)-1-[(3-methoxyphenyl)methyl]-4-oxo-N-[2-(propan-2-yloxy)ethyl]-1,4-dihydropyridine-3-carboxamide
5-(methanesulfonylmethyl)-2-(pyridin-3-yl)pyridine
2-{[4-(furan-2-yl)phenyl]methyl}-8-methyl-octahydro-1H-pyrazino[1,2-a]piperazine
N-({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)-3-(5-methyl-1H-pyrazol-1-yl)-N-(oxolan-2-ylmethyl)propanamide
(3R)-3,4,4-trimethyl-1-[1-(piperidin-4-yl)-1H-1,2,3-triazole-4-carbonyl]pyrrolidin-3-ol